Schetz JA - Search Results

1

Ring substituents on substituted benzamide ligands indirectly mediate interactions with position 7.39 of transmembrane helix 7 of the D4 dopamine receptor.

Ericksen SS, Cummings DF, Teer ME, Amdani S, Schetz JA. Ericksen SS, et al. Among authors: schetz ja. J Pharmacol Exp Ther. 2012 Aug;342(2):472-85. doi: 10.1124/jpet.112.193979. Epub 2012 May 15. J Pharmacol Exp Ther. 2012. PMID: 22588261 Free PMC article.

2

Ligand selectivity of D2 dopamine receptors is modulated by changes in local dynamics produced by sodium binding.

Ericksen SS, Cummings DF, Weinstein H, Schetz JA. Ericksen SS, et al. Among authors: schetz ja. J Pharmacol Exp Ther. 2009 Jan;328(1):40-54. doi: 10.1124/jpet.108.141531. Epub 2008 Oct 10. J Pharmacol Exp Ther. 2009. PMID: 18849360 Free PMC article.

3

Transmembrane segment five serines of the D4 dopamine receptor uniquely influence the interactions of dopamine, norepinephrine, and Ro10-4548.

Cummings DF, Ericksen SS, Goetz A, Schetz JA. Cummings DF, et al. Among authors: schetz ja. J Pharmacol Exp Ther. 2010 Jun;333(3):682-95. doi: 10.1124/jpet.109.164962. Epub 2010 Mar 9. J Pharmacol Exp Ther. 2010. PMID: 20215412 Free PMC article.

4

Three amino acids in the D2 dopamine receptor regulate selective ligand function and affinity.

Cummings DF, Ericksen SS, Schetz JA. Cummings DF, et al. Among authors: schetz ja. J Neurochem. 2009 Jul;110(1):45-57. doi: 10.1111/j.1471-4159.2009.06103.x. Epub 2009 Apr 16. J Neurochem. 2009. PMID: 19486266 Free PMC article.

5

Certain 1,4-disubstituted aromatic piperidines and piperazines with extreme selectivity for the dopamine D4 receptor interact with a common receptor microdomain.

Kortagere S, Gmeiner P, Weinstein H, Schetz JA. Kortagere S, et al. Among authors: schetz ja. Mol Pharmacol. 2004 Dec;66(6):1491-9. doi: 10.1124/mol.104.001321. Epub 2004 Sep 24. Mol Pharmacol. 2004. PMID: 15448188

6

Synthesis and structure-affinity relationships of novel small molecule natural product derivatives capable of discriminating between serotonin 5-HT1A, 5-HT2A, 5-HT2C receptor subtypes.

Cummings DF, Canseco DC, Sheth P, Johnson JE, Schetz JA. Cummings DF, et al. Among authors: schetz ja. Bioorg Med Chem. 2010 Jul 1;18(13):4783-92. doi: 10.1016/j.bmc.2010.05.017. Epub 2010 May 15. Bioorg Med Chem. 2010. PMID: 20570529 Free PMC article.

7

The binding-site crevice of the D4 dopamine receptor is coupled to three distinct sites of allosteric modulation.

Schetz JA, Sibley DR. Schetz JA, et al. J Pharmacol Exp Ther. 2001 Feb;296(2):359-63. J Pharmacol Exp Ther. 2001. PMID: 11160618

8

Molecular mechanisms of serotonergic action of the HIV-1 antiretroviral efavirenz.

Dalwadi DA, Kim S, Amdani SM, Chen Z, Huang RQ, Schetz JA. Dalwadi DA, et al. Among authors: schetz ja. Pharmacol Res. 2016 Aug;110:10-24. doi: 10.1016/j.phrs.2016.04.028. Epub 2016 May 6. Pharmacol Res. 2016. PMID: 27157251 Free PMC article.

9

Zinc modulates antagonist interactions with D2-like dopamine receptors through distinct molecular mechanisms.

Schetz JA, Chu A, Sibley DR. Schetz JA, et al. J Pharmacol Exp Ther. 1999 May;289(2):956-64. J Pharmacol Exp Ther. 1999. PMID: 10215675

10

An unambiguous assay for the cloned human sigma1 receptor reveals high affinity interactions with dopamine D4 receptor selective compounds and a distinct structure-affinity relationship for butyrophenones.

Lee IT, Chen S, Schetz JA. Lee IT, et al. Among authors: schetz ja. Eur J Pharmacol. 2008 Jan 14;578(2-3):123-36. doi: 10.1016/j.ejphar.2007.09.020. Epub 2007 Oct 2. Eur J Pharmacol. 2008. PMID: 17961544 Free PMC article.

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