Escale R - Search Results

1

Evaluation of bis-alkylamidoxime O-alkylsulfonates as orally available antimalarials.

Degardin M, Wein S, Gouni S, Tran Van Ba C, Duckert JF, Durand T, Escale R, Vial H, Vo-Hoang Y. Degardin M, et al. Among authors: escale r. ChemMedChem. 2012 Jun;7(6):991-1001. doi: 10.1002/cmdc.201200112. Epub 2012 Apr 27. ChemMedChem. 2012. PMID: 22544438

2

Design and synthesis of amidoxime derivatives for orally potent C-alkylamidine-based antimalarial agents.

Ouattara M, Wein S, Denoyelle S, Ortial S, Durand T, Escale R, Vial H, Vo-Hoang Y. Ouattara M, et al. Among authors: escale r. Bioorg Med Chem Lett. 2009 Feb 1;19(3):624-6. doi: 10.1016/j.bmcl.2008.12.058. Epub 2008 Dec 24. Bioorg Med Chem Lett. 2009. PMID: 19124242

3

N-substituted bis-C-alkyloxadiazolones as dual effectors: efficient intermediates to amidoximes or amidines and prodrug candidates of potent antimalarials.

Degardin M, Wein S, Durand T, Escale R, Vial H, Vo-Hoang Y. Degardin M, et al. Among authors: escale r. Bioorg Med Chem Lett. 2009 Sep 1;19(17):5233-6. doi: 10.1016/j.bmcl.2009.07.001. Epub 2009 Jul 4. Bioorg Med Chem Lett. 2009. PMID: 19643611

4

Synthesis and evaluation of hybrid bis-cationic salts as antimalarial drugs.

Ortial S, Denoyelle S, Wein S, Berger O, Durand T, Escale R, Pellet A, Vial H, Vo-Hoang Y. Ortial S, et al. Among authors: escale r. ChemMedChem. 2010 Jan;5(1):52-5. doi: 10.1002/cmdc.200900427. ChemMedChem. 2010. PMID: 19943278 No abstract available.

5

Reverse-benzamidine antimalarial agents: design, synthesis, and biological evaluation.

Berger O, Wein S, Duckert JF, Maynadier M, El Fangour S, Escale R, Durand T, Vial H, Vo-Hoang Y. Berger O, et al. Among authors: escale r. Bioorg Med Chem Lett. 2010 Oct 1;20(19):5815-7. doi: 10.1016/j.bmcl.2010.07.124. Epub 2010 Aug 3. Bioorg Med Chem Lett. 2010. PMID: 20800484

6

Development of the first oral bioprecursors of bis-alkylguanidine antimalarial drugs.

Degardin M, Wein S, Duckert JF, Maynadier M, Guy A, Durand T, Escale R, Vial H, Vo-Hoang Y. Degardin M, et al. Among authors: escale r. ChemMedChem. 2014 Feb;9(2):300-4. doi: 10.1002/cmdc.201300419. Epub 2014 Jan 8. ChemMedChem. 2014. PMID: 24403182

7

Evaluation of amidoxime derivatives as prodrug candidates of potent bis-cationic antimalarials.

Berger O, Ortial S, Wein S, Denoyelle S, Bressolle F, Durand T, Escale R, Vial HJ, Vo-Hoang Y. Berger O, et al. Among authors: escale r. Bioorg Med Chem Lett. 2019 Aug 15;29(16):2203-2207. doi: 10.1016/j.bmcl.2019.06.045. Epub 2019 Jun 24. Bioorg Med Chem Lett. 2019. PMID: 31255483

8

Synthesis and antimalarial activity of new 1,12-bis(N,N'-acetamidinyl)dodecane derivatives.

Ouattara M, Wein S, Calas M, Hoang YV, Vial H, Escale R. Ouattara M, et al. Among authors: escale r. Bioorg Med Chem Lett. 2007 Feb 1;17(3):593-6. doi: 10.1016/j.bmcl.2006.11.013. Epub 2006 Nov 10. Bioorg Med Chem Lett. 2007. PMID: 17123818

9

Pharmacokinetic properties and metabolism of a new potent antimalarial N-alkylamidine compound, M64, and its corresponding bioprecursors.

Margout D, Gattacceca F, Moarbess G, Wein S, Tran van Ba C, Le Pape S, Berger O, Escale R, Vial HJ, Bressolle FM. Margout D, et al. Among authors: escale r. Eur J Pharm Sci. 2011 Jan 18;42(1-2):81-90. doi: 10.1016/j.ejps.2010.10.012. Epub 2010 Nov 2. Eur J Pharm Sci. 2011. PMID: 21050886

10

Potent antimalarial activity of 2-aminopyridinium salts, amidines, and guanidines.

Calas M, Ouattara M, Piquet G, Ziora Z, Bordat Y, Ancelin ML, Escale R, Vial H. Calas M, et al. Among authors: escale r. J Med Chem. 2007 Dec 13;50(25):6307-15. doi: 10.1021/jm0704752. Epub 2007 Nov 16. J Med Chem. 2007. PMID: 18004799

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