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Page 1
Lead optimization of 2-(piperidin-3-yl)-1H-benzimidazoles: identification of 2-morpholin- and 2-thiomorpholin-2-yl-1H-benzimidazoles as selective and CNS penetrating H₁-antihistamines for insomnia.
Ravula SB, Yu J, Tran JA, Arellano M, Tucci FC, Moree WJ, Li BF, Petroski RE, Wen J, Malany S, Hoare SR, Madan A, Crowe PD, Beaton G. Ravula SB, et al. Among authors: arellano m. Bioorg Med Chem Lett. 2012 Jan 1;22(1):421-6. doi: 10.1016/j.bmcl.2011.10.115. Epub 2011 Nov 15. Bioorg Med Chem Lett. 2012. PMID: 22153347
Arylpropionylpiperazines as antagonists of the human melanocortin-4 receptor.
Jiang W, Tucci FC, Chen CW, Arellano M, Tran JA, White NS, Marinkovic D, Pontillo J, Fleck BA, Wen J, Saunders J, Madan A, Foster AC, Chen C. Jiang W, et al. Among authors: arellano m. Bioorg Med Chem Lett. 2006 Sep 1;16(17):4674-8. doi: 10.1016/j.bmcl.2006.05.088. Epub 2006 Jun 13. Bioorg Med Chem Lett. 2006. PMID: 16777413
Propionylpiperazines as human melanocortin-4 receptor ligands.
Chen CW, Tran JA, Jiang W, Tucci FC, Arellano M, Wen J, Fleck BA, Marinkovic D, White NS, Pontillo J, Saunders J, Madan A, Foster AC, Chen C. Chen CW, et al. Among authors: arellano m. Bioorg Med Chem Lett. 2006 Sep 15;16(18):4800-3. doi: 10.1016/j.bmcl.2006.06.075. Epub 2006 Jul 7. Bioorg Med Chem Lett. 2006. PMID: 16824757
Pyrrolidinones as potent functional antagonists of the human melanocortin-4 receptor.
Jiang W, Tucci FC, Tran JA, Fleck BA, Wen J, Markison S, Marinkovic D, Chen CW, Arellano M, Hoare SR, Johns M, Foster AC, Saunders J, Chen C. Jiang W, et al. Among authors: arellano m. Bioorg Med Chem Lett. 2007 Oct 15;17(20):5610-3. doi: 10.1016/j.bmcl.2007.07.097. Epub 2007 Aug 23. Bioorg Med Chem Lett. 2007. PMID: 17822895
Identification and characterization of pyrrolidine diastereoisomers as potent functional agonists and antagonists of the human melanocortin-4 receptor.
Chen C, Jiang W, Tran JA, Tucci FC, Fleck BA, Markison S, Wen J, Madan A, Hoare SR, Foster AC, Marinkovic D, Chen CW, Arellano M, Saunders J. Chen C, et al. Among authors: arellano m. Bioorg Med Chem Lett. 2008 Jan 1;18(1):129-36. doi: 10.1016/j.bmcl.2007.10.115. Epub 2007 Nov 4. Bioorg Med Chem Lett. 2008. PMID: 18032040
Structure-activity relationships of piperazinebenzylamines as potent and selective agonists of the human melanocortin-4 receptor.
Pontillo J, Tran JA, Arellano M, Fleck BA, Huntley R, Marinkovic D, Lanier M, Nelson J, Parker J, Saunders J, Tucci FC, Jiang W, Chen CW, White NS, Foster AC, Chen C. Pontillo J, et al. Among authors: arellano m. Bioorg Med Chem Lett. 2004 Sep 6;14(17):4417-23. doi: 10.1016/j.bmcl.2004.06.059. Bioorg Med Chem Lett. 2004. PMID: 15357964
306 results