Stevens RC - Search Results

1

Crystal structure-based virtual screening for fragment-like ligands of the human histamine H(1) receptor.

de Graaf C, Kooistra AJ, Vischer HF, Katritch V, Kuijer M, Shiroishi M, Iwata S, Shimamura T, Stevens RC, de Esch IJ, Leurs R. de Graaf C, et al. Among authors: stevens rc. J Med Chem. 2011 Dec 8;54(23):8195-206. doi: 10.1021/jm2011589. Epub 2011 Nov 7. J Med Chem. 2011. PMID: 22007643 Free PMC article.

2

Structure-based discovery of novel chemotypes for adenosine A(2A) receptor antagonists.

Katritch V, Jaakola VP, Lane JR, Lin J, Ijzerman AP, Yeager M, Kufareva I, Stevens RC, Abagyan R. Katritch V, et al. Among authors: stevens rc. J Med Chem. 2010 Feb 25;53(4):1799-809. doi: 10.1021/jm901647p. J Med Chem. 2010. PMID: 20095623 Free PMC article.

3

Structure of the human histamine H1 receptor complex with doxepin.

Shimamura T, Shiroishi M, Weyand S, Tsujimoto H, Winter G, Katritch V, Abagyan R, Cherezov V, Liu W, Han GW, Kobayashi T, Stevens RC, Iwata S. Shimamura T, et al. Among authors: stevens rc. Nature. 2011 Jun 22;475(7354):65-70. doi: 10.1038/nature10236. Nature. 2011. PMID: 21697825 Free PMC article.

4

Evaluation of molecular modeling of agonist binding in light of the crystallographic structure of an agonist-bound A₂A adenosine receptor.

Deflorian F, Kumar TS, Phan K, Gao ZG, Xu F, Wu H, Katritch V, Stevens RC, Jacobson KA. Deflorian F, et al. Among authors: stevens rc. J Med Chem. 2012 Jan 12;55(1):538-52. doi: 10.1021/jm201461q. Epub 2011 Dec 12. J Med Chem. 2012. PMID: 22104008 Free PMC article.

5

Optimization of adenosine 5'-carboxamide derivatives as adenosine receptor agonists using structure-based ligand design and fragment screening.

Tosh DK, Phan K, Gao ZG, Gakh AA, Xu F, Deflorian F, Abagyan R, Stevens RC, Jacobson KA, Katritch V. Tosh DK, et al. Among authors: stevens rc. J Med Chem. 2012 May 10;55(9):4297-308. doi: 10.1021/jm300095s. Epub 2012 Apr 30. J Med Chem. 2012. PMID: 22486652 Free PMC article.

6

Structure-function of the G protein-coupled receptor superfamily.

Katritch V, Cherezov V, Stevens RC. Katritch V, et al. Among authors: stevens rc. Annu Rev Pharmacol Toxicol. 2013;53:531-56. doi: 10.1146/annurev-pharmtox-032112-135923. Epub 2012 Nov 8. Annu Rev Pharmacol Toxicol. 2013. PMID: 23140243 Free PMC article. Review.

7

Structure-Based Discovery of New Antagonist and Biased Agonist Chemotypes for the Kappa Opioid Receptor.

Zheng Z, Huang XP, Mangano TJ, Zou R, Chen X, Zaidi SA, Roth BL, Stevens RC, Katritch V. Zheng Z, et al. Among authors: stevens rc. J Med Chem. 2017 Apr 13;60(7):3070-3081. doi: 10.1021/acs.jmedchem.7b00109. Epub 2017 Apr 3. J Med Chem. 2017. PMID: 28339199 Free PMC article.

8

Structure and Function of Peptide-Binding G Protein-Coupled Receptors.

Wu F, Song G, de Graaf C, Stevens RC. Wu F, et al. Among authors: stevens rc. J Mol Biol. 2017 Aug 18;429(17):2726-2745. doi: 10.1016/j.jmb.2017.06.022. Epub 2017 Jul 11. J Mol Biol. 2017. PMID: 28705763 Review.

9

Chemical Diversity in the G Protein-Coupled Receptor Superfamily.

Vass M, Kooistra AJ, Yang D, Stevens RC, Wang MW, de Graaf C. Vass M, et al. Among authors: stevens rc. Trends Pharmacol Sci. 2018 May;39(5):494-512. doi: 10.1016/j.tips.2018.02.004. Epub 2018 Mar 22. Trends Pharmacol Sci. 2018. PMID: 29576399 Review.

10

Diversity and modularity of G protein-coupled receptor structures.

Katritch V, Cherezov V, Stevens RC. Katritch V, et al. Among authors: stevens rc. Trends Pharmacol Sci. 2012 Jan;33(1):17-27. doi: 10.1016/j.tips.2011.09.003. Epub 2011 Oct 25. Trends Pharmacol Sci. 2012. PMID: 22032986 Free PMC article. Review.

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