Böcskei Z - Search Results

1

Structure-based design and optimization of potent renin inhibitors on 5- or 7-azaindole-scaffolds.

Matter H, Scheiper B, Steinhagen H, Böcskei Z, Fleury V, McCort G. Matter H, et al. Among authors: bocskei z. Bioorg Med Chem Lett. 2011 Sep 15;21(18):5487-92. doi: 10.1016/j.bmcl.2011.06.112. Epub 2011 Jul 2. Bioorg Med Chem Lett. 2011. PMID: 21840215

2

Structure-based optimization of potent 4- and 6-azaindole-3-carboxamides as renin inhibitors.

Scheiper B, Matter H, Steinhagen H, Böcskei Z, Fleury V, McCort G. Scheiper B, et al. Among authors: bocskei z. Bioorg Med Chem Lett. 2011 Sep 15;21(18):5480-6. doi: 10.1016/j.bmcl.2011.06.114. Epub 2011 Jul 6. Bioorg Med Chem Lett. 2011. PMID: 21840218

3

Discovery and optimization of a new class of potent and non-chiral indole-3-carboxamide-based renin inhibitors.

Scheiper B, Matter H, Steinhagen H, Stilz U, Böcskei Z, Fleury V, McCort G. Scheiper B, et al. Among authors: bocskei z. Bioorg Med Chem Lett. 2010 Nov 1;20(21):6268-72. doi: 10.1016/j.bmcl.2010.08.092. Epub 2010 Aug 21. Bioorg Med Chem Lett. 2010. PMID: 20850300

4

5-Chlorothiophene-2-carboxylic acid [(S)-2-[2-methyl-3-(2-oxopyrrolidin-1-yl)benzenesulfonylamino]-3-(4-methylpiperazin-1-yl)-3-oxopropyl]amide (SAR107375), a selective and potent orally active dual thrombin and factor Xa inhibitor.

Meneyrol J, Follmann M, Lassalle G, Wehner V, Barre G, Rousseaux T, Altenburger JM, Petit F, Bocskei Z, Schreuder H, Alet N, Herault JP, Millet L, Dol F, Florian P, Schaeffer P, Sadoun F, Klieber S, Briot C, Bono F, Herbert JM. Meneyrol J, et al. Among authors: bocskei z. J Med Chem. 2013 Dec 12;56(23):9441-56. doi: 10.1021/jm4005835. Epub 2013 Dec 3. J Med Chem. 2013. PMID: 24175584

5

SSR182289A, a selective and potent orally active thrombin inhibitor.

Altenburger JM, Lassalle GY, Matrougui M, Galtier D, Jetha JC, Bocskei Z, Berry CN, Lunven C, Lorrain J, Herault JP, Schaeffer P, O'Connor SE, Herbert JM. Altenburger JM, et al. Among authors: bocskei z. Bioorg Med Chem. 2004 Apr 1;12(7):1713-30. doi: 10.1016/j.bmc.2004.01.016. Bioorg Med Chem. 2004. PMID: 15028263

6

Human prorenin structure sheds light on a novel mechanism of its autoinhibition and on its non-proteolytic activation by the (pro)renin receptor.

Morales R, Watier Y, Böcskei Z. Morales R, et al. Among authors: bocskei z. J Mol Biol. 2012 Aug 3;421(1):100-11. doi: 10.1016/j.jmb.2012.05.003. Epub 2012 May 7. J Mol Biol. 2012. PMID: 22575890

7

Prolyl oligopeptidase inhibition by N-acyl-pro-pyrrolidine-type molecules.

Kánai K, Arányi P, Böcskei Z, Ferenczy G, Harmat V, Simon K, Bátori S, Náray-Szabo G, Hermecz I. Kánai K, et al. Among authors: bocskei z. J Med Chem. 2008 Dec 11;51(23):7514-22. doi: 10.1021/jm800944x. J Med Chem. 2008. PMID: 19006380

8

Ipriflavone, an antiostheophorotic agent.

Böcskei Z, Simon K, Varga M, Hermecz I. Böcskei Z, et al. Acta Crystallogr C. 1996 Apr 15;52 ( Pt 4):1022-4. doi: 10.1107/s0108270195015241. Acta Crystallogr C. 1996. PMID: 8624237

9

A new potent calmodulin antagonist with arylalkylamine structure: crystallographic, spectroscopic and functional studies.

Harmat V, Böcskei Z, Náray-Szabó G, Bata I, Csutor AS, Hermecz I, Arányi P, Szabó B, Liliom K, Vértessy BG, Ovádi J. Harmat V, et al. Among authors: bocskei z. J Mol Biol. 2000 Mar 31;297(3):747-55. doi: 10.1006/jmbi.2000.3607. J Mol Biol. 2000. PMID: 10731425

10

Crystallization and preliminary X-ray analysis of porcine muscle prolyl oligopeptidase.

Böcskei Z, Fuxreiter M, Náray-Szabó G, Szabó E, Polgár L. Böcskei Z, et al. Acta Crystallogr D Biol Crystallogr. 1998 Nov 1;54(Pt 6 Pt 2):1414-5. doi: 10.1107/s0907444998004181. Acta Crystallogr D Biol Crystallogr. 1998. PMID: 10089523

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