Simons C - Search Results

1

Synthesis and biological evaluation of 3-(1H-imidazol- and triazol-1-yl)-2,2-dimethyl-3-[4-(naphthalen-2-ylamino)phenyl]propyl derivatives as small molecule inhibitors of retinoic acid 4-hydroxylase (CYP26).

Gomaa MS, Bridgens CE, Veal GJ, Redfern CP, Brancale A, Armstrong JL, Simons C. Gomaa MS, et al. Among authors: simons c. J Med Chem. 2011 Oct 13;54(19):6803-11. doi: 10.1021/jm200695m. Epub 2011 Sep 8. J Med Chem. 2011. PMID: 21838328

2

Synthesis and biological evaluation of novel 2-deoxy-4-thio-imidazole nucleosides.

Wang Y, Inguaggiato G, Jasamai M, Shah M, Hughes D, Slater M, Simons C. Wang Y, et al. Among authors: simons c. Bioorg Med Chem. 1999 Mar;7(3):481-7. doi: 10.1016/s0968-0896(98)00255-7. Bioorg Med Chem. 1999. PMID: 10220034

3

1-[(Benzofuran-2-yl)phenylmethyl]-triazoles and -tetrazoles - potent competitive inhibitors of aromatase.

Vinh TK, Ahmadi M, Delgado PO, Perez SF, Walters HM, Smith HJ, Nicholls PJ, Simons C. Vinh TK, et al. Among authors: simons c. Bioorg Med Chem Lett. 1999 Jul 19;9(14):2105-8. doi: 10.1016/s0960-894x(99)00328-5. Bioorg Med Chem Lett. 1999. PMID: 10450990

4

1-[(Benzofuran-2-yl)phenylmethyl]triazoles as steroidogenic inhibitors: synthesis and in vitro inhibition of human placental CYP19 aromatase.

Vinh TK, Yee SW, Kirby AJ, Nicholls PJ, Simons C. Vinh TK, et al. Among authors: simons c. Anticancer Drug Des. 2001 Aug-Oct;16(4-5):217-25. Anticancer Drug Des. 2001. PMID: 12049480

5

Some coumarins and triphenylethene derivatives as inhibitors of human testes microsomal 17beta-hydroxysteroid dehydrogenase (17beta-HSD type 3): further studies with tamoxifen on the rat testes microsomal enzyme.

LE Lain R, Barrell KJ, Saeed GS, Nicholls PJ, Simons C, Kirby A, Smith HJ. LE Lain R, et al. Among authors: simons c. J Enzyme Inhib Med Chem. 2002 Apr;17(2):93-100. doi: 10.1080/14756360290026441. J Enzyme Inhib Med Chem. 2002. PMID: 12420755 Free article.

6

Solid-phase synthesis of diamine and polyamine amino acid derivatives as HIV-1 tat-TAR binding inhibitors.

Jimenez Bueno G, Klimkait T, Gilbert IH, Simons C. Jimenez Bueno G, et al. Among authors: simons c. Bioorg Med Chem. 2003 Jan 2;11(1):87-94. doi: 10.1016/s0968-0896(02)00305-x. Bioorg Med Chem. 2003. PMID: 12467711

7

Some 3-(4-aminophenyl)pyrrolidine-2,5-diones as all-trans-retinoic acid metabolising enzyme inhibitors (RAMBAs).

Kirby AJ, Lelain R, Mason P, Maharlouie F, Nicholls PJ, Smith HJ, Simons C. Kirby AJ, et al. Among authors: simons c. J Enzyme Inhib Med Chem. 2002 Oct;17(5):321-7. doi: 10.1080/1475636021000059100. J Enzyme Inhib Med Chem. 2002. PMID: 12683748 Free article.

8

Inhibition of retinoic acid metabolising enzymes by 2-(4-aminophenylmethyl)-6-hydroxy-3,4-dihydronaphthalen-1(2H)-one and related compounds.

Kirby AJ, Le Lain R, Maharlouie F, Mason P, Nicholls PJ, Smith HJ, Simons C. Kirby AJ, et al. Among authors: simons c. J Enzyme Inhib Med Chem. 2003 Feb;18(1):27-33. doi: 10.1080/1475636021000049221. J Enzyme Inhib Med Chem. 2003. PMID: 12751817 Free article.

9

Some 1,2-diphenylethane derivatives as inhibitors of retinoic acid--metabolising enzymes.

Greer VP, Mason P, Kirby AJ, Smith HJ, Nicholls PJ, Simons C. Greer VP, et al. Among authors: simons c. J Enzyme Inhib Med Chem. 2003 Oct;18(5):431-43. doi: 10.1080/1475636031000155427. J Enzyme Inhib Med Chem. 2003. PMID: 14692511 Free article.

10

Some aryl substituted 2-(4-nitrophenyl)-4-oxo-4-phenylbutanoates and 3-(4-nitrophenyl)-1-phenyl-1,4-butanediols and related compounds as inhibitors of rat liver microsomal retinoic acid metabolising enzymes.

Mason P, Greer VP, Kirby AJ, Simons C, Nicholls PJ, Smith HJ. Mason P, et al. Among authors: simons c. J Enzyme Inhib Med Chem. 2003 Dec;18(6):511-28. doi: 10.1080/1475636032000141881. J Enzyme Inhib Med Chem. 2003. PMID: 15008516 Free article.

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