Filacchioni G - Search Results

1

Tricyclic heteroaromatic systems. [1]benzopyranopyrrol-4-ones and [1]benzopyrano-1,2,3-triazol-4-ones as benzodiazepine receptor ligands. Synthesis and structure-activity relationships.

Colotta V, Cecchi L, Melani F, Filacchioni G, Martini C, Giannaccini G, Lucacchini A. Colotta V, et al. Among authors: filacchioni g. J Med Chem. 1990 Sep;33(9):2646-51. doi: 10.1021/jm00171a047. J Med Chem. 1990. PMID: 2167984

2

Synthesis and structure-activity relationships of a new set of 1,2,4-triazolo[4,3-a]quinoxalin-1-one derivatives as adenosine receptor antagonists.

Colotta V, Catarzi D, Varano F, Filacchioni G, Martini C, Trincavelli L, Lucacchini A. Colotta V, et al. Among authors: filacchioni g. Bioorg Med Chem. 2003 Aug 5;11(16):3541-50. doi: 10.1016/s0968-0896(03)00338-9. Bioorg Med Chem. 2003. PMID: 12878146

3

Synthesis of 4-amino-6-(hetero)arylalkylamino-1,2,4-triazolo[4,3-a]quinoxalin-1-one derivatives as potent A(2A) adenosine receptor antagonists.

Colotta V, Catarzi D, Varano F, Filacchioni G, Martini C, Trincavelli L, Lucacchini A. Colotta V, et al. Among authors: filacchioni g. Bioorg Med Chem. 2003 Dec 1;11(24):5509-18. doi: 10.1016/j.bmc.2003.09.019. Bioorg Med Chem. 2003. PMID: 14642595

4

Synthesis and biological evaluation of analogues of 7-chloro-4,5-dihydro-4- oxo-8-(1,2,4-triazol-4-yl)-1,2,4-triazolo[1,5-a]quinoxaline-2-carboxylic acid (TQX-173) as novel selective AMPA receptor antagonists.

Catarzi D, Colotta V, Varano F, Calabri FR, Filacchioni G, Galli A, Costagli C, Carlà V. Catarzi D, et al. Among authors: filacchioni g. J Med Chem. 2004 Jan 1;47(1):262-72. doi: 10.1021/jm030906q. J Med Chem. 2004. PMID: 14695840

5

1,2,4-triazolo[4,3-a]quinoxalin-1-one moiety as an attractive scaffold to develop new potent and selective human A3 adenosine receptor antagonists: synthesis, pharmacological, and ligand-receptor modeling studies.

Colotta V, Catarzi D, Varano F, Calabri FR, Lenzi O, Filacchioni G, Martini C, Trincavelli L, Deflorian F, Moro S. Colotta V, et al. Among authors: filacchioni g. J Med Chem. 2004 Jul 1;47(14):3580-90. doi: 10.1021/jm031136l. J Med Chem. 2004. PMID: 15214785

6

2-aryl-8-chloro-1,2,4-triazolo[1,5-a]quinoxalin-4-amines as highly potent A1 and A3 adenosine receptor antagonists.

Catarzi D, Colotta V, Varano F, Calabri FR, Lenzi O, Filacchioni G, Trincavelli L, Martini C, Tralli A, Montopoli C, Moro S. Catarzi D, et al. Among authors: filacchioni g. Bioorg Med Chem. 2005 Feb 1;13(3):705-15. doi: 10.1016/j.bmc.2004.10.050. Bioorg Med Chem. 2005. PMID: 15653338

7

1,2,4-Triazolo[1,5-a]quinoxaline as a versatile tool for the design of selective human A3 adenosine receptor antagonists: synthesis, biological evaluation, and molecular modeling studies of 2-(hetero)aryl- and 2-carboxy-substituted derivatives.

Catarzi D, Colotta V, Varano F, Lenzi O, Filacchioni G, Trincavelli L, Martini C, Montopoli C, Moro S. Catarzi D, et al. Among authors: filacchioni g. J Med Chem. 2005 Dec 15;48(25):7932-45. doi: 10.1021/jm0504149. J Med Chem. 2005. PMID: 16335918

8

4-amido-2-aryl-1,2,4-triazolo[4,3-a]quinoxalin-1-ones as new potent and selective human A3 adenosine receptor antagonists. synthesis, pharmacological evaluation, and ligand-receptor modeling studies.

Lenzi O, Colotta V, Catarzi D, Varano F, Filacchioni G, Martini C, Trincavelli L, Ciampi O, Varani K, Marighetti F, Morizzo E, Moro S. Lenzi O, et al. Among authors: filacchioni g. J Med Chem. 2006 Jun 29;49(13):3916-25. doi: 10.1021/jm060373w. J Med Chem. 2006. PMID: 16789747

9

Tricyclic heteroaromatic systems. Synthesis and A1 and A2a adenosine binding activities of some 1-aryl-1,4-dihydro-3-methyl[1]benzopyrano[2,3-c] pyrazol-4-ones, 1-aryl-4,9-dihydro-3-methyl-1H-pyrazolo[3,4-b]quinolin-4- ones, and 1-aryl-1H-imidazo[4,5-b]quinoxalines.

Catarzi D, Cecchi L, Colotta V, Filacchioni G, Martini C, Tacchi P, Lucacchini A. Catarzi D, et al. Among authors: filacchioni g. J Med Chem. 1995 Apr 14;38(8):1330-6. doi: 10.1021/jm00008a011. J Med Chem. 1995. PMID: 7731018

10

Synthesis of some 2-aryl-1,2,4-triazolo[1,5-c][1,3]benzoxazin-5-ones as tools to define the essential pharmacophoric descriptors of a benzodiazepine receptor ligand.

Catarzi D, Cecchi L, Colotta V, Filacchioni G, Varano F, Martini C, Giousti L, Lucacchini A. Catarzi D, et al. Among authors: filacchioni g. J Med Chem. 1995 Jun 9;38(12):2196-201. doi: 10.1021/jm00012a020. J Med Chem. 1995. PMID: 7783151

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