Rizzo G - Search Results

1

Extending SAR of bile acids as FXR ligands: discovery of 23-N-(carbocinnamyloxy)-3α,7α-dihydroxy-6α-ethyl-24-nor-5β-cholan-23-amine.

Gioiello A, Macchiarulo A, Carotti A, Filipponi P, Costantino G, Rizzo G, Adorini L, Pellicciari R. Gioiello A, et al. Among authors: rizzo g. Bioorg Med Chem. 2011 Apr 15;19(8):2650-8. doi: 10.1016/j.bmc.2011.03.004. Epub 2011 Mar 10. Bioorg Med Chem. 2011. PMID: 21459580

2

Back door modulation of the farnesoid X receptor: design, synthesis, and biological evaluation of a series of side chain modified chenodeoxycholic acid derivatives.

Pellicciari R, Gioiello A, Costantino G, Sadeghpour BM, Rizzo G, Meyer U, Parks DJ, Entrena-Guadix A, Fiorucci S. Pellicciari R, et al. Among authors: rizzo g. J Med Chem. 2006 Jul 13;49(14):4208-15. doi: 10.1021/jm060294k. J Med Chem. 2006. PMID: 16821780

3

Pyrazole[3,4-e][1,4]thiazepin-7-one derivatives as a novel class of Farnesoid X Receptor (FXR) agonists.

Marinozzi M, Carotti A, Sansone E, Macchiarulo A, Rosatelli E, Sardella R, Natalini B, Rizzo G, Adorini L, Passeri D, De Franco F, Pruzanski M, Pellicciari R. Marinozzi M, et al. Among authors: rizzo g. Bioorg Med Chem. 2012 Jun 1;20(11):3429-45. doi: 10.1016/j.bmc.2012.04.021. Epub 2012 Apr 20. Bioorg Med Chem. 2012. PMID: 22564381

4

Asymmetric synthesis of the four diastereoisomers of a novel non-steroidal farnesoid X receptor (FXR) agonist: role of the chirality on the biological activity.

Marinozzi M, Carotti A, Sardella R, Buonerba F, Ianni F, Natalini B, Passeri D, Rizzo G, Pellicciari R. Marinozzi M, et al. Among authors: rizzo g. Bioorg Med Chem. 2013 Jul 1;21(13):3780-9. doi: 10.1016/j.bmc.2013.04.038. Epub 2013 Apr 23. Bioorg Med Chem. 2013. PMID: 23684233

5

Role of FXR in regulating bile acid homeostasis and relevance for human diseases.

Rizzo G, Renga B, Mencarelli A, Pellicciari R, Fiorucci S. Rizzo G, et al. Curr Drug Targets Immune Endocr Metabol Disord. 2005 Sep;5(3):289-303. doi: 10.2174/1568008054863781. Curr Drug Targets Immune Endocr Metabol Disord. 2005. PMID: 16178789 Review.

6

Unveiling hidden features of orphan nuclear receptors: the case of the small heterodimer partner (SHP).

Macchiarulo A, Rizzo G, Costantino G, Fiorucci S, Pellicciari R. Macchiarulo A, et al. Among authors: rizzo g. J Mol Graph Model. 2006 Mar;24(5):362-72. doi: 10.1016/j.jmgm.2005.09.016. Epub 2005 Nov 9. J Mol Graph Model. 2006. PMID: 16288980

7

Avicholic Acid: A Lead Compound from Birds on the Route to Potent TGR5 Modulators.

Pellicciari R, Gioiello A, Sabbatini P, Venturoni F, Nuti R, Colliva C, Rizzo G, Adorini L, Pruzanski M, Roda A, Macchiarulo A. Pellicciari R, et al. Among authors: rizzo g. ACS Med Chem Lett. 2012 Feb 6;3(4):273-7. doi: 10.1021/ml200256d. eCollection 2012 Apr 12. ACS Med Chem Lett. 2012. PMID: 24900463 Free PMC article.

8

The farnesoid X receptor promotes adipocyte differentiation and regulates adipose cell function in vivo.

Rizzo G, Disante M, Mencarelli A, Renga B, Gioiello A, Pellicciari R, Fiorucci S. Rizzo G, et al. Mol Pharmacol. 2006 Oct;70(4):1164-73. doi: 10.1124/mol.106.023820. Epub 2006 Jun 15. Mol Pharmacol. 2006. PMID: 16778009

9

Cross-talk between farnesoid-X-receptor (FXR) and peroxisome proliferator-activated receptor gamma contributes to the antifibrotic activity of FXR ligands in rodent models of liver cirrhosis.

Fiorucci S, Rizzo G, Antonelli E, Renga B, Mencarelli A, Riccardi L, Morelli A, Pruzanski M, Pellicciari R. Fiorucci S, et al. Among authors: rizzo g. J Pharmacol Exp Ther. 2005 Oct;315(1):58-68. doi: 10.1124/jpet.105.085597. Epub 2005 Jun 24. J Pharmacol Exp Ther. 2005. PMID: 15980055

10

The methyl transferase PRMT1 functions as co-activator of farnesoid X receptor (FXR)/9-cis retinoid X receptor and regulates transcription of FXR responsive genes.

Rizzo G, Renga B, Antonelli E, Passeri D, Pellicciari R, Fiorucci S. Rizzo G, et al. Mol Pharmacol. 2005 Aug;68(2):551-8. doi: 10.1124/mol.105.012104. Epub 2005 May 23. Mol Pharmacol. 2005. PMID: 15911693

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