Janssen E - Search Results

1

Fragment growing induces conformational changes in acetylcholine-binding protein: a structural and thermodynamic analysis.

Edink E, Rucktooa P, Retra K, Akdemir A, Nahar T, Zuiderveld O, van Elk R, Janssen E, van Nierop P, van Muijlwijk-Koezen J, Smit AB, Sixma TK, Leurs R, de Esch IJ. Edink E, et al. Among authors: janssen e. J Am Chem Soc. 2011 Apr 13;133(14):5363-71. doi: 10.1021/ja110571r. Epub 2011 Feb 15. J Am Chem Soc. 2011. PMID: 21322593

2

Inhibition of brain [(3)H]cimetidine binding by improgan-like antinociceptive drugs.

Stadel R, Carpenter AB, Nalwalk JW, de Esch IJ, Janssen E, Hough LB. Stadel R, et al. Among authors: janssen e. Eur J Pharmacol. 2010 Apr 25;632(1-3):33-8. doi: 10.1016/j.ejphar.2010.01.026. Epub 2010 Feb 6. Eur J Pharmacol. 2010. PMID: 20138862 Free PMC article.

3

Synthesis, modeling and functional activity of substituted styrene-amides as small-molecule CXCR7 agonists.

Wijtmans M, Maussang D, Sirci F, Scholten DJ, Canals M, Mujić-Delić A, Chong M, Chatalic KL, Custers H, Janssen E, de Graaf C, Smit MJ, de Esch IJ, Leurs R. Wijtmans M, et al. Among authors: janssen e. Eur J Med Chem. 2012 May;51:184-92. doi: 10.1016/j.ejmech.2012.02.041. Epub 2012 Feb 27. Eur J Med Chem. 2012. PMID: 22424612

4

Pharmacological Characterization and Radiolabeling of VUF15485, a High-Affinity Small-Molecule Agonist for the Atypical Chemokine Receptor ACKR3.

Zarca AM, Adlere I, Viciano CP, Arimont-Segura M, Meyrath M, Simon IA, Bebelman JP, Laan D, Custers HGJ, Janssen E, Versteegh KL, Buzink MCML, Nesheva DN, Bosma R, de Esch IJP, Vischer HF, Wijtmans M, Szpakowska M, Chevigné A, Hoffmann C, de Graaf C, Zarzycka BA, Windhorst AD, Smit MJ, Leurs R. Zarca AM, et al. Among authors: janssen e. Mol Pharmacol. 2024 Mar 14;105(4):301-312. doi: 10.1124/molpharm.123.000835. Mol Pharmacol. 2024. PMID: 38346795

5

Antinociceptive activity of chemical congeners of improgan: optimization of side chain length leads to the discovery of a new, potent, non-opioid analgesic.

Hough LB, de Esch IJ, Janssen E, Phillips J, Svokos K, Kern B, Trachler J, Abood ME, Leurs R, Nalwalk JW. Hough LB, et al. Among authors: janssen e. Neuropharmacology. 2006 Sep;51(3):447-56. doi: 10.1016/j.neuropharm.2006.04.003. Epub 2006 Jun 23. Neuropharmacology. 2006. PMID: 16806300

6

CC12, a high-affinity ligand for [3H]cimetidine binding, is an improgan antagonist.

Hough LB, Nalwalk JW, Phillips JG, Kern B, Shan Z, Wentland MP, de Esch IJ, Janssen E, Barr T, Stadel R. Hough LB, et al. Among authors: janssen e. Neuropharmacology. 2007 Apr;52(5):1244-55. doi: 10.1016/j.neuropharm.2007.01.004. Epub 2007 Jan 20. Neuropharmacology. 2007. PMID: 17336343 Free PMC article.

7

Asymmetric synthesis of synthetic alkaloids by a tandem biocatalysis/Ugi/Pictet-Spengler-type cyclization sequence.

Znabet A, Zonneveld J, Janssen E, De Kanter FJ, Helliwell M, Turner NJ, Ruijter E, Orru RV. Znabet A, et al. Among authors: janssen e. Chem Commun (Camb). 2010 Nov 7;46(41):7706-8. doi: 10.1039/c0cc02938f. Epub 2010 Sep 27. Chem Commun (Camb). 2010. PMID: 20871902

8

A highly efficient synthesis of telaprevir by strategic use of biocatalysis and multicomponent reactions.

Znabet A, Polak MM, Janssen E, de Kanter FJ, Turner NJ, Orru RV, Ruijter E. Znabet A, et al. Among authors: janssen e. Chem Commun (Camb). 2010 Nov 14;46(42):7918-20. doi: 10.1039/c0cc02823a. Epub 2010 Sep 20. Chem Commun (Camb). 2010. PMID: 20856952

9

Stereoselective synthesis of N-aryl proline amides by biotransformation-Ugi-Smiles sequence.

Znabet A, Blanken S, Janssen E, de Kanter FJ, Helliwell M, Turner NJ, Ruijter E, Orru RV. Znabet A, et al. Among authors: janssen e. Org Biomol Chem. 2012 Feb 7;10(5):941-4. doi: 10.1039/c1ob06699d. Epub 2011 Dec 19. Org Biomol Chem. 2012. PMID: 22179495

10

A multicomponent reaction towards N-(cyanomethyl)amides.

Elders N, Ruijter E, de Kanter FJ, Janssen E, Lutz M, Spek AL, Orru RV. Elders N, et al. Among authors: janssen e. Chemistry. 2009 Jun 15;15(25):6096-9. doi: 10.1002/chem.200900785. Chemistry. 2009. PMID: 19462390 No abstract available.

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

788 results

Search Page

Filters