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971 results

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Page 1
Design of potent and selective GSK3beta inhibitors with acceptable safety profile and pharmacokinetics.
Lesuisse D, Tiraboschi G, Krick A, Abecassis PY, Dutruc-Rosset G, Babin D, Halley F, Châtreau F, Lachaud S, Chevalier A, Quarteronet D, Burgevin MC, Amara C, Bertrand P, Rooney T. Lesuisse D, et al. Among authors: bertrand p. Bioorg Med Chem Lett. 2010 Apr 1;20(7):2344-9. doi: 10.1016/j.bmcl.2010.01.132. Epub 2010 Feb 2. Bioorg Med Chem Lett. 2010. PMID: 20189807
Rational design of potent GSK3beta inhibitors with selectivity for Cdk1 and Cdk2.
Lesuisse D, Dutruc-Rosset G, Tiraboschi G, Dreyer MK, Maignan S, Chevalier A, Halley F, Bertrand P, Burgevin MC, Quarteronet D, Rooney T. Lesuisse D, et al. Among authors: bertrand p. Bioorg Med Chem Lett. 2010 Mar 15;20(6):1985-9. doi: 10.1016/j.bmcl.2010.01.114. Epub 2010 Jan 25. Bioorg Med Chem Lett. 2010. PMID: 20167481
Inside HDAC with HDAC inhibitors.
Bertrand P. Bertrand P. Eur J Med Chem. 2010 Jun;45(6):2095-116. doi: 10.1016/j.ejmech.2010.02.030. Epub 2010 Feb 14. Eur J Med Chem. 2010. PMID: 20223566 Review.
Cross metathesis with hydroxamate and benzamide BOC-protected alkenes to access HDAC inhibitors and their biological evaluation highlighted intrinsic activity of BOC-protected dihydroxamates.
Zwick V, Nurisso A, Simões-Pires C, Bouchet S, Martinet N, Lehotzky A, Ovadi J, Cuendet M, Blanquart C, Bertrand P. Zwick V, et al. Among authors: bertrand p. Bioorg Med Chem Lett. 2016 Jan 1;26(1):154-9. doi: 10.1016/j.bmcl.2015.11.011. Epub 2015 Nov 11. Bioorg Med Chem Lett. 2016. PMID: 26611919
Synthesis of a selective HDAC6 inhibitor active in neuroblasts.
Zwick V, Simões-Pires CA, Nurisso A, Petit C, Dos Santos Passos C, Randazzo GM, Martinet N, Bertrand P, Cuendet M. Zwick V, et al. Among authors: bertrand p. Bioorg Med Chem Lett. 2016 Oct 15;26(20):4955-4959. doi: 10.1016/j.bmcl.2016.09.011. Epub 2016 Sep 7. Bioorg Med Chem Lett. 2016. PMID: 27650925
SAR110894, a potent histamine H3-receptor antagonist, displays disease-modifying activity in a transgenic mouse model of tauopathy.
Delay-Goyet P, Blanchard V, Schussler N, Lopez-Grancha M, Ménager J, Mary V, Sultan E, Buzy A, Guillemot JC, Stemmelin J, Bertrand P, Rooney T, Pradier L, Barnéoud P. Delay-Goyet P, et al. Among authors: bertrand p. Alzheimers Dement (N Y). 2016 Nov 3;2(4):267-280. doi: 10.1016/j.trci.2016.10.002. eCollection 2016 Nov. Alzheimers Dement (N Y). 2016. PMID: 29067314 Free PMC article.
Mitotic-like tau phosphorylation by p25-Cdk5 kinase complex.
Hamdane M, Sambo AV, Delobel P, Bégard S, Violleau A, Delacourte A, Bertrand P, Benavides J, Buée L. Hamdane M, et al. Among authors: bertrand p. J Biol Chem. 2003 Sep 5;278(36):34026-34. doi: 10.1074/jbc.M302872200. Epub 2003 Jun 24. J Biol Chem. 2003. PMID: 12826674 Free article.
Synthesis of rigid trichostatin A analogs as HDAC inhibitors.
Charrier C, Bertrand P, Gesson JP, Roche J. Charrier C, et al. Among authors: bertrand p. Bioorg Med Chem Lett. 2006 Oct 15;16(20):5339-44. doi: 10.1016/j.bmcl.2006.07.080. Epub 2006 Aug 14. Bioorg Med Chem Lett. 2006. PMID: 16904890
971 results