Holzgrabe U - Search Results

1

Interaction of (benzylidene-hydrazono)-1,4-dihydropyridines with beta-amyloid, acetylcholine, and butyrylcholine esterases.

Alptüzün V, Prinz M, Hörr V, Scheiber J, Radacki K, Fallarero A, Vuorela P, Engels B, Braunschweig H, Erciyas E, Holzgrabe U. Alptüzün V, et al. Among authors: holzgrabe u. Bioorg Med Chem. 2010 Mar 1;18(5):2049-59. doi: 10.1016/j.bmc.2010.01.002. Epub 2010 Jan 15. Bioorg Med Chem. 2010. PMID: 20149667

2

[Synthesis and stereochemistry of potentially powerful analgesics: 2,4-m-diaryl substituted 3,7-diazabicyclo(3,3,1)nonan-9-one-1,5-diesters].

Holzgrabe U, Erciyas E. Holzgrabe U, et al. Arch Pharm (Weinheim). 1992 Oct;325(10):657-63. doi: 10.1002/ardp.19923251008. Arch Pharm (Weinheim). 1992. PMID: 1334646 German.

3

Cooperative interactions at M2 muscarinic acetylcholine receptors: structure/activity relationships in stepwise shortened bispyridinium- and bis(ammonio)alkane-type allosteric modulators.

Gilsbach R, Grossmüller M, Alptüzün V, Erciyas E, Tränkle C, Holzgrabe U, Mohr K. Gilsbach R, et al. Among authors: holzgrabe u. Neurochem Res. 2003 Apr;28(3-4):667-73. doi: 10.1023/a:1022858414900. Neurochem Res. 2003. PMID: 12675159

4

Synthesis and biological activity of pyridinium-type acetylcholinesterase inhibitors.

Alptüzün V, Kapková P, Baumann K, Erciyas E, Holzgrabe U. Alptüzün V, et al. Among authors: holzgrabe u. J Pharm Pharmacol. 2003 Oct;55(10):1397-404. doi: 10.1211/0022357021855. J Pharm Pharmacol. 2003. PMID: 14607022

5

Synthesis, biological activity, and docking studies of new acetylcholinesterase inhibitors of the bispyridinium type.

Kapková P, Stiefl N, Sürig U, Engels B, Baumann K, Holzgrabe U. Kapková P, et al. Among authors: holzgrabe u. Arch Pharm (Weinheim). 2003 Nov;336(11):523-40. doi: 10.1002/ardp.200300795. Arch Pharm (Weinheim). 2003. PMID: 14639745

6

Search for dual function inhibitors for Alzheimer's disease: synthesis and biological activity of acetylcholinesterase inhibitors of pyridinium-type and their Abeta fibril formation inhibition capacity.

Kapková P, Alptüzün V, Frey P, Erciyas E, Holzgrabe U. Kapková P, et al. Among authors: holzgrabe u. Bioorg Med Chem. 2006 Jan 15;14(2):472-8. doi: 10.1016/j.bmc.2005.08.034. Epub 2005 Sep 29. Bioorg Med Chem. 2006. PMID: 16198581

Lancet Neurol.2003, 2, 539] In view of the development of new AChE inhibitors as drugs capable of reducing the symptoms of AD, the capacity of newly synthesized AChE inhibitors of pyridinium-type to inhibit the AChE was examined and compared to those of other inhibitors of this t …

Lancet Neurol.2003, 2, 539] In view of the development of new AChE inhibitors as drugs capable of reducing the symptoms of AD, the capacity …

7

Targeting acetylcholinesterase to treat neurodegeneration.

Holzgrabe U, Kapková P, Alptüzün V, Scheiber J, Kugelmann E. Holzgrabe U, et al. Expert Opin Ther Targets. 2007 Feb;11(2):161-79. doi: 10.1517/14728222.11.2.161. Expert Opin Ther Targets. 2007. PMID: 17227232 Review.

8

Pipecolic acid derivatives as small-molecule inhibitors of the Legionella MIP protein.

Juli C, Sippel M, Jäger J, Thiele A, Weiwad M, Schweimer K, Rösch P, Steinert M, Sotriffer CA, Holzgrabe U. Juli C, et al. Among authors: holzgrabe u. J Med Chem. 2011 Jan 13;54(1):277-83. doi: 10.1021/jm101156y. Epub 2010 Dec 13. J Med Chem. 2011. PMID: 21142106

9

4-[(2E)-2-(4-Chloro-benzyl-idene)hydrazinyl-idene]-1-methyl-1,4-dihydro-pyridine monohydrate.

Aydın A, Akkurt M, Alptüzün V, Büyükgüngör O, Holzgrabe U, Radacki K. Aydın A, et al. Among authors: holzgrabe u. Acta Crystallogr Sect E Struct Rep Online. 2010 May 12;66(Pt 6):o1324-5. doi: 10.1107/S1600536810015709. Acta Crystallogr Sect E Struct Rep Online. 2010. PMID: 21579416 Free PMC article.

10

Identification and characterization of diarylimidazoles as hybrid inhibitors of butyrylcholinesterase and amyloid beta fibril formation.

Karlsson D, Fallarero A, Brunhofer G, Guzik P, Prinz M, Holzgrabe U, Erker T, Vuorela P. Karlsson D, et al. Among authors: holzgrabe u. Eur J Pharm Sci. 2012 Jan 23;45(1-2):169-83. doi: 10.1016/j.ejps.2011.11.004. Epub 2011 Nov 16. Eur J Pharm Sci. 2012. PMID: 22108346

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