Rocheville M - Search Results

1

The identification of structurally novel, selective, orally bioavailable positive modulators of mGluR2.

D'Alessandro PL, Corti C, Roth A, Ugolini A, Sava A, Montanari D, Bianchi F, Garland SL, Powney B, Koppe EL, Rocheville M, Osborne G, Perez P, de la Fuente J, De Los Frailes M, Smith PW, Branch C, Nash D, Watson SP. D'Alessandro PL, et al. Among authors: rocheville m. Bioorg Med Chem Lett. 2010 Jan 15;20(2):759-62. doi: 10.1016/j.bmcl.2009.11.032. Epub 2009 Nov 26. Bioorg Med Chem Lett. 2010. PMID: 20005096

2

In vitro and in vivo characterization of the novel GABAB receptor positive allosteric modulator, 2-{1-[2-(4-chlorophenyl)-5-methylpyrazolo[1,5-a]pyrimidin-7-yl]-2-piperidinyl}ethanol (CMPPE).

Perdona' E, Costantini VJ, Tessari M, Martinelli P, Carignani C, Valerio E, Mok MH, Zonzini L, Visentini F, Gianotti M, Gordon L, Rocheville M, Corsi M, Capelli AM. Perdona' E, et al. Among authors: rocheville m. Neuropharmacology. 2011 Oct-Nov;61(5-6):957-66. doi: 10.1016/j.neuropharm.2011.06.024. Epub 2011 Jul 5. Neuropharmacology. 2011. PMID: 21756923

3

Evaluation of the mGlu8 receptor as a putative therapeutic target in schizophrenia.

Robbins MJ, Starr KR, Honey A, Soffin EM, Rourke C, Jones GA, Kelly FM, Strum J, Melarange RA, Harris AJ, Rocheville M, Rupniak T, Murdock PR, Jones DN, Kew JN, Maycox PR. Robbins MJ, et al. Among authors: rocheville m. Brain Res. 2007 Jun 4;1152:215-27. doi: 10.1016/j.brainres.2007.03.028. Epub 2007 Mar 15. Brain Res. 2007. PMID: 17434465

4

7TM pharmacology measured by label-free: a holistic approach to cell signalling.

Rocheville M, Jerman JC. Rocheville M, et al. Curr Opin Pharmacol. 2009 Oct;9(5):643-9. doi: 10.1016/j.coph.2009.06.015. Epub 2009 Aug 9. Curr Opin Pharmacol. 2009. PMID: 19671497 Review.

5

Mining the potential of label-free biosensors for seven-transmembrane receptor drug discovery.

Rocheville M, Martin J, Jerman J, Kostenis E. Rocheville M, et al. Prog Mol Biol Transl Sci. 2013;115:123-42. doi: 10.1016/B978-0-12-394587-7.00003-8. Prog Mol Biol Transl Sci. 2013. PMID: 23415093 Review.

6

Agonist-induced up-regulation of human somatostatin receptor type 1 is regulated by beta-arrestin-1 and requires an essential serine residue in the receptor C-tail.

Ramírez JL, Watt HL, Rocheville M, Kumar U. Ramírez JL, et al. Among authors: rocheville m. Biochim Biophys Acta. 2005 May 20;1669(2):182-92. doi: 10.1016/j.bbamem.2005.02.004. Epub 2005 Feb 22. Biochim Biophys Acta. 2005. PMID: 15893521 Free article.

7

Ligand binding to somatostatin receptors induces receptor-specific oligomer formation in live cells.

Patel RC, Kumar U, Lamb DC, Eid JS, Rocheville M, Grant M, Rani A, Hazlett T, Patel SC, Gratton E, Patel YC. Patel RC, et al. Among authors: rocheville m. Proc Natl Acad Sci U S A. 2002 Mar 5;99(5):3294-9. doi: 10.1073/pnas.042705099. Proc Natl Acad Sci U S A. 2002. PMID: 11880655 Free PMC article.

8

Receptors for dopamine and somatostatin: formation of hetero-oligomers with enhanced functional activity.

Rocheville M, Lange DC, Kumar U, Patel SC, Patel RC, Patel YC. Rocheville M, et al. Science. 2000 Apr 7;288(5463):154-7. doi: 10.1126/science.288.5463.154. Science. 2000. PMID: 10753124

9

Subtypes of the somatostatin receptor assemble as functional homo- and heterodimers.

Rocheville M, Lange DC, Kumar U, Sasi R, Patel RC, Patel YC. Rocheville M, et al. J Biol Chem. 2000 Mar 17;275(11):7862-9. doi: 10.1074/jbc.275.11.7862. J Biol Chem. 2000. PMID: 10713101 Free article.

10

Agonist-dependent up-regulation of human somatostatin receptor type 1 requires molecular signals in the cytoplasmic C-tail.

Hukovic N, Rocheville M, Kumar U, Sasi R, Khare S, Patel YC. Hukovic N, et al. Among authors: rocheville m. J Biol Chem. 1999 Aug 27;274(35):24550-8. doi: 10.1074/jbc.274.35.24550. J Biol Chem. 1999. PMID: 10455118 Free article.

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