Felock PJ - Search Results

1

Total synthesis, characterization, and conformational analysis of the naturally occurring hexadecapeptide integramide A and a diastereomer.

De Zotti M, Damato F, Formaggio F, Crisma M, Schievano E, Mammi S, Kaptein B, Broxterman QB, Felock PJ, Hazuda DJ, Singh SB, Kirschbaum J, Brückner H, Toniolo C. De Zotti M, et al. Among authors: felock pj. Chemistry. 2010 Jan 4;16(1):316-27. doi: 10.1002/chem.200900945. Chemistry. 2010. PMID: 19937615

2

Complete absolute configuration of integramide A, a natural, 16-mer peptide inhibitor of HIV-1 integrase, elucidated by total synthesis.

De Zotti M, Formaggio F, Kaptein B, Broxterman QB, Felock PJ, Hazuda DJ, Singh SB, Brückner H, Toniolo C. De Zotti M, et al. Among authors: felock pj. Chembiochem. 2009 Jan 5;10(1):87-90. doi: 10.1002/cbic.200800443. Chembiochem. 2009. PMID: 18850604 No abstract available.

3

Triple Hyp→Pro replacement in integramide A, a peptaib inhibitor of HIV-1 integrase: Effect on conformation and bioactivity.

De Zotti M, De Borggraeve W, Kaptein B, Broxterman QB, Singh SB, Felock PJ, Hazuda DJ, Formaggio F, Toniolo C. De Zotti M, et al. Among authors: felock pj. Biopolymers. 2011;96(1):49-59. doi: 10.1002/bip.21461. Biopolymers. 2011. PMID: 20560143

4

Isolation, structure and HIV-1 integrase inhibitory activity of exophillic acid, a novel fungal metabolite from Exophiala pisciphila.

Ondeyka JG, Zink DL, Dombrowski AW, Polishook JD, Felock PJ, Hazuda DJ, Singh SB. Ondeyka JG, et al. Among authors: felock pj. J Antibiot (Tokyo). 2003 Dec;56(12):1018-23. doi: 10.7164/antibiotics.56.1018. J Antibiot (Tokyo). 2003. PMID: 15015729 Free article.

5

Isolation, structure, absolute stereochemistry, and HIV-1 integrase inhibitory activity of integrasone, a novel fungal polyketide.

Herath KB, Jayasuriya H, Bills GF, Polishook JD, Dombrowski AW, Guan Z, Felock PJ, Hazuda DJ, Singh SB. Herath KB, et al. Among authors: felock pj. J Nat Prod. 2004 May;67(5):872-4. doi: 10.1021/np0340504. J Nat Prod. 2004. PMID: 15165153

6

Chemical and enzymatic modifications of integric acid and HIV-1 integrase inhibitory activity.

Singh SB, Felock P, Hazuda DJ. Singh SB, et al. Bioorg Med Chem Lett. 2000 Feb 7;10(3):235-8. doi: 10.1016/s0960-894x(99)00666-6. Bioorg Med Chem Lett. 2000. PMID: 10698443

7

Chemistry and structure-activity relationship of HIV-1 integrase inhibitor integracide B and related natural products.

Singh SB, Ondeyka JG, Schleif WA, Felock P, Hazuda DJ. Singh SB, et al. J Nat Prod. 2003 Oct;66(10):1338-44. doi: 10.1021/np030211s. J Nat Prod. 2003. PMID: 14575434

8

Integramides A and B, two novel non-ribosomal linear peptides containing nine C(alpha)-methyl amino acids produced by fungal fermentations that are inhibitors of HIV-1 integrase.

Singh SB, Herath K, Guan Z, Zink DL, Dombrowski AW, Polishook JD, Silverman KC, Lingham RB, Felock PJ, Hazuda DJ. Singh SB, et al. Among authors: felock pj. Org Lett. 2002 May 2;4(9):1431-4. doi: 10.1021/ol025540a. Org Lett. 2002. PMID: 11975596

9

Isolation, structure, and HIV-1 integrase inhibitory activity of Cytosporic acid, a fungal metabolite produced by a Cytospora sp.

Jayasuriya H, Guan Z, Polishook JD, Dombrowski AW, Felock PJ, Hazuda DJ, Singh SB. Jayasuriya H, et al. Among authors: felock pj. J Nat Prod. 2003 Apr;66(4):551-3. doi: 10.1021/np020533g. J Nat Prod. 2003. PMID: 12713414

10

Design and synthesis of substituted 4-oxo-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carboxamides, novel HIV-1 integrase inhibitors.

Langford HM, Williams PD, Homnick CF, Vacca JP, Felock PJ, Stillmock KA, Witmer MV, Hazuda DJ, Gabryelski LJ, Schleif WA. Langford HM, et al. Among authors: felock pj. Bioorg Med Chem Lett. 2008 Jan 15;18(2):721-5. doi: 10.1016/j.bmcl.2007.11.049. Epub 2007 Nov 19. Bioorg Med Chem Lett. 2008. PMID: 18078751

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