Cai H - Search Results

1

Pyrazole-based arylalkyne cathepsin S inhibitors. Part II: optimization of cellular potency.

Ameriks MK, Cai H, Edwards JP, Gebauer D, Gleason E, Gu Y, Karlsson L, Nguyen S, Sun S, Thurmond RL, Zhu J. Ameriks MK, et al. Among authors: cai h. Bioorg Med Chem Lett. 2009 Nov 1;19(21):6135-9. doi: 10.1016/j.bmcl.2009.09.013. Epub 2009 Sep 10. Bioorg Med Chem Lett. 2009. PMID: 19783435

2

Identification of a potent and selective noncovalent cathepsin S inhibitor.

Thurmond RL, Sun S, Sehon CA, Baker SM, Cai H, Gu Y, Jiang W, Riley JP, Williams KN, Edwards JP, Karlsson L. Thurmond RL, et al. Among authors: cai h. J Pharmacol Exp Ther. 2004 Jan;308(1):268-76. doi: 10.1124/jpet.103.056879. Epub 2003 Oct 17. J Pharmacol Exp Ther. 2004. PMID: 14566006

3

Nonpeptidic, noncovalent inhibitors of the cysteine protease cathepsin S.

Thurmond RL, Beavers MP, Cai H, Meduna SP, Gustin DJ, Sun S, Almond HJ, Karlsson L, Edwards JP. Thurmond RL, et al. Among authors: cai h. J Med Chem. 2004 Sep 23;47(20):4799-801. doi: 10.1021/jm0496133. J Med Chem. 2004. PMID: 15369380

4

Discovery and SAR studies of a novel series of noncovalent cathepsin S inhibitors.

Gustin DJ, Sehon CA, Wei J, Cai H, Meduna SP, Khatuya H, Sun S, Gu Y, Jiang W, Thurmond RL, Karlsson L, Edwards JP. Gustin DJ, et al. Among authors: cai h. Bioorg Med Chem Lett. 2005 Mar 15;15(6):1687-91. doi: 10.1016/j.bmcl.2005.01.045. Bioorg Med Chem Lett. 2005. PMID: 15745822

5

Preparation and biological evaluation of indole, benzimidazole, and thienopyrrole piperazine carboxamides: potent human histamine h(4) antagonists.

Venable JD, Cai H, Chai W, Dvorak CA, Grice CA, Jablonowski JA, Shah CR, Kwok AK, Ly KS, Pio B, Wei J, Desai PJ, Jiang W, Nguyen S, Ling P, Wilson SJ, Dunford PJ, Thurmond RL, Lovenberg TW, Karlsson L, Carruthers NI, Edwards JP. Venable JD, et al. Among authors: cai h. J Med Chem. 2005 Dec 29;48(26):8289-98. doi: 10.1021/jm0502081. J Med Chem. 2005. PMID: 16366610

6

Pyrazole-based cathepsin S inhibitors with improved cellular potency.

Wei J, Pio BA, Cai H, Meduna SP, Sun S, Gu Y, Jiang W, Thurmond RL, Karlsson L, Edwards JP. Wei J, et al. Among authors: cai h. Bioorg Med Chem Lett. 2007 Oct 15;17(20):5525-8. doi: 10.1016/j.bmcl.2007.08.038. Epub 2007 Aug 22. Bioorg Med Chem Lett. 2007. PMID: 17822900

7

Triamino pyrimidines and pyridines as histamine H(4) receptor modulators.

Meduna SP, Savall BM, Cai H, Edwards JP, Thurmond RL, McGovern PM. Meduna SP, et al. Among authors: cai h. Bioorg Med Chem Lett. 2011 May 15;21(10):3113-6. doi: 10.1016/j.bmcl.2011.03.017. Epub 2011 Mar 30. Bioorg Med Chem Lett. 2011. PMID: 21458260

8

Diaminopyrimidines, diaminopyridines and diaminopyridazines as histamine H4 receptor modulators.

Savall BM, Meduna SP, Tays K, Cai H, Thurmond RL, McGovern P, Gaul M, Zhao BP, Edwards JP. Savall BM, et al. Among authors: cai h. Bioorg Med Chem Lett. 2015 Feb 15;25(4):956-9. doi: 10.1016/j.bmcl.2014.12.027. Epub 2014 Dec 23. Bioorg Med Chem Lett. 2015. PMID: 25595684

9

Selective inhibition of peripheral cathepsin S reverses tactile allodynia following peripheral nerve injury in mouse.

Eckert WA 3rd, Wiener JJM, Cai H, Ameriks MK, Zhu J, Ngo K, Nguyen S, Fung-Leung WP, Thurmond RL, Grice C, Edwards JP, Chaplan SR, Karlsson L, Sun S. Eckert WA 3rd, et al. Among authors: cai h. Eur J Pharmacol. 2020 Aug 5;880:173171. doi: 10.1016/j.ejphar.2020.173171. Epub 2020 May 11. Eur J Pharmacol. 2020. PMID: 32437743

10

Effects of functional training on physical and technical performance among the athletic population: a systematic review and narrative synthesis.

Xiao W, Bu T, Zhang J, Cai H, Zhu W, Bai X, Zhang L, Geok SK. Xiao W, et al. Among authors: cai h. BMC Sports Sci Med Rehabil. 2025 Jan 3;17(1):2. doi: 10.1186/s13102-024-01040-y. BMC Sports Sci Med Rehabil. 2025. PMID: 39754208 Free PMC article.

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

8,880 results

Search Page

Filters