He R - Search Results

1

Stereoselective HDAC inhibition from cysteine-derived zinc-binding groups.

Butler KV, He R, McLaughlin K, Vistoli G, Langley B, Kozikowski AP. Butler KV, et al. Among authors: he r. ChemMedChem. 2009 Aug;4(8):1292-301. doi: 10.1002/cmdc.200900088. ChemMedChem. 2009. PMID: 19551801

2

Studies of benzamide- and thiol-based histone deacetylase inhibitors in models of oxidative-stress-induced neuronal death: identification of some HDAC3-selective inhibitors.

Chen Y, He R, Chen Y, D'Annibale MA, Langley B, Kozikowski AP. Chen Y, et al. Among authors: he r. ChemMedChem. 2009 May;4(5):842-52. doi: 10.1002/cmdc.200800461. ChemMedChem. 2009. PMID: 19350613

3

Isoxazole moiety in the linker region of HDAC inhibitors adjacent to the Zn-chelating group: effects on HDAC biology and antiproliferative activity.

Tapadar S, He R, Luchini DN, Billadeau DD, Kozikowski AP. Tapadar S, et al. Among authors: he r. Bioorg Med Chem Lett. 2009 Jun 1;19(11):3023-6. doi: 10.1016/j.bmcl.2009.04.058. Epub 2009 Apr 20. Bioorg Med Chem Lett. 2009. PMID: 19419863 Free PMC article.

4

Further structure-activity relationship studies of piperidine-based monoamine transporter inhibitors: effects of piperidine ring stereochemistry on potency. Identification of norepinephrine transporter selective ligands and broad-spectrum transporter inhibitors.

He R, Kurome T, Giberson KM, Johnson KM, Kozikowski AP. He R, et al. J Med Chem. 2005 Dec 15;48(25):7970-9. doi: 10.1021/jm050694s. J Med Chem. 2005. PMID: 16335921

5

Modification of the side chain of micromolide, an anti-tuberculosis natural product.

Yuan H, He R, Wan B, Wang Y, Pauli GF, Franzblau SG, Kozikowski AP. Yuan H, et al. Among authors: he r. Bioorg Med Chem Lett. 2008 Oct 1;18(19):5311-5. doi: 10.1016/j.bmcl.2008.08.027. Epub 2008 Aug 14. Bioorg Med Chem Lett. 2008. PMID: 18774716

6

Structure-activity relationships of compounds targeting mycobacterium tuberculosis 1-deoxy-D-xylulose 5-phosphate synthase.

Mao J, Eoh H, He R, Wang Y, Wan B, Franzblau SG, Crick DC, Kozikowski AP. Mao J, et al. Among authors: he r. Bioorg Med Chem Lett. 2008 Oct 1;18(19):5320-3. doi: 10.1016/j.bmcl.2008.08.034. Epub 2008 Aug 14. Bioorg Med Chem Lett. 2008. PMID: 18783951 Free PMC article.

7

Chemistry and pharmacology of nicotinic ligands based on 6-[5-(azetidin-2-ylmethoxy)pyridin-3-yl]hex-5-yn-1-ol (AMOP-H-OH) for possible use in depression.

Kozikowski AP, Eaton JB, Bajjuri KM, Chellappan SK, Chen Y, Karadi S, He R, Caldarone B, Manzano M, Yuen PW, Lukas RJ. Kozikowski AP, et al. Among authors: he r. ChemMedChem. 2009 Aug;4(8):1279-91. doi: 10.1002/cmdc.200900079. ChemMedChem. 2009. PMID: 19569163 Free PMC article.

8

Synthesis and biological evaluation of triazol-4-ylphenyl-bearing histone deacetylase inhibitors as anticancer agents.

He R, Chen Y, Chen Y, Ougolkov AV, Zhang JS, Savoy DN, Billadeau DD, Kozikowski AP. He R, et al. J Med Chem. 2010 Feb 11;53(3):1347-56. doi: 10.1021/jm901667k. J Med Chem. 2010. PMID: 20055418 Free PMC article.

9

Stereochemistry at the forefront in the design and discovery of novel anti-tuberculosis agents.

Huang Q, He R, Kozikowski AP. Huang Q, et al. Among authors: he r. Curr Top Med Chem. 2011;11(7):810-8. doi: 10.2174/156802611795165205. Curr Top Med Chem. 2011. PMID: 21291395 Review.

10

Identification, synthesis, and pharmacological evaluation of tetrahydroindazole based ligands as novel antituberculosis agents.

Guo S, Song Y, Huang Q, Yuan H, Wan B, Wang Y, He R, Beconi MG, Franzblau SG, Kozikowski AP. Guo S, et al. Among authors: he r. J Med Chem. 2010 Jan 28;53(2):649-59. doi: 10.1021/jm901235p. J Med Chem. 2010. PMID: 20000470

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