Miah A - Search Results

1

Identification of PDE4B Over 4D subtype-selective inhibitors revealing an unprecedented binding mode.

Kranz M, Wall M, Evans B, Miah A, Ballantine S, Delves C, Dombroski B, Gross J, Schneck J, Villa JP, Neu M, Somers DO. Kranz M, et al. Among authors: miah a. Bioorg Med Chem. 2009 Jul 15;17(14):5336-41. doi: 10.1016/j.bmc.2009.03.061. Epub 2009 Apr 5. Bioorg Med Chem. 2009. PMID: 19525117

2

Synthesis and structure-activity relationships of indazole arylsulfonamides as allosteric CC-chemokine receptor 4 (CCR4) antagonists.

Procopiou PA, Barrett JW, Barton NP, Begg M, Clapham D, Copley RC, Ford AJ, Graves RH, Hall DA, Hancock AP, Hill AP, Hobbs H, Hodgson ST, Jumeaux C, Lacroix YM, Miah AH, Morriss KM, Needham D, Sheriff EB, Slack RJ, Smith CE, Sollis SL, Staton H. Procopiou PA, et al. Among authors: miah ah. J Med Chem. 2013 Mar 14;56(5):1946-60. doi: 10.1021/jm301572h. Epub 2013 Feb 27. J Med Chem. 2013. PMID: 23409871

3

Lead identification of benzimidazolone and azabenzimidazolone arylsulfonamides as CC-chemokine receptor 4 (CCR4) antagonists.

Miah AH, Abas H, Begg M, Marsh BJ, O'Flynn DE, Ford AJ, Percy JM, Procopiou PA, Richards SA, Rumley SA. Miah AH, et al. Bioorg Med Chem. 2014 Aug 1;22(15):4298-311. doi: 10.1016/j.bmc.2014.05.021. Epub 2014 May 21. Bioorg Med Chem. 2014. PMID: 24909677 Free article.

4

2,8-Diazaspiro[4.5]decan-8-yl)pyrimidin-4-amine potent CCR4 antagonists capable of inducing receptor endocytosis.

Shukla L, Ajram LA, Begg M, Evans B, Graves RH, Hodgson ST, Lynn SM, Miah AH, Percy JM, Procopiou PA, Richards SA, Slack RJ. Shukla L, et al. Among authors: miah ah. Eur J Med Chem. 2016 Jun 10;115:14-25. doi: 10.1016/j.ejmech.2016.02.058. Epub 2016 Feb 27. Eur J Med Chem. 2016. PMID: 26991939 Free article.

5

Identification of pyrazolopyrimidine arylsulfonamides as CC-chemokine receptor 4 (CCR4) antagonists.

Miah AH, Champigny AC, Graves RH, Hodgson ST, Percy JM, Procopiou PA. Miah AH, et al. Bioorg Med Chem. 2017 Oct 15;25(20):5327-5340. doi: 10.1016/j.bmc.2017.07.052. Epub 2017 Jul 29. Bioorg Med Chem. 2017. PMID: 28801066

6

Structure-based optimisation of orally active & reversible MetAP-2 inhibitors maintaining a tight 'molecular budget'.

Hirst DJ, Brandt M, Bruton G, Christodoulou E, Cutler L, Deeks N, Goodacre JD, Jack T, Lindon M, Miah A, Page K, Parr N, Shukla L, Sims M, Thomas P, Thorpe J, Holmes DS. Hirst DJ, et al. Among authors: miah a. Bioorg Med Chem Lett. 2020 Nov 1;30(21):127533. doi: 10.1016/j.bmcl.2020.127533. Epub 2020 Sep 10. Bioorg Med Chem Lett. 2020. PMID: 32919012

7

Lead identification and structure-activity relationships of heteroarylpyrazole arylsulfonamides as allosteric CC-chemokine receptor 4 (CCR4) antagonists.

Miah AH, Copley RC, O'Flynn D, Percy JM, Procopiou PA. Miah AH, et al. Org Biomol Chem. 2014 Mar 21;12(11):1779-92. doi: 10.1039/c3ob42443j. Org Biomol Chem. 2014. PMID: 24515101 Free article.

8

Optimization of a Series of RIPK2 PROTACs.

Miah AH, Smith IED, Rackham M, Mares A, Thawani AR, Nagilla R, Haile PA, Votta BJ, Gordon LJ, Watt G, Denyer J, Fisher DT, Dace P, Giffen P, Goncalves A, Churcher I, Scott-Stevens P, Harling JD. Miah AH, et al. J Med Chem. 2021 Sep 9;64(17):12978-13003. doi: 10.1021/acs.jmedchem.1c01118. Epub 2021 Aug 25. J Med Chem. 2021. PMID: 34432979

9

Integrated Direct-to-Biology Platform for the Nanoscale Synthesis and Biological Evaluation of PROTACs.

Stevens R, Bendito-Moll E, Battersby DJ, Miah AH, Wellaway N, Law RP, Stacey P, Klimaszewska D, Macina JM, Burley GA, Harling JD. Stevens R, et al. Among authors: miah ah. J Med Chem. 2023 Nov 23;66(22):15437-15452. doi: 10.1021/acs.jmedchem.3c01604. Epub 2023 Nov 7. J Med Chem. 2023. PMID: 37933562

10

Expanding the reaction toolbox for nanoscale direct-to-biology PROTAC synthesis and biological evaluation.

Stevens R, Shrives HJ, Cryan J, Klimaszewska D, Stacey P, Burley GA, Harling JD, Battersby DJ, Miah AH. Stevens R, et al. Among authors: miah ah. RSC Med Chem. 2024 Dec 23. doi: 10.1039/d4md00760c. Online ahead of print. RSC Med Chem. 2024. PMID: 39720740 Free PMC article.

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