Haemers A - Search Results

1

Synthesis and antiplasmodial activity of aminoalkylamino-substituted neocryptolepine derivatives.

El Sayed I, Van der Veken P, Steert K, Dhooghe L, Hostyn S, Van Baelen G, Lemière G, Maes BU, Cos P, Maes L, Joossens J, Haemers A, Pieters L, Augustyns K. El Sayed I, et al. Among authors: haemers a. J Med Chem. 2009 May 14;52(9):2979-88. doi: 10.1021/jm801490z. J Med Chem. 2009. PMID: 19364118

2

Design, synthesis, and SAR of potent and selective dipeptide-derived inhibitors for dipeptidyl peptidases.

Senten K, Van der Veken P, De Meester I, Lambeir AM, Scharpé S, Haemers A, Augustyns K. Senten K, et al. Among authors: haemers a. J Med Chem. 2003 Nov 6;46(23):5005-14. doi: 10.1021/jm0308803. J Med Chem. 2003. PMID: 14584950

3

Gamma-amino-substituted analogues of 1-[(S)-2,4-diaminobutanoyl]piperidine as highly potent and selective dipeptidyl peptidase II inhibitors.

Senten K, Van Der Veken P, De Meester I, Lambeir AM, Scharpé S, Haemers A, Augustyns K. Senten K, et al. Among authors: haemers a. J Med Chem. 2004 May 20;47(11):2906-16. doi: 10.1021/jm031122f. J Med Chem. 2004. PMID: 15139769

4

Synthesis and dipeptidyl peptidase inhibition of N-(4-substituted-2,4-diaminobutanoyl)piperidines.

Soroka A, Van der Veken P, De Meester I, Lambeir AM, Maes MB, Scharpé S, Haemers A, Augustyns K. Soroka A, et al. Among authors: haemers a. Bioorg Med Chem Lett. 2006 Sep 15;16(18):4777-9. doi: 10.1016/j.bmcl.2006.06.082. Epub 2006 Jul 17. Bioorg Med Chem Lett. 2006. PMID: 16844373

5

Diphenyl phosphonate inhibitors for the urokinase-type plasminogen activator: optimization of the P4 position.

Joossens J, Van der Veken P, Surpateanu G, Lambeir AM, El-Sayed I, Ali OM, Augustyns K, Haemers A. Joossens J, et al. Among authors: haemers a. J Med Chem. 2006 Sep 21;49(19):5785-93. doi: 10.1021/jm060622g. J Med Chem. 2006. PMID: 16970403

6

Prolyl peptidases related to dipeptidyl peptidase IV: potential of specific inhibitors in drug discovery.

Van der Veken P, Haemers A, Augustyns K. Van der Veken P, et al. Among authors: haemers a. Curr Top Med Chem. 2007;7(6):621-35. doi: 10.2174/156802607780091046. Curr Top Med Chem. 2007. PMID: 17352682 Review.

7

Dipeptidyl alpha-fluorovinyl Michael acceptors: synthesis and activity against cysteine proteases.

Steert K, El-Sayed I, Van der Veken P, Krishtal A, Van Alsenoy C, Westrop GD, Mottram JC, Coombs GH, Augustyns K, Haemers A. Steert K, et al. Among authors: haemers a. Bioorg Med Chem Lett. 2007 Dec 1;17(23):6563-6. doi: 10.1016/j.bmcl.2007.09.075. Epub 2007 Oct 23. Bioorg Med Chem Lett. 2007. PMID: 17936625

8

Irreversible inhibition of dipeptidyl peptidase 8 by dipeptide-derived diaryl phosphonates.

Van der Veken P, Soroka A, Brandt I, Chen YS, Maes MB, Lambeir AM, Chen X, Haemers A, Scharpé S, Augustyns K, De Meester I. Van der Veken P, et al. Among authors: haemers a. J Med Chem. 2007 Nov 15;50(23):5568-70. doi: 10.1021/jm701005a. Epub 2007 Oct 24. J Med Chem. 2007. PMID: 17958345

9

Small, potent, and selective diaryl phosphonate inhibitors for urokinase-type plasminogen activator with in vivo antimetastatic properties.

Joossens J, Ali OM, El-Sayed I, Surpateanu G, Van der Veken P, Lambeir AM, Setyono-Han B, Foekens JA, Schneider A, Schmalix W, Haemers A, Augustyns K. Joossens J, et al. Among authors: haemers a. J Med Chem. 2007 Dec 27;50(26):6638-46. doi: 10.1021/jm700962j. Epub 2007 Dec 1. J Med Chem. 2007. PMID: 18052026

10

Design and evaluation of Trypanosoma brucei metacaspase inhibitors.

Berg M, Van der Veken P, Joossens J, Muthusamy V, Breugelmans M, Moss CX, Rudolf J, Cos P, Coombs GH, Maes L, Haemers A, Mottram JC, Augustyns K. Berg M, et al. Among authors: haemers a. Bioorg Med Chem Lett. 2010 Mar 15;20(6):2001-6. doi: 10.1016/j.bmcl.2010.01.099. Epub 2010 Jan 25. Bioorg Med Chem Lett. 2010. PMID: 20167486 Free PMC article.

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