Gupte A - Search Results

1

Inhibition of siderophore biosynthesis by 2-triazole substituted analogues of 5'-O-[N-(salicyl)sulfamoyl]adenosine: antibacterial nucleosides effective against Mycobacterium tuberculosis.

Gupte A, Boshoff HI, Wilson DJ, Neres J, Labello NP, Somu RV, Xing C, Barry CE, Aldrich CC. Gupte A, et al. J Med Chem. 2008 Dec 11;51(23):7495-507. doi: 10.1021/jm8008037. J Med Chem. 2008. PMID: 19053762 Free PMC article.

2

5'-O-[(N-acyl)sulfamoyl]adenosines as antitubercular agents that inhibit MbtA: an adenylation enzyme required for siderophore biosynthesis of the mycobactins.

Qiao C, Gupte A, Boshoff HI, Wilson DJ, Bennett EM, Somu RV, Barry CE 3rd, Aldrich CC. Qiao C, et al. Among authors: gupte a. J Med Chem. 2007 Nov 29;50(24):6080-94. doi: 10.1021/jm070905o. Epub 2007 Oct 30. J Med Chem. 2007. PMID: 17967002 Free PMC article.

3

Synthesis of deuterium-labelled 5'-O-[N-(Salicyl)sulfamoyl]adenosine (Sal-AMS-d(4)) as an internal standard for quantitation of Sal-AMS.

Gupte A, Subramanian M, Remmel RP, Aldrich CC. Gupte A, et al. J Labelled Comp Radiopharm. 2008 Feb;51(2):118-122. doi: 10.1002/jlcr.1490. J Labelled Comp Radiopharm. 2008. PMID: 19050743 Free PMC article.

4

Copper(II)-Catalyzed Conversion of Aryl/Heteroaryl Boronic Acids, Boronates, and Trifluoroborates into the Corresponding Azides: Substrate Scope and Limitations.

Grimes KD, Gupte A, Aldrich CC. Grimes KD, et al. Among authors: gupte a. Synthesis (Stuttg). 2010 May 1;2010(9):1441-1448. doi: 10.1055/s-0029-1218683. Synthesis (Stuttg). 2010. PMID: 20526454 Free PMC article.

5

Novel C2-purine position analogs of nitrobenzylmercaptopurine riboside as human equilibrative nucleoside transporter 1 inhibitors.

Gupte A, Buolamwini JK. Gupte A, et al. Bioorg Med Chem. 2007 Dec 15;15(24):7726-37. doi: 10.1016/j.bmc.2007.08.058. Epub 2007 Sep 1. Bioorg Med Chem. 2007. PMID: 17881236 Free PMC article.

6

Synthesis and biological evaluation of isoxazole, oxazole, and oxadiazole containing heteroaryl analogs of biaryl ureas as DGAT1 inhibitors.

Jadhav RD, Kadam KS, Kandre S, Guha T, Reddy MM, Brahma MK, Deshmukh NJ, Dixit A, Doshi L, Potdar N, Enose AA, Vishwakarma RA, Sivaramakrishnan H, Srinivasan S, Nemmani KV, Gupte A, Gangopadhyay AK, Sharma R. Jadhav RD, et al. Among authors: gupte a. Eur J Med Chem. 2012 Aug;54:324-42. doi: 10.1016/j.ejmech.2012.05.016. Epub 2012 May 22. Eur J Med Chem. 2012. PMID: 22683241

7

Evaluation of thiazole containing biaryl analogs as diacylglycerol acyltransferase 1 (DGAT1) inhibitors.

Kadam KS, Jadhav RD, Kandre S, Guha T, Reddy MM, Brahma MK, Deshmukh NJ, Dixit A, Doshi L, Srinivasan S, Devle J, Damre A, Nemmani KV, Gupte A, Sharma R. Kadam KS, et al. Among authors: gupte a. Eur J Med Chem. 2013 Jul;65:337-47. doi: 10.1016/j.ejmech.2013.05.006. Epub 2013 May 14. Eur J Med Chem. 2013. PMID: 23735282

8

Synthesis and evaluation of cyclohexane carboxylic acid head group containing isoxazole and thiazole analogs as DGAT1 inhibitors.

Kandre S, Bhagat PR, Reddy MM, Dalal R, Dixit A, Deshmukh NJ, Anthony J, Bose J, Anupindi R, Sharma R, Gupte A. Kandre S, et al. Among authors: gupte a. Eur J Med Chem. 2014 May 22;79:203-15. doi: 10.1016/j.ejmech.2014.03.077. Epub 2014 Mar 28. Eur J Med Chem. 2014. PMID: 24735646

9

Novel halogenated nitrobenzylthioinosine analogs as es nucleoside transporter inhibitors.

Gupte A, Buolamwini JK. Gupte A, et al. Bioorg Med Chem Lett. 2004 May 3;14(9):2257-60. doi: 10.1016/j.bmcl.2004.02.016. Bioorg Med Chem Lett. 2004. PMID: 15081020

10

CoMFA and CoMSIA 3D-QSAR studies on S(6)-(4-nitrobenzyl)mercaptopurine riboside (NBMPR) analogs as inhibitors of human equilibrative nucleoside transporter 1 (hENT1).

Gupte A, Buolamwini JK. Gupte A, et al. Bioorg Med Chem Lett. 2009 Jan 15;19(2):314-8. doi: 10.1016/j.bmcl.2008.11.092. Epub 2008 Nov 27. Bioorg Med Chem Lett. 2009. PMID: 19091561

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