Klotz KN - Search Results

1

Pyrazolo-triazolo-pyrimidines as adenosine receptor antagonists: A complete structure-activity profile.

Cacciari B, Bolcato C, Spalluto G, Klotz KN, Bacilieri M, Deflorian F, Moro S. Cacciari B, et al. Among authors: klotz kn. Purinergic Signal. 2007 Jun;3(3):183-93. doi: 10.1007/s11302-006-9027-x. Epub 2006 Nov 14. Purinergic Signal. 2007. PMID: 18404432 Free PMC article.

2

Linear and nonlinear 3D-QSAR approaches in tandem with ligand-based homology modeling as a computational strategy to depict the pyrazolo-triazolo-pyrimidine antagonists binding site of the human adenosine A2A receptor.

Michielan L, Bacilieri M, Schiesaro A, Bolcato C, Pastorin G, Spalluto G, Cacciari B, Klotz KN, Kaseda C, Moro S. Michielan L, et al. Among authors: klotz kn. J Chem Inf Model. 2008 Feb;48(2):350-63. doi: 10.1021/ci700300w. Epub 2008 Jan 24. J Chem Inf Model. 2008. PMID: 18215030

3

Pyrazolo-triazolo-pyrimidine Scaffold as a Molecular Passepartout for the Pan-Recognition of Human Adenosine Receptors.

Salmaso V, Persico M, Da Ros T, Spalluto G, Kachler S, Klotz KN, Moro S, Federico S. Salmaso V, et al. Among authors: klotz kn. Biomolecules. 2023 Nov 3;13(11):1610. doi: 10.3390/biom13111610. Biomolecules. 2023. PMID: 38002292 Free PMC article.

4

[1,2,4]Triazolo[1,5-c]pyrimidines as Tools to Investigate A₃ Adenosine Receptors in Cancer Cell Lines.

Federico S, Persico M, Trevisan L, Biasinutto C, Bolcato G, Salmaso V, Da Ros T, Gianferrara T, Prencipe F, Kachler S, Klotz KN, Pacor S, Moro S, Spalluto G. Federico S, et al. Among authors: klotz kn. ChemMedChem. 2023 Nov 2;18(21):e202300299. doi: 10.1002/cmdc.202300299. Epub 2023 Sep 22. ChemMedChem. 2023. PMID: 37675643

5

A_2A Adenosine Receptor Antagonists: Are Triazolotriazine and Purine Scaffolds Interchangeable?

Spinaci A, Lambertucci C, Buccioni M, Dal Ben D, Graiff C, Barbalace MC, Hrelia S, Angeloni C, Tayebati SK, Ubaldi M, Masi A, Klotz KN, Volpini R, Marucci G. Spinaci A, et al. Among authors: klotz kn. Molecules. 2022 Apr 7;27(8):2386. doi: 10.3390/molecules27082386. Molecules. 2022. PMID: 35458588 Free PMC article.

6

Potent and selective A₃ adenosine receptor antagonists bearing aminoesters as heterobifunctional moieties.

Federico S, Margiotta E, Moro S, Kachler S, Klotz KN, Spalluto G. Federico S, et al. Among authors: klotz kn. RSC Med Chem. 2020 Dec 14;12(2):254-262. doi: 10.1039/d0md00380h. eCollection 2021 Mar 4. RSC Med Chem. 2020. PMID: 34046614 Free PMC article.

7

Pharmacological characterisation of novel adenosine A₃ receptor antagonists.

Barkan K, Lagarias P, Stampelou M, Stamatis D, Hoare S, Safitri D, Klotz KN, Vrontaki E, Kolocouris A, Ladds G. Barkan K, et al. Among authors: klotz kn. Sci Rep. 2020 Nov 27;10(1):20781. doi: 10.1038/s41598-020-74521-y. Sci Rep. 2020. PMID: 33247159 Free PMC article.

8

Bronchospasmolytic and Adenosine Binding Activity of 8- (Proline / Pyrazole)- Substituted Xanthine Derivatives.

Singh S, Ojha M, Yadav D, Kachler S, Klotz KN, Yadav R. Singh S, et al. Among authors: klotz kn. Curr Drug Discov Technol. 2021;18(5):e22092020186181. doi: 10.2174/1570163817666200922121005. Curr Drug Discov Technol. 2021. PMID: 32962622

9

Adenosine Receptor Ligands: Coumarin-Chalcone Hybrids as Modulating Agents on the Activity of hARs.

Vazquez-Rodriguez S, Vilar S, Kachler S, Klotz KN, Uriarte E, Borges F, Matos MJ. Vazquez-Rodriguez S, et al. Among authors: klotz kn. Molecules. 2020 Sep 19;25(18):4306. doi: 10.3390/molecules25184306. Molecules. 2020. PMID: 32961824 Free PMC article.

10

Correction to: Agonists activate different A_2B adenosine receptor signaling pathways in MDA-MB-231 breast cancer cells with distinct potencies.

Koussémou M, Klotz KN. Koussémou M, et al. Among authors: klotz kn. Naunyn Schmiedebergs Arch Pharmacol. 2020 Nov;393(11):2239. doi: 10.1007/s00210-020-01969-0. Naunyn Schmiedebergs Arch Pharmacol. 2020. PMID: 32870337

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