Tai A - Search Results

1

Cyclooxygenase-1-selective inhibitors are attractive candidates for analgesics that do not cause gastric damage. design and in vitro/in vivo evaluation of a benzamide-type cyclooxygenase-1 selective inhibitor.

Kakuta H, Zheng X, Oda H, Harada S, Sugimoto Y, Sasaki K, Tai A. Kakuta H, et al. Among authors: tai a. J Med Chem. 2008 Apr 24;51(8):2400-11. doi: 10.1021/jm701191z. Epub 2008 Mar 26. J Med Chem. 2008. PMID: 18363350

2

Analgesic agents without gastric damage: design and synthesis of structurally simple benzenesulfonanilide-type cyclooxygenase-1-selective inhibitors.

Zheng X, Oda H, Takamatsu K, Sugimoto Y, Tai A, Akaho E, Ali HI, Oshiki T, Kakuta H, Sasaki K. Zheng X, et al. Among authors: tai a. Bioorg Med Chem. 2007 Jan 15;15(2):1014-21. doi: 10.1016/j.bmc.2006.10.029. Epub 2006 Oct 18. Bioorg Med Chem. 2007. PMID: 17079150

3

Effect of the oral absorption of benzenesulfonanilide-type cyclooxygenase-1 inhibitors on analgesic action and gastric ulcer formation.

Zheng X, Oda H, Harada S, Sugimoto Y, Tai A, Sasaki K, Kakuta H. Zheng X, et al. Among authors: tai a. J Pharm Sci. 2008 Dec;97(12):5446-52. doi: 10.1002/jps.21388. J Pharm Sci. 2008. PMID: 18452178

4

Design and synthesis of benzenesulfonanilides active against methicillin-resistant Staphylococcus aureus and vancomycin-resistant Enterococcus.

Namba K, Zheng X, Motoshima K, Kobayashi H, Tai A, Takahashi E, Sasaki K, Okamoto K, Kakuta H. Namba K, et al. Among authors: tai a. Bioorg Med Chem. 2008 Jun 1;16(11):6131-44. doi: 10.1016/j.bmc.2008.04.040. Epub 2008 Apr 24. Bioorg Med Chem. 2008. PMID: 18468909

5

Identification of urine metabolites of TFAP, a cyclooxygenase-1 inhibitor.

Kakuta H, Fukai R, Xiaoxia Z, Ohsawa F, Bamba T, Hirata K, Tai A. Kakuta H, et al. Among authors: tai a. Bioorg Med Chem Lett. 2010 Mar 15;20(6):1840-3. doi: 10.1016/j.bmcl.2010.01.161. Epub 2010 Feb 6. Bioorg Med Chem Lett. 2010. PMID: 20185310

6

Design and synthesis of novel cyclooxygenase-1 inhibitors as analgesics: 5-amino-2-ethoxy-N-(substituted-phenyl)benzamides.

Fukai R, Zheng X, Motoshima K, Tai A, Yazama F, Kakuta H. Fukai R, et al. Among authors: tai a. ChemMedChem. 2011 Mar 7;6(3):550-60. doi: 10.1002/cmdc.201000462. Epub 2011 Jan 7. ChemMedChem. 2011. PMID: 21360824

7

Synthesis and characterization of a series of novel monoacylated ascorbic acid derivatives, 6-O-acyl-2-O-alpha-D-glucopyranosyl-L-ascorbic acids, as skin antioxidants.

Yamamoto I, Tai A, Fujinami Y, Sasaki K, Okazaki S. Yamamoto I, et al. Among authors: tai a. J Med Chem. 2002 Jan 17;45(2):462-8. doi: 10.1021/jm010379f. J Med Chem. 2002. PMID: 11784150

8

Pyridinium cationic-dimer antimalarials, unlike chloroquine, act selectively between the schizont stage and the ring stage of Plasmodium falciparum.

Yoshikawa M, Motoshima K, Fujimoto K, Tai A, Kakuta H, Sasaki K. Yoshikawa M, et al. Among authors: tai a. Bioorg Med Chem. 2008 Jun 1;16(11):6027-33. doi: 10.1016/j.bmc.2008.04.051. Epub 2008 Apr 25. Bioorg Med Chem. 2008. PMID: 18479926

9

Replacing alkyl sulfonamide with aromatic sulfonamide in sulfonamide-type RXR agonists favors switch towards antagonist activity.

Morishita K, Yakushiji N, Ohsawa F, Takamatsu K, Matsuura N, Makishima M, Kawahata M, Yamaguchi K, Tai A, Sasaki K, Kakuta H. Morishita K, et al. Among authors: tai a. Bioorg Med Chem Lett. 2009 Feb 1;19(3):1001-3. doi: 10.1016/j.bmcl.2008.11.086. Epub 2008 Nov 27. Bioorg Med Chem Lett. 2009. PMID: 19095448

10

Modification at the acidic domain of RXR agonists has little effect on permissive RXR-heterodimer activation.

Fujii S, Ohsawa F, Yamada S, Shinozaki R, Fukai R, Makishima M, Enomoto S, Tai A, Kakuta H. Fujii S, et al. Among authors: tai a. Bioorg Med Chem Lett. 2010 Sep 1;20(17):5139-42. doi: 10.1016/j.bmcl.2010.07.012. Epub 2010 Jul 8. Bioorg Med Chem Lett. 2010. PMID: 20656484

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