Petukhov PA - Search Results

1

5-tert-butyl-N-pyrazol-4-yl-4,5,6,7-tetrahydrobenzo[d]isoxazole-3-carboxamide derivatives as novel potent inhibitors of Mycobacterium tuberculosis pantothenate synthetase: initiating a quest for new antitubercular drugs.

Velaparthi S, Brunsteiner M, Uddin R, Wan B, Franzblau SG, Petukhov PA. Velaparthi S, et al. Among authors: petukhov pa. J Med Chem. 2008 Apr 10;51(7):1999-2002. doi: 10.1021/jm701372r. Epub 2008 Mar 13. J Med Chem. 2008. PMID: 18335974 Review.

2

Synthesis of urea-based inhibitors as active site probes of glutamate carboxypeptidase II: efficacy as analgesic agents.

Kozikowski AP, Zhang J, Nan F, Petukhov PA, Grajkowska E, Wroblewski JT, Yamamoto T, Bzdega T, Wroblewska B, Neale JH. Kozikowski AP, et al. Among authors: petukhov pa. J Med Chem. 2004 Mar 25;47(7):1729-38. doi: 10.1021/jm0306226. J Med Chem. 2004. PMID: 15027864

3

Synthesis, molecular modeling, and biological studies of novel piperidine-based analogues of cocaine: evidence of unfavorable interactions proximal to the 3alpha-position of the piperidine ring.

Petukhov PA, Zhang J, Wang CZ, Ye YP, Johnson KM, Kozikowski AP. Petukhov PA, et al. J Med Chem. 2004 Jun 3;47(12):3009-18. doi: 10.1021/jm0303296. J Med Chem. 2004. PMID: 15163183

4

CoMFA study of piperidine analogues of cocaine at the dopamine transporter: exploring the binding mode of the 3 alpha-substituent of the piperidine ring using pharmacophore-based flexible alignment.

Yuan H, Kozikowski AP, Petukhov PA. Yuan H, et al. Among authors: petukhov pa. J Med Chem. 2004 Dec 2;47(25):6137-43. doi: 10.1021/jm049544s. J Med Chem. 2004. PMID: 15566285

5

Chemistry and biology of mercaptoacetamides as novel histone deacetylase inhibitors.

Chen B, Petukhov PA, Jung M, Velena A, Eliseeva E, Dritschilo A, Kozikowski AP. Chen B, et al. Among authors: petukhov pa. Bioorg Med Chem Lett. 2005 Mar 1;15(5):1389-92. doi: 10.1016/j.bmcl.2005.01.006. Bioorg Med Chem Lett. 2005. PMID: 15713393

6

Novel pyridyl ring C5 substituted analogues of epibatidine and 3-(1-methyl-2(S)-pyrrolidinylmethoxy)pyridine (A-84543) as highly selective agents for neuronal nicotinic acetylcholine receptors containing beta2 subunits.

Wei ZL, Xiao Y, Yuan H, Baydyuk M, Petukhov PA, Musachio JL, Kellar KJ, Kozikowski AP. Wei ZL, et al. Among authors: petukhov pa. J Med Chem. 2005 Mar 24;48(6):1721-4. doi: 10.1021/jm0492406. J Med Chem. 2005. PMID: 15771418

7

Computational evidence for the ligand selectivity to the alpha4beta2 and alpha3beta4 nicotinic acetylcholine receptors.

Yuan H, Petukhov PA. Yuan H, et al. Among authors: petukhov pa. Bioorg Med Chem. 2006 Dec 1;14(23):7936-42. doi: 10.1016/j.bmc.2006.07.049. Epub 2006 Aug 21. Bioorg Med Chem. 2006. PMID: 16919961

8

Improved 3D-QSAR CoMFA of the dopamine transporter blockers with multiple conformations using the genetic algorithm.

Yuan H, Petukhov PA. Yuan H, et al. Among authors: petukhov pa. Bioorg Med Chem Lett. 2006 Dec 15;16(24):6267-72. doi: 10.1016/j.bmcl.2006.09.037. Epub 2006 Oct 5. Bioorg Med Chem Lett. 2006. PMID: 17027270

9

Benzothiophene selective estrogen receptor modulators with modulated oxidative activity and receptor affinity.

Qin Z, Kastrati I, Chandrasena RE, Liu H, Yao P, Petukhov PA, Bolton JL, Thatcher GR. Qin Z, et al. Among authors: petukhov pa. J Med Chem. 2007 May 31;50(11):2682-92. doi: 10.1021/jm070079j. Epub 2007 May 10. J Med Chem. 2007. PMID: 17489582

10

Receptor-based modeling and 3D-QSAR for a quantitative production of the butyrylcholinesterase inhibitors based on genetic algorithm.

Zaheer-ul H, Uddin R, Yuan H, Petukhov PA, Choudhary MI, Madura JD. Zaheer-ul H, et al. Among authors: petukhov pa. J Chem Inf Model. 2008 May;48(5):1092-103. doi: 10.1021/ci8000056. Epub 2008 Apr 29. J Chem Inf Model. 2008. PMID: 18444627

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