Emmerson PJ - Search Results

1

Structure activity relationship studies of carboxamido-biaryl ethers as opioid receptor antagonists (OpRAs). Part 2.

Takeuchi K, Holloway WG, Mitch CH, Quimby SJ, McKinzie JH, Suter TM, Statnick MA, Surface PL, Emmerson PJ, Thomas EM, Siegel MG. Takeuchi K, et al. Among authors: emmerson pj. Bioorg Med Chem Lett. 2007 Dec 15;17(24):6841-6. doi: 10.1016/j.bmcl.2007.10.025. Epub 2007 Oct 17. Bioorg Med Chem Lett. 2007. PMID: 17980586

2

Galanin receptor-mediated inhibition of glutamate release in the arcuate nucleus of the hypothalamus.

Kinney GA, Emmerson PJ, Miller RJ. Kinney GA, et al. Among authors: emmerson pj. J Neurosci. 1998 May 15;18(10):3489-500. doi: 10.1523/JNEUROSCI.18-10-03489.1998. J Neurosci. 1998. PMID: 9570780 Free PMC article.

3

Regulation of neurotransmission in the arcuate nucleus of the rat by different neuropeptide Y receptors.

Rhim H, Kinney GA, Emmerson PJ, Miller RJ. Rhim H, et al. Among authors: emmerson pj. J Neurosci. 1997 May 1;17(9):2980-9. doi: 10.1523/JNEUROSCI.17-09-02980.1997. J Neurosci. 1997. PMID: 9157196 Free PMC article.

4

Na+-dependent high affinity binding of [3H]LY515300, a 3,4-dimethyl-4-(3-hydroxyphenyl)piperidine opioid receptor inverse agonist.

Statnick MA, Suter TM, Gackenheimer SL, Emmerson PJ, Quimby SJ, Gehlert DR, Wheeler WJ, Mitch CH. Statnick MA, et al. Among authors: emmerson pj. Eur J Pharmacol. 2003 Dec 15;482(1-3):139-50. doi: 10.1016/j.ejphar.2003.09.043. Eur J Pharmacol. 2003. PMID: 14660015

5

Synthesis and structure-activity relationships of novel arylpiperazines as potent and selective agonists of the melanocortin subtype-4 receptor.

Richardson TI, Ornstein PL, Briner K, Fisher MJ, Backer RT, Biggers CK, Clay MP, Emmerson PJ, Hertel LW, Hsiung HM, Husain S, Kahl SD, Lee JA, Lindstrom TD, Martinelli MJ, Mayer JP, Mullaney JT, O'Brien TP, Pawlak JM, Revell KD, Shah J, Zgombick JM, Herr RJ, Melekhov A, Sampson PB, King CH. Richardson TI, et al. Among authors: emmerson pj. J Med Chem. 2004 Jan 29;47(3):744-55. doi: 10.1021/jm0304109. J Med Chem. 2004. PMID: 14736255

6

Development of displacement binding and GTPgammaS scintillation proximity assays for the identification of antagonists of the micro-opioid receptor.

Rodgers G, Hubert C, McKinzie J, Suter T, Statnick M, Emmerson P, Stancato L. Rodgers G, et al. Assay Drug Dev Technol. 2003 Oct;1(5):627-36. doi: 10.1089/154065803770380986. Assay Drug Dev Technol. 2003. PMID: 15090235

7

Na+ modulation, inverse agonism, and anorectic potency of 4-phenylpiperidine opioid antagonists.

Emmerson PJ, McKinzie JH, Surface PL, Suter TM, Mitch CH, Statnick MA. Emmerson PJ, et al. Eur J Pharmacol. 2004 Jun 28;494(2-3):121-30. doi: 10.1016/j.ejphar.2004.04.050. Eur J Pharmacol. 2004. PMID: 15212965

8

Discovery of a beta-MSH-derived MC-4R selective agonist.

Mayer JP, Hsiung HM, Flora DB, Edwards P, Smith DP, Zhang XY, Gadski RA, Heiman ML, Hertel JL, Emmerson PJ, Husain S, O'brien TP, Kahl SD, Smiley DL, Zhang L, Dimarchi RD, Yan LZ. Mayer JP, et al. Among authors: emmerson pj. J Med Chem. 2005 May 5;48(9):3095-8. doi: 10.1021/jm0501432. J Med Chem. 2005. PMID: 15857110

9

SAR and biological evaluation of novel trans-3,4-dimethyl-4-arylpiperidine derivatives as opioid antagonists.

Díaz N, Benvenga M, Emmerson P, Favors R, Mangold M, McKinzie J, Patel N, Peters S, Quimby S, Shannon H, Siegel M, Statnick M, Thomas E, Woodland J, Surface P, Mitch C. Díaz N, et al. Bioorg Med Chem Lett. 2005 Sep 1;15(17):3844-8. doi: 10.1016/j.bmcl.2005.05.123. Bioorg Med Chem Lett. 2005. PMID: 15993591

10

Potent and selective MC-4 receptor agonists based on a novel disulfide scaffold.

Yan LZ, Flora D, Edwards P, Smiley DL, Emmerson PJ, Hsiung HM, Gadski R, Hertel J, Heiman ML, Husain S, O'Brien TP, Kahl SD, Zhang L, Dimarchi RD, Mayer JP. Yan LZ, et al. Among authors: emmerson pj. Bioorg Med Chem Lett. 2005 Oct 15;15(20):4611-4. doi: 10.1016/j.bmcl.2005.06.081. Bioorg Med Chem Lett. 2005. PMID: 16105738

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