Varani K - Search Results

1

Design, synthesis, and preliminary pharmacological evaluation of new quinoline derivatives as nicotinic ligands.

Guandalini L, Norcini M, Varani K, Pistolozzi M, Gotti C, Bazzicalupi C, Martini E, Dei S, Manetti D, Scapecchi S, Teodori E, Bertucci C, Ghelardini C, Romanelli MN. Guandalini L, et al. Among authors: varani k. J Med Chem. 2007 Oct 4;50(20):4993-5002. doi: 10.1021/jm070325r. Epub 2007 Sep 12. J Med Chem. 2007. PMID: 17850058

2

Design, synthesis, and biological evaluation of a second generation of pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as potent and selective A2A adenosine receptor antagonists.

Baraldi PG, Cacciari B, Spalluto G, Bergonzoni M, Dionisotti S, Ongini E, Varani K, Borea PA. Baraldi PG, et al. Among authors: varani k. J Med Chem. 1998 Jun 4;41(12):2126-33. doi: 10.1021/jm9708689. J Med Chem. 1998. PMID: 9622554

3

Hybridized and isosteric analogues of N1-acetyl-N4-dimethyl-piperazinium iodide (ADMP) and N1-phenyl-N4-dimethyl-piperazinium iodide (DMPP) with central nicotinic action.

Manetti D, Bartolini A, Borea PA, Bellucci C, Dei S, Ghelardini C, Gualtieri F, Romanelli MN, Scapecchi S, Teodori E, Varani K. Manetti D, et al. Among authors: varani k. Bioorg Med Chem. 1999 Mar;7(3):457-65. doi: 10.1016/s0968-0896(98)00259-4. Bioorg Med Chem. 1999. PMID: 10220032

4

Further studies on nociceptin-related peptides: discovery of a new chemical template with antagonist activity on the nociceptin receptor.

Guerrini R, Caló G, Bigoni R, Rizzi A, Varani K, Toth G, Gessi S, Hashiba E, Hashimoto Y, Lambert DG, Borea PA, Tomatis R, Salvadori S, Regoli D. Guerrini R, et al. Among authors: varani k. J Med Chem. 2000 Jul 27;43(15):2805-13. doi: 10.1021/jm990075h. J Med Chem. 2000. PMID: 10956188

5

Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives as highly potent and selective human A(3) adenosine receptor antagonists: influence of the chain at the N(8) pyrazole nitrogen.

Baraldi PG, Cacciari B, Romagnoli R, Spalluto G, Moro S, Klotz KN, Leung E, Varani K, Gessi S, Merighi S, Borea PA. Baraldi PG, et al. Among authors: varani k. J Med Chem. 2000 Dec 14;43(25):4768-80. doi: 10.1021/jm001047y. J Med Chem. 2000. PMID: 11123985

6

Ala scan analogues of HOE 140. Synthesis and biological activities.

Quartara L, Ricci R, Meini S, Patacchini R, Giolitti A, Amadesi S, Rizzi C, Rizzi A, Varani K, Borea PA, Maggi CA, Regoli D. Quartara L, et al. Among authors: varani k. Eur J Med Chem. 2000 Nov;35(11):1001-10. doi: 10.1016/s0223-5234(00)01182-x. Eur J Med Chem. 2000. PMID: 11137228

7

Structure-affinity relationships of a unique nicotinic ligand: N(1)-dimethyl-N(4)-phenylpiperazinium iodide (DMPP).

Romanelli MN, Manetti D, Scapecchi S, Borea PA, Dei S, Bartolini A, Ghelardini C, Gualtieri F, Guandalini L, Varani K. Romanelli MN, et al. Among authors: varani k. J Med Chem. 2001 Nov 8;44(23):3946-55. doi: 10.1021/jm010901y. J Med Chem. 2001. PMID: 11689081

8

Structure-activity studies of the Phe(4) residue of nociceptin(1-13)-NH(2): identification of highly potent agonists of the nociceptin/orphanin FQ receptor.

Guerrini R, Caló G, Bigoni R, Rizzi D, Rizzi A, Zucchini M, Varani K, Hashiba E, Lambert DG, Toth G, Borea PA, Salvadori S, Regoli D. Guerrini R, et al. Among authors: varani k. J Med Chem. 2001 Nov 8;44(23):3956-64. doi: 10.1021/jm010221v. J Med Chem. 2001. PMID: 11689082

9

Synthesis, biological activity, and molecular modeling investigation of new pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine derivatives as human A(3) adenosine receptor antagonists.

Baraldi PG, Cacciari B, Moro S, Spalluto G, Pastorin G, Da Ros T, Klotz KN, Varani K, Gessi S, Borea PA. Baraldi PG, et al. Among authors: varani k. J Med Chem. 2002 Feb 14;45(4):770-80. doi: 10.1021/jm0109614. J Med Chem. 2002. PMID: 11831890

10

Synthesis and pharmacological evaluation of some (pyridyl)cyclopropylmethyl amines and their methiodides as nicotinic receptor ligands.

Guandalini L, Dei S, Manetti D, Romanelli MN, Scapecchi S, Teodori E, Varani K. Guandalini L, et al. Among authors: varani k. Farmaco. 2002 Jun;57(6):487-96. doi: 10.1016/s0014-827x(02)01234-x. Farmaco. 2002. PMID: 12088064

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

300 results

Search Page

Filters