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Page 1
C1'-cycloalkyl side chain pharmacophore in tetrahydrocannabinols.
Papahatjis DP, Nahmias VR, Nikas SP, Andreou T, Alapafuja SO, Tsotinis A, Guo J, Fan P, Makriyannis A. Papahatjis DP, et al. Among authors: alapafuja so. J Med Chem. 2007 Aug 23;50(17):4048-60. doi: 10.1021/jm070121a. Epub 2007 Aug 2. J Med Chem. 2007. PMID: 17672444
Novel 1',1'-chain substituted hexahydrocannabinols: 9β-hydroxy-3-(1-hexyl-cyclobut-1-yl)-hexahydrocannabinol (AM2389) a highly potent cannabinoid receptor 1 (CB1) agonist.
Nikas SP, Alapafuja SO, Papanastasiou I, Paronis CA, Shukla VG, Papahatjis DP, Bowman AL, Halikhedkar A, Han X, Makriyannis A. Nikas SP, et al. Among authors: alapafuja so. J Med Chem. 2010 Oct 14;53(19):6996-7010. doi: 10.1021/jm100641g. J Med Chem. 2010. PMID: 20925434 Free PMC article.
Sulfonyl fluoride inhibitors of fatty acid amide hydrolase.
Alapafuja SO, Nikas SP, Bharathan IT, Shukla VG, Nasr ML, Bowman AL, Zvonok N, Li J, Shi X, Engen JR, Makriyannis A. Alapafuja SO, et al. J Med Chem. 2012 Nov 26;55(22):10074-89. doi: 10.1021/jm301205j. Epub 2012 Nov 2. J Med Chem. 2012. PMID: 23083016 Free PMC article.
Synthesis and evaluation of potent and selective MGL inhibitors as a glaucoma treatment.
Alapafuja SO, Malamas MS, Shukla V, Zvonok A, Miller S, Daily L, Rajarshi G, Miyabe CY, Chandrashekhar H, Wood J, Tyukhtenko S, Straiker A, Makriyannis A. Alapafuja SO, et al. Bioorg Med Chem. 2019 Jan 1;27(1):55-64. doi: 10.1016/j.bmc.2018.11.003. Epub 2018 Nov 3. Bioorg Med Chem. 2019. PMID: 30446439 Free PMC article.
Inhibitor of fatty acid amide hydrolase normalizes cardiovascular function in hypertension without adverse metabolic effects.
Godlewski G, Alapafuja SO, Bátkai S, Nikas SP, Cinar R, Offertáler L, Osei-Hyiaman D, Liu J, Mukhopadhyay B, Harvey-White J, Tam J, Pacak K, Blankman JL, Cravatt BF, Makriyannis A, Kunos G. Godlewski G, et al. Among authors: alapafuja so. Chem Biol. 2010 Nov 24;17(11):1256-66. doi: 10.1016/j.chembiol.2010.08.013. Chem Biol. 2010. PMID: 21095576 Free PMC article.
Design and Structure-Activity Relationships of Isothiocyanates as Potent and Selective N-Acylethanolamine-Hydrolyzing Acid Amidase Inhibitors.
Malamas MS, Pavlopoulos S, Alapafuja SO, Farah SI, Zvonok A, Mohammad KA, West J, Perry NT, Pelekoudas DN, Rajarshi G, Shields C, Chandrashekhar H, Wood J, Makriyannis A. Malamas MS, et al. Among authors: alapafuja so. J Med Chem. 2021 May 13;64(9):5956-5972. doi: 10.1021/acs.jmedchem.1c00076. Epub 2021 Apr 26. J Med Chem. 2021. PMID: 33900772
Effects of fatty acid amide hydrolase (FAAH) inhibitors on working memory in rats.
Panlilio LV, Thorndike EB, Nikas SP, Alapafuja SO, Bandiera T, Cravatt BF, Makriyannis A, Piomelli D, Goldberg SR, Justinova Z. Panlilio LV, et al. Among authors: alapafuja so. Psychopharmacology (Berl). 2016 May;233(10):1879-88. doi: 10.1007/s00213-015-4140-6. Epub 2015 Nov 12. Psychopharmacology (Berl). 2016. PMID: 26558620 Free PMC article.
Cannabinoid Antagonist Drug Discrimination in Nonhuman Primates.
Kangas BD, Zakarian AS, Vemuri K, Alapafuja SO, Jiang S, Nikas SP, Makriyannis A, Bergman J. Kangas BD, et al. Among authors: alapafuja so. J Pharmacol Exp Ther. 2020 Jan;372(1):119-127. doi: 10.1124/jpet.119.261818. Epub 2019 Oct 22. J Pharmacol Exp Ther. 2020. PMID: 31641018 Free PMC article.
16 results