Gelain A - Search Results

1

Structure-activity studies and analgesic efficacy of N-(3-pyridinyl)-bridged bicyclic diamines, exceptionally potent agonists at nicotinic acetylcholine receptors.

Bunnelle WH, Daanen JF, Ryther KB, Schrimpf MR, Dart MJ, Gelain A, Meyer MD, Frost JM, Anderson DJ, Buckley M, Curzon P, Cao YJ, Puttfarcken P, Searle X, Ji J, Putman CB, Surowy C, Toma L, Barlocco D. Bunnelle WH, et al. Among authors: gelain a. J Med Chem. 2007 Jul 26;50(15):3627-44. doi: 10.1021/jm070018l. Epub 2007 Jun 22. J Med Chem. 2007. PMID: 17585748

2

6-Chloropyridazin-3-yl derivatives active as nicotinic agents: synthesis, binding, and modeling studies.

Toma L, Quadrelli P, Bunnelle WH, Anderson DJ, Meyer MD, Cignarella G, Gelain A, Barlocco D. Toma L, et al. Among authors: gelain a. J Med Chem. 2002 Aug 29;45(18):4011-7. doi: 10.1021/jm0208830. J Med Chem. 2002. PMID: 12190322

3

Novel 3-arylamino- and 3-cycloalkylamino-5, 6-diphenyl-pyridazines active as ACAT inhibitors.

Toma L, Giovannoni MP, Vergelli C, Dal Piaz V, Kwon BM, Kim YK, Gelain A, Barlocco D. Toma L, et al. Among authors: gelain a. Arch Pharm (Weinheim). 2002;335(11-12):563-6. doi: 10.1002/ardp.200290010. Arch Pharm (Weinheim). 2002. PMID: 12596221

4

ortho-Halogen naphthaleins as specific inhibitors of Lactobacillus casei thymidylate synthase. Conformational properties and biological activity.

Ghelli S, Rinaldi M, Barlocco D, Gelain A, Pecorari P, Tondi D, Rastelli G, Costi MP. Ghelli S, et al. Among authors: gelain a. Bioorg Med Chem. 2003 Mar 20;11(6):951-63. doi: 10.1016/s0968-0896(02)00541-2. Bioorg Med Chem. 2003. PMID: 12614880

5

Mono- or diphenylpyridazines connected to N-(2,4-difluorophenyl)-N'-heptylurea as acyl-CoA:cholesterol acyltransferase inhibitors.

Gelain A, Bettinelli I, Barlocco D, Kwon BM, Jeong TS, Cho KH, Toma L. Gelain A, et al. J Med Chem. 2005 Dec 1;48(24):7708-13. doi: 10.1021/jm050703x. J Med Chem. 2005. PMID: 16302810

6

Antibacterial agent discovery using thymidylate synthase biolibrary screening.

Costi MP, Gelain A, Barlocco D, Ghelli S, Soragni F, Reniero F, Rossi T, Ruberto A, Guillou C, Cavazzuti A, Casolari C, Ferrari S. Costi MP, et al. Among authors: gelain a. J Med Chem. 2006 Oct 5;49(20):5958-68. doi: 10.1021/jm051187d. J Med Chem. 2006. PMID: 17004711

7

3-heptylamino-5-phenylpyridazine derivatives as analogues of Acyl-CoA: cholesterol acyltransferase inhibitors containing the N-heptyl-N'-arylureidic moiety.

Gelain A, Barlocco D, Kwon BM, Jeong TS, Im KR, Legnani L, Toma L. Gelain A, et al. Arch Pharm (Weinheim). 2006 Dec;339(12):645-51. doi: 10.1002/ardp.200600106. Arch Pharm (Weinheim). 2006. PMID: 17109461

8

Biphenyl versus phenylpyridazine derivatives: the role of the heterocycle in a series of acyl-CoA:cholesterol acyl transferase inhibitors.

Gelain A, Barlocco D, Kwon BM, Jeong TS, Im KR, Legnani L, Toma L. Gelain A, et al. J Med Chem. 2008 Mar 13;51(5):1474-7. doi: 10.1021/jm701474c. Epub 2008 Feb 20. J Med Chem. 2008. PMID: 18284184

9

Semicarbazide-sensitive amine oxidase/vascular adhesion protein 1: recent developments concerning substrates and inhibitors of a promising therapeutic target.

Dunkel P, Gelain A, Barlocco D, Haider N, Gyires K, Sperlágh B, Magyar K, Maccioni E, Fadda A, Mátyus P. Dunkel P, et al. Among authors: gelain a. Curr Med Chem. 2008;15(18):1827-39. doi: 10.2174/092986708785133022. Curr Med Chem. 2008. PMID: 18691041 Review.

10

Signal transducer and activator of transcription 3 (STAT3): a promising target for anticancer therapy.

Masciocchi D, Gelain A, Villa S, Meneghetti F, Barlocco D. Masciocchi D, et al. Among authors: gelain a. Future Med Chem. 2011 Apr;3(5):567-97. doi: 10.4155/fmc.11.22. Future Med Chem. 2011. PMID: 21526897 Review.

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