Pochet L - Search Results

1

Mechanism-based thrombin inhibitors: design, synthesis, and molecular docking of a new selective 2-oxo-2H-1-benzopyran derivative.

Frédérick R, Robert S, Charlier C, Wouters J, Masereel B, Pochet L. Frédérick R, et al. Among authors: pochet l. J Med Chem. 2007 Jul 26;50(15):3645-50. doi: 10.1021/jm061368v. Epub 2007 Jun 20. J Med Chem. 2007. PMID: 17580844

2

Esters and amides of 6-(chloromethyl)-2-oxo-2H-1-benzopyran-3-carboxylic acid as inhibitors of alpha-chymotrypsin: significance of the "aromatic" nature of the novel ester-type coumarin for strong inhibitory activity.

Pochet L, Doucet C, Schynts M, Thierry N, Boggetto N, Pirotte B, Jiang KY, Masereel B, de Tullio P, Delarge J, Reboud-Ravaux M. Pochet L, et al. J Med Chem. 1996 Jun 21;39(13):2579-85. doi: 10.1021/jm960090b. J Med Chem. 1996. PMID: 8691456

3

Design, synthesis, and anticonvulsant activity of 1-(pyrid-3-ylsulfonamido)-2-nitroethylenes.

Masereel B, Wouters J, Pochet L, Lambert D. Masereel B, et al. Among authors: pochet l. J Med Chem. 1998 Aug 13;41(17):3239-44. doi: 10.1021/jm981022n. J Med Chem. 1998. PMID: 9703469

4

Insulinotropic effect of new glibenclamide isosteres.

Ouedraogo R, Nguyen QA, Kane MH, Dunne MJ, Pochet L, Masereel B, Lebrun P. Ouedraogo R, et al. Among authors: pochet l. J Pharmacol Exp Ther. 1999 May;289(2):625-31. J Pharmacol Exp Ther. 1999. PMID: 10215632

5

Thromboxane A2 receptor antagonism in man and rat by a sulphonylcyanoguanidine (BM-144) and a sulphonylurea (BM-500).

Masereel B, Damas J, Fontaine J, Lembege M, Lacan F, Nuhrich A, Delarge J, Pochet L, Dogne JM. Masereel B, et al. Among authors: pochet l. J Pharm Pharmacol. 1999 Jun;51(6):695-701. doi: 10.1211/0022357991772998. J Pharm Pharmacol. 1999. PMID: 10454046

6

6-Substituted 2-oxo-2H-1-benzopyran-3-carboxylic acid as a core structure for specific inhibitors of human leukocyte elastase.

Doucet C, Pochet L, Thierry N, Pirotte B, Delarge J, Reboud-Ravaux M. Doucet C, et al. Among authors: pochet l. J Med Chem. 1999 Oct 7;42(20):4161-71. doi: 10.1021/jm990070k. J Med Chem. 1999. PMID: 10514286

7

Coumarinic derivatives as mechanism-based inhibitors of alpha-chymotrypsin and human leukocyte elastase.

Pochet L, Doucet C, Dive G, Wouters J, Masereel B, Reboud-Ravaux M, Pirotte B. Pochet L, et al. Bioorg Med Chem. 2000 Jun;8(6):1489-501. doi: 10.1016/s0968-0896(00)00071-7. Bioorg Med Chem. 2000. PMID: 10896125 Free article.

8

Design, synthesis and biological evaluation of a sulfonylcyanoguanidine as thromboxane A2 receptor antagonist and thromboxane synthase inhibitor.

Dogné JM, Wouters J, Rolin S, Michaux C, Pochet L, Durant F, Delarge J, Masereel B. Dogné JM, et al. Among authors: pochet l. J Pharm Pharmacol. 2001 May;53(5):669-80. doi: 10.1211/0022357011775992. J Pharm Pharmacol. 2001. PMID: 11370706

9

Structural approach of the mechanism of inhibition of alpha-chymotrypsin by coumarins.

Wouters J, Huygens M, Pochet L, Pirotte B, Durant F, Masereel B. Wouters J, et al. Among authors: pochet l. Bioorg Med Chem Lett. 2002 Apr 8;12(7):1109-12. doi: 10.1016/s0960-894x(02)00073-2. Bioorg Med Chem Lett. 2002. PMID: 11909728

10

3-Bromophenyl 6-acetoxymethyl-2-oxo-2H-1-benzopyran-3-carboxylate inhibits cancer cell invasion in vitro and tumour growth in vivo.

Kempen I, Papapostolou D, Thierry N, Pochet L, Counerotte S, Masereel B, Foidart JM, Reboud-Ravaux M, Noël A, Pirotte B. Kempen I, et al. Among authors: pochet l. Br J Cancer. 2003 Apr 7;88(7):1111-8. doi: 10.1038/sj.bjc.6600856. Br J Cancer. 2003. PMID: 12671713 Free PMC article.

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