Samuelsson B - Search Results

1

Variations of the P2 group in HIV-1 protease inhibitors containing a tertiary alcohol in the transition-state mimicking scaffold.

Ekegren JK, Gising J, Wallberg H, Larhed M, Samuelsson B, Hallberg A. Ekegren JK, et al. Among authors: samuelsson b. Org Biomol Chem. 2006 Aug 21;4(16):3040-3. doi: 10.1039/b606859f. Epub 2006 Jul 6. Org Biomol Chem. 2006. PMID: 16886068

2

Synthesis, X-ray analysis, and biological evaluation of a new class of stereopure lactam-based HIV-1 protease inhibitors.

Wu X, Ohrngren P, Joshi AA, Trejos A, Persson M, Arvela RK, Wallberg H, Vrang L, Rosenquist A, Samuelsson BB, Unge J, Larhed M. Wu X, et al. Among authors: samuelsson bb. J Med Chem. 2012 Mar 22;55(6):2724-36. doi: 10.1021/jm201620t. Epub 2012 Mar 13. J Med Chem. 2012. PMID: 22376008 Free PMC article.

3

Relationships between structure and interaction kinetics for HIV-1 protease inhibitors.

Markgren PO, Schaal W, Hämäläinen M, Karlén A, Hallberg A, Samuelsson B, Danielson UH. Markgren PO, et al. Among authors: samuelsson b. J Med Chem. 2002 Dec 5;45(25):5430-9. doi: 10.1021/jm0208370. J Med Chem. 2002. PMID: 12459011

4

Cyclic sulfamide HIV-1 protease inhibitors, with sidechains spanning from P2/P2' to P1/P1'.

Ax A, Schaal W, Vrang L, Samuelsson B, Hallberg A, Karlén A. Ax A, et al. Among authors: samuelsson b. Bioorg Med Chem. 2005 Feb 1;13(3):755-64. doi: 10.1016/j.bmc.2004.10.042. Bioorg Med Chem. 2005. PMID: 15653343

5

High-speed synthesis of potent C2-symmetric HIV-1 protease inhibitors by in-situ aminocarbonylations.

Wannberg J, Kaiser NF, Vrang L, Samuelsson B, Larhed M, Hallberg A. Wannberg J, et al. Among authors: samuelsson b. J Comb Chem. 2005 Jul-Aug;7(4):611-7. doi: 10.1021/cc050016r. J Comb Chem. 2005. PMID: 16004505

6

A new class of HIV-1 protease inhibitors containing a tertiary alcohol in the transition-state mimicking scaffold.

Ekegren JK, Unge T, Safa MZ, Wallberg H, Samuelsson B, Hallberg A. Ekegren JK, et al. Among authors: samuelsson b. J Med Chem. 2005 Dec 15;48(25):8098-102. doi: 10.1021/jm050790t. J Med Chem. 2005. PMID: 16335934

7

Microwave-accelerated synthesis of P1'-extended HIV-1 protease inhibitors encompassing a tertiary alcohol in the transition-state mimicking scaffold.

Ekegren JK, Ginman N, Johansson A, Wallberg H, Larhed M, Samuelsson B, Unge T, Hallberg A. Ekegren JK, et al. Among authors: samuelsson b. J Med Chem. 2006 Mar 9;49(5):1828-32. doi: 10.1021/jm051239z. J Med Chem. 2006. PMID: 16509598

8

A new structural theme in C2-symmetric HIV-1 protease inhibitors: ortho-substituted P1/P1' side chains.

Wannberg J, Sabnis YA, Vrang L, Samuelsson B, Karlén A, Hallberg A, Larhed M. Wannberg J, et al. Among authors: samuelsson b. Bioorg Med Chem. 2006 Aug 1;14(15):5303-15. doi: 10.1016/j.bmc.2006.03.045. Epub 2006 Apr 18. Bioorg Med Chem. 2006. PMID: 16621572

9

Two-carbon-elongated HIV-1 protease inhibitors with a tertiary-alcohol-containing transition-state mimic.

Wu X, Ohrngren P, Ekegren JK, Unge J, Unge T, Wallberg H, Samuelsson B, Hallberg A, Larhed M. Wu X, et al. Among authors: samuelsson b. J Med Chem. 2008 Feb 28;51(4):1053-7. doi: 10.1021/jm070680h. Epub 2008 Jan 24. J Med Chem. 2008. PMID: 18215014

10

Design and synthesis of novel P2 substituents in diol-based HIV protease inhibitors.

Adrian Meredith J, Wallberg H, Vrang L, Oscarson S, Parkes K, Hallberg A, Samuelsson B. Adrian Meredith J, et al. Among authors: samuelsson b. Eur J Med Chem. 2010 Jan;45(1):160-70. doi: 10.1016/j.ejmech.2009.09.038. Epub 2009 Oct 6. Eur J Med Chem. 2010. PMID: 19926360

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

679 results

Search Page

Filters