Tran JA - Search Results

1

Propionylpiperazines as human melanocortin-4 receptor ligands.

Chen CW, Tran JA, Jiang W, Tucci FC, Arellano M, Wen J, Fleck BA, Marinkovic D, White NS, Pontillo J, Saunders J, Madan A, Foster AC, Chen C. Chen CW, et al. Among authors: tran ja. Bioorg Med Chem Lett. 2006 Sep 15;16(18):4800-3. doi: 10.1016/j.bmcl.2006.06.075. Epub 2006 Jul 7. Bioorg Med Chem Lett. 2006. PMID: 16824757

2

4-{(2R)-[3-Aminopropionylamido]-3-(2,4-dichlorophenyl)propionyl}-1-{2-[(2-thienyl)ethylaminomethyl]phenyl}piperazine as a potent and selective melanocortin-4 receptor antagonist--design, synthesis, and characterization.

Chen C, Pontillo J, Fleck BA, Gao Y, Wen J, Tran JA, Tucci FC, Marinkovic D, Foster AC, Saunders J. Chen C, et al. Among authors: tran ja. J Med Chem. 2004 Dec 30;47(27):6821-30. doi: 10.1021/jm049278i. J Med Chem. 2004. PMID: 15615531

3

Identification of agonists and antagonists of the human melanocortin-4 receptor from piperazinebenzylamines.

Tran JA, Pontillo J, Arellano M, White NS, Fleck BA, Marinkovic D, Tucci FC, Lanier M, Nelson J, Saunders J, Foster AC, Chen C. Tran JA, et al. Bioorg Med Chem Lett. 2005 Feb 1;15(3):833-7. doi: 10.1016/j.bmcl.2004.10.096. Bioorg Med Chem Lett. 2005. PMID: 15664867

4

Potent and orally active non-peptide antagonists of the human melanocortin-4 receptor based on a series of trans-2-disubstituted cyclohexylpiperazines.

Tucci FC, White NS, Markison S, Joppa M, Tran JA, Fleck BA, Madan A, Dyck BP, Parker J, Pontillo J, Arellano LM, Marinkovic D, Jiang W, Chen CW, Gogas KR, Goodfellow VS, Saunders J, Foster AC, Chen C. Tucci FC, et al. Among authors: tran ja. Bioorg Med Chem Lett. 2005 Oct 1;15(19):4389-95. doi: 10.1016/j.bmcl.2005.06.071. Bioorg Med Chem Lett. 2005. PMID: 16098742

5

Optimization of piperazinebenzylamines with a N-(1-methoxy-2-propyl) side chain as potent and selective antagonists of the human melanocortin-4 receptor.

Pontillo J, Marinkovic D, Tran JA, Arellano M, Fleck BA, Wen J, Tucci FC, Nelson J, Saunders J, Foster AC, Chen C. Pontillo J, et al. Among authors: tran ja. Bioorg Med Chem Lett. 2005 Oct 15;15(20):4615-8. doi: 10.1016/j.bmcl.2005.06.058. Bioorg Med Chem Lett. 2005. PMID: 16105734

6

Structure-activity relationship studies on a series of cyclohexylpiperazines bearing a phanylacetamide as ligands of the human melanocortin-4 receptor.

Pontillo J, Tran JA, White NS, Arellano M, Fleck BA, Marinkovic D, Tucci FC, Saunders J, Foster AC, Chen C. Pontillo J, et al. Among authors: tran ja. Bioorg Med Chem Lett. 2005 Dec 1;15(23):5237-40. doi: 10.1016/j.bmcl.2005.08.061. Epub 2005 Sep 23. Bioorg Med Chem Lett. 2005. PMID: 16183282

7

Design, synthesis, and SAR studies on a series of 2-pyridinylpiperazines as potent antagonists of the melanocortin-4 receptor.

Tran JA, Pontillo J, Fleck BA, Marinkovic D, Arellano M, Tucci FC, Lanier M, Saunders J, Jiang W, Chen CW, Foster AC, Chen C. Tran JA, et al. Bioorg Med Chem Lett. 2006 Jul 15;16(14):3693-6. doi: 10.1016/j.bmcl.2006.04.069. Epub 2006 May 11. Bioorg Med Chem Lett. 2006. PMID: 16697187

8

Arylpropionylpiperazines as antagonists of the human melanocortin-4 receptor.

Jiang W, Tucci FC, Chen CW, Arellano M, Tran JA, White NS, Marinkovic D, Pontillo J, Fleck BA, Wen J, Saunders J, Madan A, Foster AC, Chen C. Jiang W, et al. Among authors: tran ja. Bioorg Med Chem Lett. 2006 Sep 1;16(17):4674-8. doi: 10.1016/j.bmcl.2006.05.088. Epub 2006 Jun 13. Bioorg Med Chem Lett. 2006. PMID: 16777413

9

Pyrrolidinones as orally bioavailable antagonists of the human melanocortin-4 receptor with anti-cachectic activity.

Tran JA, Tucci FC, Jiang W, Marinkovic D, Chen CW, Arellano M, Markison S, Fleck BA, Wen J, White NS, Pontillo J, Saunders J, Marks D, Hoare SR, Madan A, Foster AC, Chen C. Tran JA, et al. Bioorg Med Chem. 2007 Aug 1;15(15):5166-76. doi: 10.1016/j.bmc.2007.05.026. Epub 2007 May 17. Bioorg Med Chem. 2007. PMID: 17544282

10

Pyrrolidines as potent functional agonists of the human melanocortin-4 receptor.

Tran JA, Chen CW, Jiang W, Tucci FC, Fleck BA, Marinkovic D, Arellano M, Chen C. Tran JA, et al. Bioorg Med Chem Lett. 2007 Sep 15;17(18):5165-70. doi: 10.1016/j.bmcl.2007.06.088. Epub 2007 Jul 4. Bioorg Med Chem Lett. 2007. PMID: 17629702

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