Schirmeister T - Search Results

1

A new lead for nonpeptidic active-site-directed inhibitors of the severe acute respiratory syndrome coronavirus main protease discovered by a combination of screening and docking methods.

Kaeppler U, Stiefl N, Schiller M, Vicik R, Breuning A, Schmitz W, Rupprecht D, Schmuck C, Baumann K, Ziebuhr J, Schirmeister T. Kaeppler U, et al. Among authors: schirmeister t. J Med Chem. 2005 Nov 3;48(22):6832-42. doi: 10.1021/jm0501782. J Med Chem. 2005. PMID: 16250642

2

New peptidic cysteine protease inhibitors derived from the electrophilic alpha-amino acid aziridine-2,3-dicarboxylic acid.

Schirmeister T. Schirmeister T. J Med Chem. 1999 Feb 25;42(4):560-72. doi: 10.1021/jm981061z. J Med Chem. 1999. PMID: 10052963

3

Aziridinyl peptides as inhibitors of cysteine proteases: effect of a free carboxylic acid function on inhibition.

Schirmeister T, Peric M. Schirmeister T, et al. Bioorg Med Chem. 2000 Jun;8(6):1281-91. doi: 10.1016/s0968-0896(00)00058-4. Bioorg Med Chem. 2000. PMID: 10896108

4

(S)-Thiirancarboxylic acid as a reactive building block for a new class of cysteine protease inhibitors.

Schirmeister T. Schirmeister T. Bioorg Med Chem Lett. 2000 Dec 4;10(23):2647-51. doi: 10.1016/s0960-894x(00)00549-7. Bioorg Med Chem Lett. 2000. PMID: 11128643

5

Non-peptidic inhibitors of cysteine proteases.

Schirmeister T, Kaeppler U. Schirmeister T, et al. Mini Rev Med Chem. 2003 Jun;3(4):361-73. doi: 10.2174/1389557033488079. Mini Rev Med Chem. 2003. PMID: 12678829 Review.

6

Cysteine protease inhibitors containing small rings.

Schirmeister T, Klockow A. Schirmeister T, et al. Mini Rev Med Chem. 2003 Sep;3(6):585-96. doi: 10.2174/1389557033487935. Mini Rev Med Chem. 2003. PMID: 12871161 Review.

7

Thiirancarboxamides as inhibitors of papain.

Bruno G, Schirmeister T. Bruno G, et al. Among authors: schirmeister t. Arch Pharm (Weinheim). 2004 Feb;337(2):90-5. doi: 10.1002/ardp.200300820. Arch Pharm (Weinheim). 2004. PMID: 14981665

8

Synthesis and antiplasmodial activity of a cysteine protease-inhibiting biotinylated aziridine-2,3-dicarboxylate.

Gelhaus C, Vicik R, Hilgenfeld R, Schmidt CL, Leippe M, Schirmeister T. Gelhaus C, et al. Among authors: schirmeister t. Biol Chem. 2004 May;385(5):435-8. doi: 10.1515/BC.2004.050. Biol Chem. 2004. PMID: 15196005

9

Theoretical studies about the influence of different ring substituents on the nucleophilic ring opening of three-membered heterocycles and possible implications for the mechanisms of cysteine protease inhibitors.

Helten H, Schirmeister T, Engels B. Helten H, et al. Among authors: schirmeister t. J Org Chem. 2005 Jan 7;70(1):233-7. doi: 10.1021/jo048373w. J Org Chem. 2005. PMID: 15624927

10

Blocking effect of a biotinylated protease inhibitor on the egress of Plasmodium falciparum merozoites from infected red blood cells.

Gelhaus C, Vicik R, Schirmeister T, Leippe M. Gelhaus C, et al. Among authors: schirmeister t. Biol Chem. 2005 May;386(5):499-502. doi: 10.1515/BC.2005.059. Biol Chem. 2005. PMID: 15927894

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