Donevan SD - Search Results

1

Novel cyclopropyl beta-amino acid analogues of pregabalin and gabapentin that target the alpha2-delta protein.

Schwarz JB, Gibbons SE, Graham SR, Colbry NL, Guzzo PR, Le VD, Vartanian MG, Kinsora JJ, Lotarski SM, Li Z, Dickerson MR, Su TZ, Weber ML, El-Kattan A, Thorpe AJ, Donevan SD, Taylor CP, Wustrow DJ. Schwarz JB, et al. Among authors: donevan sd. J Med Chem. 2005 Apr 21;48(8):3026-35. doi: 10.1021/jm0491086. J Med Chem. 2005. PMID: 15828841

2

Carboxylate bioisosteres of pregabalin.

Schwarz JB, Colbry NL, Zhu Z, Nichelson B, Barta NS, Lin K, Hudack RA, Gibbons SE, Galatsis P, DeOrazio RJ, Manning DD, Vartanian MG, Kinsora JJ, Lotarski SM, Li Z, Dickerson MR, El-Kattan A, Thorpe AJ, Donevan SD, Taylor CP, Wustrow DJ. Schwarz JB, et al. Among authors: donevan sd. Bioorg Med Chem Lett. 2006 Jul 1;16(13):3559-63. doi: 10.1016/j.bmcl.2006.03.083. Epub 2006 Apr 18. Bioorg Med Chem Lett. 2006. PMID: 16621528

3

Oxadiazolone bioisosteres of pregabalin and gabapentin.

Wustrow DJ, Belliotti TR, Capiris T, Kneen CO, Bryans JS, Field MJ, Williams D, El-Kattan A, Buchholz L, Kinsora JJ, Lotarski SM, Vartanian MG, Taylor CP, Donevan SD, Thorpe AJ, Schwarz JB. Wustrow DJ, et al. Among authors: donevan sd. Bioorg Med Chem Lett. 2009 Jan 1;19(1):247-50. doi: 10.1016/j.bmcl.2008.10.101. Epub 2008 Oct 25. Bioorg Med Chem Lett. 2009. PMID: 19010672

4

Anxiolytic-like activity of pregabalin in the Vogel conflict test in α2δ-1 (R217A) and α2δ-2 (R279A) mouse mutants.

Lotarski SM, Donevan S, El-Kattan A, Osgood S, Poe J, Taylor CP, Offord J. Lotarski SM, et al. J Pharmacol Exp Ther. 2011 Aug;338(2):615-21. doi: 10.1124/jpet.111.180976. Epub 2011 May 10. J Pharmacol Exp Ther. 2011. PMID: 21558437

5

Pregabalin is a potent and selective ligand for α(2)δ-1 and α(2)δ-2 calcium channel subunits.

Li Z, Taylor CP, Weber M, Piechan J, Prior F, Bian F, Cui M, Hoffman D, Donevan S. Li Z, et al. Eur J Pharmacol. 2011 Sep 30;667(1-3):80-90. doi: 10.1016/j.ejphar.2011.05.054. Epub 2011 Jun 1. Eur J Pharmacol. 2011. PMID: 21651903

6

Ca2+ channel alpha2delta ligands: novel modulators of neurotransmission.

Dooley DJ, Taylor CP, Donevan S, Feltner D. Dooley DJ, et al. Trends Pharmacol Sci. 2007 Feb;28(2):75-82. doi: 10.1016/j.tips.2006.12.006. Epub 2007 Jan 10. Trends Pharmacol Sci. 2007. PMID: 17222465 Review.

7

Anticonvulsant activity of pregabalin in the maximal electroshock-induced seizure assay in α2δ1 (R217A) and α2δ2 (R279A) mouse mutants.

Lotarski S, Hain H, Peterson J, Galvin S, Strenkowski B, Donevan S, Offord J. Lotarski S, et al. Epilepsy Res. 2014 Jul;108(5):833-42. doi: 10.1016/j.eplepsyres.2014.03.002. Epub 2014 Mar 21. Epilepsy Res. 2014. PMID: 24698052

8

How modeling and simulation have enhanced decision making in new drug development.

Miller R, Ewy W, Corrigan BW, Ouellet D, Hermann D, Kowalski KG, Lockwood P, Koup JR, Donevan S, El-Kattan A, Li CS, Werth JL, Feltner DE, Lalonde RL. Miller R, et al. J Pharmacokinet Pharmacodyn. 2005 Apr;32(2):185-97. doi: 10.1007/s10928-005-0074-7. Epub 2005 Nov 7. J Pharmacokinet Pharmacodyn. 2005. PMID: 16283534 Review.

9

Central sensitization and Ca(V)α₂δ ligands in chronic pain syndromes: pathologic processes and pharmacologic effect.

Tuchman M, Barrett JA, Donevan S, Hedberg TG, Taylor CP. Tuchman M, et al. J Pain. 2010 Dec;11(12):1241-9. doi: 10.1016/j.jpain.2010.02.024. Epub 2010 May 15. J Pain. 2010. PMID: 20472509 Free article. Review.

10

Voltage-dependent block of N-methyl-D-aspartate receptors by the novel anticonvulsant dibenzylamine, a bioactive constituent of L-(+)-beta-hydroxybutyrate.

Donevan SD, White HS, Anderson GD, Rho JM. Donevan SD, et al. Epilepsia. 2003 Oct;44(10):1274-9. doi: 10.1046/j.1528-1157.2003.07203.x. Epilepsia. 2003. PMID: 14510820 Free article.

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