Venet M - Search Results

1

Synthesis, structure-activity relationship, and receptor pharmacology of a new series of quinoline derivatives acting as selective, noncompetitive mGlu1 antagonists.

Mabire D, Coupa S, Adelinet C, Poncelet A, Simonnet Y, Venet M, Wouters R, Lesage AS, Van Beijsterveldt L, Bischoff F. Mabire D, et al. Among authors: venet m. J Med Chem. 2005 Mar 24;48(6):2134-53. doi: 10.1021/jm049499o. J Med Chem. 2005. PMID: 15771457

2

5-imidazolyl-quinolinones, -quinazolinones and -benzo-azepinones as farnesyltransferase inhibitors.

Angibaud P, Bourdrez X, Devine A, End DW, Freyne E, Ligny Y, Muller P, Mannens G, Pilatte I, Poncelet V, Skrzat S, Smets G, Van Dun J, Van Remoortere P, Venet M, Wouters W. Angibaud P, et al. Among authors: venet m. Bioorg Med Chem Lett. 2003 May 5;13(9):1543-7. doi: 10.1016/s0960-894x(03)00180-x. Bioorg Med Chem Lett. 2003. PMID: 12699751

3

4-methyl-1,2,4-triazol-3-yl heterocycle as an alternative to the 1-methylimidazol-5-yl moiety in the farnesyltransferase inhibitor ZARNESTRA.

Angibaud P, Saha AK, Bourdrez X, End DW, Freyne E, Lezouret P, Mannens G, Mevellec L, Meyer C, Pilatte I, Poncelet V, Roux B, Smets G, Van Dun J, Venet M, Wouters W. Angibaud P, et al. Among authors: venet m. Bioorg Med Chem Lett. 2003 Dec 15;13(24):4361-4. doi: 10.1016/j.bmcl.2003.09.043. Bioorg Med Chem Lett. 2003. PMID: 14643326

4

Substituted azoloquinolines and -quinazolines as new potent farnesyl protein transferase inhibitors.

Angibaud P, Bourdrez X, End DW, Freyne E, Janicot M, Lezouret P, Ligny Y, Mannens G, Damsch S, Mevellec L, Meyer C, Muller P, Pilatte I, Poncelet V, Roux B, Smets G, Van Dun J, Van Remoortere P, Venet M, Wouters W. Angibaud P, et al. Among authors: venet m. Bioorg Med Chem Lett. 2003 Dec 15;13(24):4365-9. doi: 10.1016/j.bmcl.2003.08.080. Bioorg Med Chem Lett. 2003. PMID: 14643327

5

Impact on farnesyltransferase inhibition of 4-chlorophenyl moiety replacement in the Zarnestra series.

Angibaud P, Mevellec L, Meyer C, Bourdrez X, Lezouret P, Pilatte I, Poncelet V, Roux B, Merillon S, End DW, Van Dun J, Wouters W, Venet M. Angibaud P, et al. Among authors: venet m. Eur J Med Chem. 2007 May;42(5):702-14. doi: 10.1016/j.ejmech.2006.12.007. Epub 2007 Jan 9. Eur J Med Chem. 2007. PMID: 17316920

6

Farnesyl protein transferase inhibitor ZARNESTRA R115777 - history of a discovery.

Venet M, End D, Angibaud P. Venet M, et al. Curr Top Med Chem. 2003;3(10):1095-102. doi: 10.2174/1568026033452050. Curr Top Med Chem. 2003. PMID: 12769710 Review.

7

Synthesis of LIAZAL, a retinoic acid metabolism blocking agent (RAMBA) with potential clinical applications in oncology and dermatology.

Freyne E, Raeymaekers A, Venet M, Sanz G, Wouters W, De Coster R, Wauwe JV. Freyne E, et al. Among authors: venet m. Bioorg Med Chem Lett. 1998 Feb 3;8(3):267-72. doi: 10.1016/s0960-894x(98)00004-3. Bioorg Med Chem Lett. 1998. PMID: 9871667

8

Inhibition of all-TRANS-retinoic acid metabolism by R116010 induces antitumour activity.

Van Heusden J, Van Ginckel R, Bruwiere H, Moelans P, Janssen B, Floren W, van der Leede BJ, van Dun J, Sanz G, Venet M, Dillen L, Van Hove C, Willemsens G, Janicot M, Wouters W. Van Heusden J, et al. Among authors: venet m. Br J Cancer. 2002 Feb 12;86(4):605-11. doi: 10.1038/sj.bjc.6600056. Br J Cancer. 2002. PMID: 11870544 Free PMC article.

9

Characterization of the antitumor effects of the selective farnesyl protein transferase inhibitor R115777 in vivo and in vitro.

End DW, Smets G, Todd AV, Applegate TL, Fuery CJ, Angibaud P, Venet M, Sanz G, Poignet H, Skrzat S, Devine A, Wouters W, Bowden C. End DW, et al. Among authors: venet m. Cancer Res. 2001 Jan 1;61(1):131-7. Cancer Res. 2001. PMID: 11196150

10

Comparative effects of the aromatase inhibitor R76713 and of its enantiomers R83839 and R83842 on steroid biosynthesis in vitro and in vivo.

Wouters W, De Coster R, van Dun J, Krekels MD, Dillen A, Raeymaekers A, Freyne E, Van Gelder J, Sanz G, Venet M, et al. Wouters W, et al. Among authors: venet m. J Steroid Biochem Mol Biol. 1990 Dec 20;37(6):1049-54. doi: 10.1016/0960-0760(90)90464-v. J Steroid Biochem Mol Biol. 1990. PMID: 2178362

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