Curtis MP - Search Results

1

D-amino acid homopiperazine amides: discovery of A-320436, a potent and selective non-imidazole histamine H(3)-receptor antagonist.

Curtis MP, Dwight W, Pratt J, Cowart M, Esbenshade TA, Krueger KM, Fox GB, Pan JB, Pagano TG, Hancock AA, Faghih R, Bennani YL. Curtis MP, et al. Arch Pharm (Weinheim). 2004 Apr;337(4):219-29. doi: 10.1002/ardp.200300844. Arch Pharm (Weinheim). 2004. PMID: 15146898

2

Synthesis and SAR of 5-amino- and 5-(aminomethyl)benzofuran histamine H3 receptor antagonists with improved potency.

Sun M, Zhao C, Gfesser GA, Thiffault C, Miller TR, Marsh K, Wetter J, Curtis M, Faghih R, Esbenshade TA, Hancock AA, Cowart M. Sun M, et al. J Med Chem. 2005 Oct 6;48(20):6482-90. doi: 10.1021/jm0504398. J Med Chem. 2005. PMID: 16190774

3

4-(2-[2-(2(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl)benzonitrile and related 2-aminoethylbenzofuran H3 receptor antagonists potently enhance cognition and attention.

Cowart M, Faghih R, Curtis MP, Gfesser GA, Bennani YL, Black LA, Pan L, Marsh KC, Sullivan JP, Esbenshade TA, Fox GB, Hancock AA. Cowart M, et al. Among authors: curtis mp. J Med Chem. 2005 Jan 13;48(1):38-55. doi: 10.1021/jm040118g. J Med Chem. 2005. PMID: 15634000

4

The medicinal chemistry of novel H(3) antagonists.

Cowart M, Faghih R, Gfesser G, Curtis M, Pratt JK, Bennani Y, Fox GB, Esbenshade TA, Hancock AA. Cowart M, et al. Inflamm Res. 2004 Mar;53 Suppl 1:S69-70. doi: 10.1007/s00011-003-0333-2. Epub 2004 Mar 5. Inflamm Res. 2004. PMID: 15054624 No abstract available.

5

Structure-activity relationships of arylbenzofuran H3 receptor antagonists.

Gfesser GA, Faghih R, Bennani YL, Curtis MP, Esbenshade TA, Hancock AA, Cowart MD. Gfesser GA, et al. Among authors: curtis mp. Bioorg Med Chem Lett. 2005 May 16;15(10):2559-63. doi: 10.1016/j.bmcl.2005.03.047. Bioorg Med Chem Lett. 2005. PMID: 15863316

6

Achievement of behavioral efficacy and improved potency in new heterocyclic analogs of benzofuran H3 antagonists.

Cowart M, Faghih R, Gfesser G, Curtis M, Sun M, Zhao C, Bennani Y, Wetter J, Marsh K, Miller TR, Krueger K, Pan JB, Drescher K, Fox GB, Esbenshade TA, Hancock AA. Cowart M, et al. Inflamm Res. 2005 Apr;54 Suppl 1:S25-6. doi: 10.1007/s00011-004-0411-0. Inflamm Res. 2005. PMID: 15928820 No abstract available.

7

Discovery of 4-(5-(4-chlorophenyl)-2-methyl-3-propionyl-1H-pyrrol-1-yl)benzenesulfonamide (A-867744) as a novel positive allosteric modulator of the alpha7 nicotinic acetylcholine receptor.

Faghih R, Gopalakrishnan SM, Gronlien JH, Malysz J, Briggs CA, Wetterstrand C, Ween H, Curtis MP, Sarris KA, Gfesser GA, El-Kouhen R, Robb HM, Radek RJ, Marsh KC, Bunnelle WH, Gopalakrishnan M. Faghih R, et al. Among authors: curtis mp. J Med Chem. 2009 May 28;52(10):3377-84. doi: 10.1021/jm9003818. J Med Chem. 2009. PMID: 19419141

8

Tricyclic aminopyrimidine histamine H4 receptor antagonists.

Savall BM, Gomez L, Chavez F, Curtis M, Meduna SP, Kearney A, Dunford P, Cowden J, Thurmond RL, Grice C, Edwards JP. Savall BM, et al. Bioorg Med Chem Lett. 2011 Nov 1;21(21):6577-81. doi: 10.1016/j.bmcl.2011.08.014. Epub 2011 Aug 19. Bioorg Med Chem Lett. 2011. PMID: 21920744

9

The discovery of isoxazoline oxime ethers as a new class of ectoparasiticides for the control of Haematobia irritans (horn fly) in cattle.

Curtis MP, Chubb N, Ellsworth E, Goodwin R, Holzmer S, Koch J, McTier T, Menon S, Mills K, Pullins A, Stuk T, Zinser E. Curtis MP, et al. Bioorg Med Chem Lett. 2014 Nov 1;24(21):5011-4. doi: 10.1016/j.bmcl.2014.09.023. Epub 2014 Sep 16. Bioorg Med Chem Lett. 2014. PMID: 25278232

10

Design and synthesis of sarolaner, a novel, once-a-month, oral isoxazoline for the control of fleas and ticks on dogs.

Curtis MP, Vaillancourt V, Goodwin RM, Chubb NA, Howson W, McTier TL, Pullins A, Zinser EW, Meeus PF, Woods DJ, Hedges L, Stuk T, Price JE, Koch JD, Menon SR. Curtis MP, et al. Bioorg Med Chem Lett. 2016 Apr 1;26(7):1831-5. doi: 10.1016/j.bmcl.2016.02.027. Epub 2016 Feb 12. Bioorg Med Chem Lett. 2016. PMID: 26920802

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