Kelley JA - Search Results

1

Macrocyclization in the design of non-phosphorus-containing Grb2 SH2 domain-binding ligands.

Shi ZD, Wei CQ, Lee K, Liu H, Zhang M, Araki T, Roberts LR, Worthy KM, Fisher RJ, Neel BG, Kelley JA, Yang D, Burke TR Jr. Shi ZD, et al. Among authors: kelley ja. J Med Chem. 2004 Apr 8;47(8):2166-9. doi: 10.1021/jm030510e. J Med Chem. 2004. PMID: 15056012

2

Potent inhibition of Grb2 SH2 domain binding by non-phosphate-containing ligands.

Yao ZJ, King CR, Cao T, Kelley J, Milne GW, Voigt JH, Burke TR Jr. Yao ZJ, et al. J Med Chem. 1999 Jan 14;42(1):25-35. doi: 10.1021/jm980388x. J Med Chem. 1999. PMID: 9888830

3

Inhibition of Grb2 SH2 domain binding by non-phosphate-containing ligands. 2. 4-(2-Malonyl)phenylalanine as a potent phosphotyrosyl mimetic.

Gao Y, Luo J, Yao ZJ, Guo R, Zou H, Kelley J, Voigt JH, Yang D, Burke TR Jr. Gao Y, et al. J Med Chem. 2000 Mar 9;43(5):911-20. doi: 10.1021/jm9904248. J Med Chem. 2000. PMID: 10715157

4

Enantioselective synthesis of N(alpha)-Fmoc protected (2S,3R)-3-phenylpipecolic acid. A constrained phenylalanine analogue suitably protected for solid-phase peptide synthesis.

Liu DG, Gao Y, Wang X, Kelley JA, Burke TR Jr. Liu DG, et al. Among authors: kelley ja. J Org Chem. 2002 Mar 8;67(5):1448-52. doi: 10.1021/jo010124+. J Org Chem. 2002. PMID: 11871872

5

Design and synthesis of Fmoc-Thr[PO(OH)(OPOM)] for the preparation of peptide prodrugs containing phosphothreonine in fully protected form.

Qian WJ, Lai CC, Kelley JA, Burke TR Jr. Qian WJ, et al. Among authors: kelley ja. Chem Biodivers. 2014 May;11(5):784-91. doi: 10.1002/cbdv.201300202. Chem Biodivers. 2014. PMID: 24827688 Free PMC article.

6

Mono-anionic phosphopeptides produced by unexpected histidine alkylation exhibit high Plk1 polo-box domain-binding affinities and enhanced antiproliferative effects in HeLa cells.

Qian WJ, Park JE, Lim D, Lai CC, Kelley JA, Park SY, Lee KW, Yaffe MB, Lee KS, Burke TR Jr. Qian WJ, et al. Among authors: kelley ja. Biopolymers. 2014 Nov;102(6):444-55. doi: 10.1002/bip.22569. Biopolymers. 2014. PMID: 25283071 Free PMC article.

7

Synthesis and biological study of a flavone acetic acid analogue containing an azido reporting group designed as a multifunctional binding site probe.

Malolanarasimhan K, Lai CC, Kelley JA, Iaccarino L, Reynolds D, Young HA, Marquez VE. Malolanarasimhan K, et al. Among authors: kelley ja. Bioorg Med Chem. 2005 Apr 15;13(8):2717-22. doi: 10.1016/j.bmc.2005.02.035. Bioorg Med Chem. 2005. PMID: 15781383

8

Neighbor-directed histidine N (τ)-alkylation: A route to imidazolium-containing phosphopeptide macrocycles.

Qian WJ, Park JE, Grant R, Lai CC, Kelley JA, Yaffe MB, Lee KS, Burke TR Jr. Qian WJ, et al. Among authors: kelley ja. Biopolymers. 2015 Nov;104(6):663-73. doi: 10.1002/bip.22698. Biopolymers. 2015. PMID: 26152807 Free PMC article.

9

Conformationally constrained analogues of diacylglycerol (DAG). 27. Modulation of membrane translocation of protein kinase C (PKC) isozymes alpha and delta by diacylglycerol lactones (DAG-lactones) containing rigid-rod acyl groups.

Malolanarasimhan K, Kedei N, Sigano DM, Kelley JA, Lai CC, Lewin NE, Surawski RJ, Pavlyukovets VA, Garfield SH, Wincovitch S, Blumberg PM, Marquez VE. Malolanarasimhan K, et al. Among authors: kelley ja. J Med Chem. 2007 Mar 8;50(5):962-78. doi: 10.1021/jm061289j. Epub 2007 Feb 7. J Med Chem. 2007. PMID: 17284021

10

Conformationally constrained analogues of diacylglycerol. 29. Cells sort diacylglycerol-lactone chemical zip codes to produce diverse and selective biological activities.

Duan D, Sigano DM, Kelley JA, Lai CC, Lewin NE, Kedei N, Peach ML, Lee J, Abeyweera TP, Rotenberg SA, Kim H, Kim YH, El Kazzouli S, Chung JU, Young HA, Young MR, Baker A, Colburn NH, Haimovitz-Friedman A, Truman JP, Parrish DA, Deschamps JR, Perry NA, Surawski RJ, Blumberg PM, Marquez VE. Duan D, et al. Among authors: kelley ja. J Med Chem. 2008 Sep 11;51(17):5198-220. doi: 10.1021/jm8001907. Epub 2008 Aug 13. J Med Chem. 2008. PMID: 18698758 Free PMC article.

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