Peiper SC - Search Results

1

Enhancement of the T140-based pharmacophores leads to the development of more potent and bio-stable CXCR4 antagonists.

Tamamura H, Hiramatsu K, Mizumoto M, Ueda S, Kusano S, Terakubo S, Akamatsu M, Yamamoto N, Trent JO, Wang Z, Peiper SC, Nakashima H, Otaka A, Fujii N. Tamamura H, et al. Among authors: peiper sc. Org Biomol Chem. 2003 Nov 7;1(21):3663-9. doi: 10.1039/b306613b. Org Biomol Chem. 2003. PMID: 14649897

2

Molecular-size reduction of a potent CXCR4-chemokine antagonist using orthogonal combination of conformation- and sequence-based libraries.

Fujii N, Oishi S, Hiramatsu K, Araki T, Ueda S, Tamamura H, Otaka A, Kusano S, Terakubo S, Nakashima H, Broach JA, Trent JO, Wang ZX, Peiper SC. Fujii N, et al. Among authors: peiper sc. Angew Chem Int Ed Engl. 2003 Jul 21;42(28):3251-3. doi: 10.1002/anie.200351024. Angew Chem Int Ed Engl. 2003. PMID: 12876735 No abstract available.

3

Synthesis of potent CXCR4 inhibitors possessing low cytotoxicity and improved biostability based on T140 derivatives.

Tamamura H, Hiramatsu K, Kusano aS, Terakubo S, Yamamoto N, Trent JO, Wang Z, Peiper SC, Nakashima H, Otaka A, Fujii N. Tamamura H, et al. Among authors: peiper sc. Org Biomol Chem. 2003 Nov 7;1(21):3656-62. doi: 10.1039/b306473p. Org Biomol Chem. 2003. PMID: 14649896

4

Topochemical exploration of potent compounds using retro-enantiomer libraries of cyclic pentapeptides.

Tamamura H, Mizumoto M, Hiramatsu K, Kusano S, Terakubo S, Yamamoto N, Trent JO, Wang Z, Peiper SC, Nakashima H, Otaka A, Fujii N. Tamamura H, et al. Among authors: peiper sc. Org Biomol Chem. 2004 Apr 21;2(8):1255-7. doi: 10.1039/b401485p. Epub 2004 Mar 23. Org Biomol Chem. 2004. PMID: 15064805

5

Stereoselective synthesis of [L-Arg-L/D-3-(2-naphthyl)alanine]-type (E)-alkene dipeptide isosteres and its application to the synthesis and biological evaluation of pseudopeptide analogues of the CXCR4 antagonist FC131.

Tamamura H, Hiramatsu K, Ueda S, Wang Z, Kusano S, Terakubo S, Trent JO, Peiper SC, Yamamoto N, Nakashima H, Otaka A, Fujii N. Tamamura H, et al. Among authors: peiper sc. J Med Chem. 2005 Jan 27;48(2):380-91. doi: 10.1021/jm049429h. J Med Chem. 2005. PMID: 15658852

6

Identification of novel low molecular weight CXCR4 antagonists by structural tuning of cyclic tetrapeptide scaffolds.

Tamamura H, Araki T, Ueda S, Wang Z, Oishi S, Esaka A, Trent JO, Nakashima H, Yamamoto N, Peiper SC, Otaka A, Fujii N. Tamamura H, et al. Among authors: peiper sc. J Med Chem. 2005 May 5;48(9):3280-9. doi: 10.1021/jm050009h. J Med Chem. 2005. PMID: 15857134

7

Structure-activity relationship studies on CXCR4 antagonists having cyclic pentapeptide scaffolds.

Tamamura H, Esaka A, Ogawa T, Araki T, Ueda S, Wang Z, Trent JO, Tsutsumi H, Masuno H, Nakashima H, Yamamoto N, Peiper SC, Otaka A, Fujii N. Tamamura H, et al. Among authors: peiper sc. Org Biomol Chem. 2005 Dec 21;3(24):4392-4. doi: 10.1039/b513145f. Epub 2005 Nov 15. Org Biomol Chem. 2005. PMID: 16327900

8

Stereoselective synthesis of 3,6-disubstituted-3,6-dihydropyridin-2-ones as potential diketopiperazine mimetics using organocopper-mediated anti-SN2' reactions and their use in the preparation of low-molecule CXCR4 antagonists.

Niida A, Tanigaki H, Inokuchi E, Sasaki Y, Oishi S, Ohno H, Tamamura H, Wang Z, Peiper SC, Kitaura K, Otaka A, Fujii N. Niida A, et al. Among authors: peiper sc. J Org Chem. 2006 May 12;71(10):3942-51. doi: 10.1021/jo060390t. J Org Chem. 2006. PMID: 16674071

9

Development of a linear type of low molecular weight CXCR4 antagonists based on T140 analogs.

Tamamura H, Tsutsumi H, Masuno H, Mizokami S, Hiramatsu K, Wang Z, Trent JO, Nakashima H, Yamamoto N, Peiper SC, Fujii N. Tamamura H, et al. Among authors: peiper sc. Org Biomol Chem. 2006 Jun 21;4(12):2354-7. doi: 10.1039/b603818b. Epub 2006 May 12. Org Biomol Chem. 2006. PMID: 16763678

10

Structure-activity relationships of cyclic peptide-based chemokine receptor CXCR4 antagonists: disclosing the importance of side-chain and backbone functionalities.

Ueda S, Oishi S, Wang ZX, Araki T, Tamamura H, Cluzeau J, Ohno H, Kusano S, Nakashima H, Trent JO, Peiper SC, Fujii N. Ueda S, et al. Among authors: peiper sc. J Med Chem. 2007 Jan 25;50(2):192-8. doi: 10.1021/jm0607350. J Med Chem. 2007. PMID: 17228861

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