Jacobson KA - Search Results

1

Molecular modeling of adenosine receptors. I. The ligand binding site on the A1 receptor.

IJzerman AP, Van Galen PJ, Jacobson KA. IJzerman AP, et al. Among authors: jacobson ka. Drug Des Discov. 1992;9(1):49-67. Drug Des Discov. 1992. PMID: 1457698 Free PMC article.

2

A1 adenosine-receptor antagonists activate chloride efflux from cystic fibrosis cells.

Eidelman O, Guay-Broder C, van Galen PJ, Jacobson KA, Fox C, Turner RJ, Cabantchik ZI, Pollard HB. Eidelman O, et al. Among authors: jacobson ka. Proc Natl Acad Sci U S A. 1992 Jun 15;89(12):5562-6. doi: 10.1073/pnas.89.12.5562. Proc Natl Acad Sci U S A. 1992. PMID: 1376923 Free PMC article.

3

Synthesis and biological activity of N6-(p-sulfophenyl)alkyl and N6-sulfoalkyl derivatives of adenosine: water-soluble and peripherally selective adenosine agonists.

Jacobson KA, Nikodijevic O, Ji XD, Berkich DA, Eveleth D, Dean RL, Hiramatsu K, Kassell NF, van Galen PJ, Lee KS, et al. Jacobson KA, et al. J Med Chem. 1992 Oct 30;35(22):4143-9. doi: 10.1021/jm00100a020. J Med Chem. 1992. PMID: 1433217 Free PMC article.

4

Adenosine A1 and A2 receptors: structure--function relationships.

van Galen PJ, Stiles GL, Michaels G, Jacobson KA. van Galen PJ, et al. Among authors: jacobson ka. Med Res Rev. 1992 Sep;12(5):423-71. doi: 10.1002/med.2610120502. Med Res Rev. 1992. PMID: 1513184 Free PMC article. Review. No abstract available.

5

Characterization of human striatal A2-adenosine receptors using radioligand binding and photoaffinity labeling.

Ji XD, Stiles GL, van Galen PJ, Jacobson KA. Ji XD, et al. Among authors: jacobson ka. J Recept Res. 1992;12(2):149-69. doi: 10.3109/10799899209074789. J Recept Res. 1992. PMID: 1583620 Free PMC article.

6

Adenosine receptors: pharmacology, structure-activity relationships, and therapeutic potential.

Jacobson KA, van Galen PJ, Williams M. Jacobson KA, et al. J Med Chem. 1992 Feb 7;35(3):407-22. doi: 10.1021/jm00081a001. J Med Chem. 1992. PMID: 1738138 Free PMC article. Review. No abstract available.

7

Trifunctional agents as a design strategy for tailoring ligand properties: irreversible inhibitors of A1 adenosine receptors.

Boring DL, Ji XD, Zimmet J, Taylor KE, Stiles GL, Jacobson KA. Boring DL, et al. Among authors: jacobson ka. Bioconjug Chem. 1991 Mar-Apr;2(2):77-88. doi: 10.1021/bc00008a002. Bioconjug Chem. 1991. PMID: 1868116 Free PMC article.

8

Electrophilic derivatives of purines as irreversible inhibitors of A1 adenosine receptors.

Jacobson KA, Barone S, Kammula U, Stiles GL. Jacobson KA, et al. J Med Chem. 1989 May;32(5):1043-51. doi: 10.1021/jm00125a019. J Med Chem. 1989. PMID: 2709373 Free PMC article.

9

Sulfur-containing 1,3-dialkylxanthine derivatives as selective antagonists at A1-adenosine receptors.

Jacobson KA, Kiriasis L, Barone S, Bradbury BJ, Kammula U, Campagne JM, Secunda S, Daly JW, Neumeyer JL, Pfleiderer W. Jacobson KA, et al. J Med Chem. 1989 Aug;32(8):1873-9. doi: 10.1021/jm00128a031. J Med Chem. 1989. PMID: 2754711 Free PMC article.

10

8-Substituted xanthines as antagonists at A1- and A2-adenosine receptors.

Jacobson KA, de la Cruz R, Schulick R, Kiriasis L, Padgett W, Pfleiderer W, Kirk KL, Neumeyer JL, Daly JW. Jacobson KA, et al. Biochem Pharmacol. 1988 Oct 1;37(19):3653-61. doi: 10.1016/0006-2952(88)90398-x. Biochem Pharmacol. 1988. PMID: 3178879 Free PMC article.

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