Chibale K - Search Results

1

Synthesis and evaluation of isatins and thiosemicarbazone derivatives against cruzain, falcipain-2 and rhodesain.

Chiyanzu I, Hansell E, Gut J, Rosenthal PJ, McKerrow JH, Chibale K. Chiyanzu I, et al. Among authors: chibale k. Bioorg Med Chem Lett. 2003 Oct 20;13(20):3527-30. doi: 10.1016/s0960-894x(03)00756-x. Bioorg Med Chem Lett. 2003. PMID: 14505663

2

Synthesis and evaluation of 9,9-dimethylxanthene tricyclics against trypanothione reductase, Trypanosoma brucei, Trypanosoma cruzi and Leishmania donovani.

Chibale K, Visser M, Yardley V, Croft SL, Fairlamb AH. Chibale K, et al. Bioorg Med Chem Lett. 2000 Jun 5;10(11):1147-50. doi: 10.1016/s0960-894x(00)00154-2. Bioorg Med Chem Lett. 2000. PMID: 10866368

3

Modulation of human mammary cell sensitivity to paclitaxel by new quinoline sulfonamides.

Chibale K, Ojima I, Haupt H, Geng X, Pera P, Bernacki RJ. Chibale K, et al. Bioorg Med Chem Lett. 2001 Sep 17;11(18):2457-60. doi: 10.1016/s0960-894x(01)00462-0. Bioorg Med Chem Lett. 2001. PMID: 11549446

4

Antiprotozoal and cytotoxicity evaluation of sulfonamide and urea analogues of quinacrine.

Chibale K, Haupt H, Kendrick H, Yardley V, Saravanamuthu A, Fairlamb AH, Croft SL. Chibale K, et al. Bioorg Med Chem Lett. 2001 Oct 8;11(19):2655-7. doi: 10.1016/s0960-894x(01)00528-5. Bioorg Med Chem Lett. 2001. PMID: 11551771

5

Synthesis of totarol amino alcohol derivatives and their antiplasmodial activity and cytotoxicity.

Clarkson C, Musonda CC, Chibale K, Campbell WE, Smith P. Clarkson C, et al. Among authors: chibale k. Bioorg Med Chem. 2003 Oct 1;11(20):4417-22. doi: 10.1016/s0968-0896(03)00491-7. Bioorg Med Chem. 2003. PMID: 13129578

6

Synthesis and structure-activity relationships of parasiticidal thiosemicarbazone cysteine protease inhibitors against Plasmodium falciparum, Trypanosoma brucei, and Trypanosoma cruzi.

Greenbaum DC, Mackey Z, Hansell E, Doyle P, Gut J, Caffrey CR, Lehrman J, Rosenthal PJ, McKerrow JH, Chibale K. Greenbaum DC, et al. Among authors: chibale k. J Med Chem. 2004 Jun 3;47(12):3212-9. doi: 10.1021/jm030549j. J Med Chem. 2004. PMID: 15163200

7

Application of multi-component reactions to antimalarial drug discovery. Part 1: Parallel synthesis and antiplasmodial activity of new 4-aminoquinoline Ugi adducts.

Musonda CC, Taylor D, Lehman J, Gut J, Rosenthal PJ, Chibale K. Musonda CC, et al. Among authors: chibale k. Bioorg Med Chem Lett. 2004 Aug 2;14(15):3901-5. doi: 10.1016/j.bmcl.2004.05.063. Bioorg Med Chem Lett. 2004. PMID: 15225694

8

Application of combinatorial and parallel synthesis chemistry methodologies to antiparasitic drug discovery.

Musonda CC, Chibale K. Musonda CC, et al. Among authors: chibale k. Curr Med Chem. 2004 Oct;11(19):2519-33. doi: 10.2174/0929867043364469. Curr Med Chem. 2004. PMID: 15544460 Review.

9

Design, synthesis and anti-plasmodial evaluation in vitro of new 4-aminoquinoline isatin derivatives.

Chiyanzu I, Clarkson C, Smith PJ, Lehman J, Gut J, Rosenthal PJ, Chibale K. Chiyanzu I, et al. Among authors: chibale k. Bioorg Med Chem. 2005 May 2;13(9):3249-61. doi: 10.1016/j.bmc.2005.02.037. Bioorg Med Chem. 2005. PMID: 15809160

10

Exploiting a basic chemosensitizing pharmacophore hypothesis. Part 1: synthesis and biological evaluation of novel arylbromide and bicyclic chemosensitizers against drug-resistant malaria parasites.

Chouteau F, Ramanitrahasimbola D, Rasoanaivo P, Chibale K. Chouteau F, et al. Among authors: chibale k. Bioorg Med Chem Lett. 2005 Jun 15;15(12):3024-8. doi: 10.1016/j.bmcl.2005.04.033. Bioorg Med Chem Lett. 2005. PMID: 15908208

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

293 results

Search Page

Filters