Krogsgaard-Larsen P - Search Results

1

Design and synthesis of a new series of 4-alkylated 3-isoxazolol GABA A antagonists.

Frølund B, Tagmose L, Jørgensen AT, Kristiansen U, Stensbøl TB, Liljefors T, Krogsgaard-Larsen P. Frølund B, et al. Eur J Med Chem. 2003 Apr;38(4):447-9. doi: 10.1016/s0223-5234(03)00056-4. Eur J Med Chem. 2003. PMID: 12750034

2

Novel 1-hydroxyazole bioisosteres of glutamic acid. Synthesis, protolytic properties, and pharmacology.

Stensbøl TB, Uhlmann P, Morel S, Eriksen BL, Felding J, Kromann H, Hermit MB, Greenwood JR, Braüner-Osborne H, Madsen U, Junager F, Krogsgaard-Larsen P, Begtrup M, Vedsø P. Stensbøl TB, et al. J Med Chem. 2002 Jan 3;45(1):19-31. doi: 10.1021/jm010303j. J Med Chem. 2002. PMID: 11754576

3

Selective antagonists at group I metabotropic glutamate receptors: synthesis and molecular pharmacology of 4-aryl-3-isoxazolol amino acids.

Kromann H, Sløk FA, Stensbøl TB, Bräuner-Osborne H, Madsen U, Krogsgaard-Larsen P. Kromann H, et al. J Med Chem. 2002 Feb 14;45(4):988-91. doi: 10.1021/jm010443t. J Med Chem. 2002. PMID: 11831912

4

Novel class of potent 4-arylalkyl substituted 3-isoxazolol GABA(A) antagonists: synthesis, pharmacology, and molecular modeling.

Frølund B, Jørgensen AT, Tagmose L, Stensbøl TB, Vestergaard HT, Engblom C, Kristiansen U, Sanchez C, Krogsgaard-Larsen P, Liljefors T. Frølund B, et al. J Med Chem. 2002 Jun 6;45(12):2454-68. doi: 10.1021/jm020027o. J Med Chem. 2002. PMID: 12036354

5

GABA(A) receptor ligands and their therapeutic potentials.

Frølund B, Ebert B, Kristiansen U, Liljefors T, Krogsgaard-Larsen P. Frølund B, et al. Curr Top Med Chem. 2002 Aug;2(8):817-32. doi: 10.2174/1568026023393525. Curr Top Med Chem. 2002. PMID: 12171573 Review.

6

Selective agonists at group II metabotropic glutamate receptors: synthesis, stereochemistry, and molecular pharmacology of (S)- and (R)-2-amino-4-(4-hydroxy[1,2,5]thiadiazol-3-yl)butyric acid.

Clausen RP, Bräuner-Osborne H, Greenwood JR, Hermit MB, Stensbøl TB, Nielsen B, Krogsgaard-Larsen P. Clausen RP, et al. J Med Chem. 2002 Sep 12;45(19):4240-5. doi: 10.1021/jm020122x. J Med Chem. 2002. PMID: 12213064

7

Activity of novel 4-PIOL analogues at human alpha 1 beta 2 gamma 2S GABA(A) receptors--correlation with hydrophobicity.

Mortensen M, Frølund B, Jørgensen AT, Liljefors T, Krogsgaard-Larsen P, Ebert B. Mortensen M, et al. Eur J Pharmacol. 2002 Sep 13;451(2):125-32. doi: 10.1016/s0014-2999(02)02271-9. Eur J Pharmacol. 2002. PMID: 12231381

8

Specific GABA(A) agonists and partial agonists.

Krogsgaard-Larsen P, Frølund B, Liljefors T. Krogsgaard-Larsen P, et al. Chem Rec. 2002;2(6):419-30. doi: 10.1002/tcr.10040. Chem Rec. 2002. PMID: 12469353 Review.

9

(S)-2-Amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic acid, a potent and selective agonist at the GluR5 subtype of ionotropic glutamate receptors. Synthesis, modeling, and molecular pharmacology.

Brehm L, Greenwood JR, Hansen KB, Nielsen B, Egebjerg J, Stensbøl TB, Bräuner-Osborne H, Sløk FA, Kronborg TT, Krogsgaard-Larsen P. Brehm L, et al. J Med Chem. 2003 Apr 10;46(8):1350-8. doi: 10.1021/jm0204441. J Med Chem. 2003. PMID: 12672235

10

Aza-THIP and related analogues of THIP as GABA C antagonists.

Krehan D, Frølund B, Ebert B, Nielsen B, Krogsgaard-Larsen P, Johnston GA, Chebib M. Krehan D, et al. Bioorg Med Chem. 2003 Nov 17;11(23):4891-6. doi: 10.1016/j.bmc.2003.09.016. Bioorg Med Chem. 2003. PMID: 14604650

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