Rothman RB - Search Results

1

Structure-activity relationship studies of highly selective inhibitors of the dopamine transporter: N-benzylpiperidine analogues of 1-[2-[bis(4-fluorophenyl)methoxy]ethyl]-4-(3-phenylpropyl)piperazine.

Greiner E, Prisinzano T, Johnson EM 2nd, Dersch CM, Marcus J, Partilla JS, Rothman RB, Jacobson AE, Rice KC. Greiner E, et al. Among authors: rothman rb. J Med Chem. 2003 Apr 10;46(8):1465-9. doi: 10.1021/jm020419v. J Med Chem. 2003. PMID: 12672246

2

Synthesis and biological activity of 8beta-substituted hydrocodone indole and hydromorphone indole derivatives.

Yu H, Prisinzano T, Dersch CM, Marcus J, Rothman RB, Jacobson AE, Rice KC. Yu H, et al. Among authors: rothman rb. Bioorg Med Chem Lett. 2002 Jan 21;12(2):165-8. doi: 10.1016/s0960-894x(01)00689-8. Bioorg Med Chem Lett. 2002. PMID: 11755345

3

Development of long-acting dopamine transporter ligands as potential cocaine-abuse therapeutic agents: chiral hydroxyl-containing derivatives of 1-[2-[bis(4-fluorophenyl)methoxy]ethyl]-4-(3-phenylpropyl)piperazine and 1-[2-(diphenylmethoxy)ethyl]-4-(3-phenylpropyl)piperazine.

Hsin LW, Dersch CM, Baumann MH, Stafford D, Glowa JR, Rothman RB, Jacobson AE, Rice KC. Hsin LW, et al. Among authors: rothman rb. J Med Chem. 2002 Mar 14;45(6):1321-9. doi: 10.1021/jm010430f. J Med Chem. 2002. PMID: 11882001

4

Identification of a novel partial inhibitor of dopamine transporter among 4-substituted 2-phenylquinazolines.

Ananthan S, Saini SK, Khare R, Clayton SD, Dersch CM, Rothman RB. Ananthan S, et al. Among authors: rothman rb. Bioorg Med Chem Lett. 2002 Aug 19;12(16):2225-8. doi: 10.1016/s0960-894x(02)00348-7. Bioorg Med Chem Lett. 2002. PMID: 12127543

5

Probes for narcotic receptor mediated phenomena. Part 28: new opioid antagonists from enantiomeric analogues of 5-(3-hydroxyphenyl)-N-phenylethylmorphan.

Hashimoto A, Jacobson AE, Rothman RB, Dersch CM, George C, Flippen-Anderson JL, Rice KC. Hashimoto A, et al. Among authors: rothman rb. Bioorg Med Chem. 2002 Oct;10(10):3319-29. doi: 10.1016/s0968-0896(02)00219-5. Bioorg Med Chem. 2002. PMID: 12150879

6

Piperidine analogues of 1-[2-[bis(4-fluorophenyl)methoxy]ethyl]-4-(3-phenylpropyl)piperazine (GBR 12909): high affinity ligands for the dopamine transporter.

Prisinzano T, Greiner E, Johnson EM 2nd, Dersch CM, Marcus J, Partilla JS, Rothman RB, Jacobson AE, Rice KC. Prisinzano T, et al. Among authors: rothman rb. J Med Chem. 2002 Sep 12;45(19):4371-4. doi: 10.1021/jm020264r. J Med Chem. 2002. PMID: 12213078

7

Synthesis and biological evaluation of 14-alkoxymorphinans. 17. Highly delta opioid receptor selective 14-alkoxy-substituted indolo- and benzofuromorphinans.

Schütz J, Dersch CM, Horel R, Spetea M, Koch M, Meditz R, Greiner E, Rothman RB, Schmidhammer H. Schütz J, et al. Among authors: rothman rb. J Med Chem. 2002 Nov 21;45(24):5378-83. doi: 10.1021/jm020940p. J Med Chem. 2002. PMID: 12431065

8

Synthesis and dopamine transporter affinity of chiral 1-[2-[bis(4-fluorophenyl)methoxy]ethyl]-4-(2-hydroxypropyl)piperazines as potential cocaine abuse therapeutic agents.

Hsin LW, Prisinzano T, Wilkerson CR, Dersch CM, Horel R, Jacobson AE, Rothman RB, Rice KC. Hsin LW, et al. Among authors: rothman rb. Bioorg Med Chem Lett. 2003 Feb 10;13(3):553-6. doi: 10.1016/s0960-894x(02)00940-x. Bioorg Med Chem Lett. 2003. PMID: 12565970

9

Further exploration of 1-[2-[Bis-(4-fluorophenyl)methoxy]ethyl]piperazine (GBR 12909): role of N-aromatic, N-heteroaromatic, and 3-oxygenated N-phenylpropyl substituents on affinity for the dopamine and serotonin transporter.

Lewis D, Zhang Y, Prisinzano T, Dersch CM, Rothman RB, Jacobson AE, Rice KC. Lewis D, et al. Among authors: rothman rb. Bioorg Med Chem Lett. 2003 Apr 7;13(7):1385-9. doi: 10.1016/s0960-894x(03)00108-2. Bioorg Med Chem Lett. 2003. PMID: 12657288

10

Diaryldimethylpiperazine ligands with mu- and delta-opioid receptor affinity: Synthesis of (+)-4-[(alphaR)-alpha-(4-allyl-(2S,5S)-dimethylpiperazin-1-yl)-(3-hydroxyphenyl)methyl]-N-ethyl-N-phenylbenzamide and (-)-4-[(alphaR)-alpha-(2S,5S)-dimethylpiperazin-1-yl)-(3-hydroxyphenyl)methyl]-N-ethyl-N-phenylbenzamide.

Kim IJ, Ullrich T, Janetka JW, Furness MS, Jacobson AE, Rothman RB, Dersch CM, Flippen-Anderson JL, George C, Rice KC. Kim IJ, et al. Among authors: rothman rb. Bioorg Med Chem. 2003 Nov 3;11(22):4761-8. doi: 10.1016/s0968-0896(03)00496-6. Bioorg Med Chem. 2003. PMID: 14556791

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