Cheung AW - Search Results

1

Structure-activity relationship of cyclic peptide penta-c[Asp-His(6)-DPhe(7)-Arg(8)-Trp(9)-Lys]-NH(2) at the human melanocortin-1 and -4 receptors: His(6) substitution.

Cheung AW, Danho W, Swistok J, Qi L, Kurylko G, Rowan K, Yeon M, Franco L, Chu XJ, Chen L, Yagaloff K. Cheung AW, et al. Bioorg Med Chem Lett. 2003 Apr 7;13(7):1307-11. doi: 10.1016/s0960-894x(03)00114-8. Bioorg Med Chem Lett. 2003. PMID: 12657270

2

A predictive pharmacophore model of human melanocortin-4 receptor as derived from the solution structures of cyclic peptides.

Sun H, Greeley DN, Chu XJ, Cheung A, Danho W, Swistok J, Wang Y, Zhao C, Chen L, Fry DC. Sun H, et al. Bioorg Med Chem. 2004 May 15;12(10):2671-7. doi: 10.1016/j.bmc.2004.03.017. Bioorg Med Chem. 2004. PMID: 15110848

3

Structure-activity relationship of linear peptide Bu-His-DPhe-Arg-Trp-Gly-NH(2) at the human melanocortin-1 and -4 receptors: arginine substitution.

Cheung AW, Danho W, Swistok J, Qi L, Kurylko G, Franco L, Yagaloff K, Chen L. Cheung AW, et al. Bioorg Med Chem Lett. 2002 Sep 2;12(17):2407-10. doi: 10.1016/s0960-894x(02)00459-6. Bioorg Med Chem Lett. 2002. PMID: 12161144

4

Structure-activity relationship of linear peptide Bu-His-DPhe-Arg-Trp-Gly-NH(2) at the human melanocortin-1 and -4 receptors: histidine substitution.

Cheung AW, Danho W, Swistok J, Qi L, Kurylko G, Rowan K, Yeon M, Franco L, Chu XJ, Chen L, Yagaloff K. Cheung AW, et al. Bioorg Med Chem Lett. 2003 Jan 6;13(1):133-7. doi: 10.1016/s0960-894x(02)00830-2. Bioorg Med Chem Lett. 2003. PMID: 12467633

5

Structure-activity relationship of linear peptide Bu-His6-DPhe7-Arg8-Trp9-Gly10-NH2 at the human melanocortin-1 and -4 receptors: DPhe7 and Trp9 substitution.

Danho W, Swistok J, Cheung AW, Kurylko G, Franco L, Chu XJ, Chen L, Yagaloff K. Danho W, et al. Among authors: cheung aw. Bioorg Med Chem Lett. 2003 Feb 24;13(4):649-52. doi: 10.1016/s0960-894x(02)01052-1. Bioorg Med Chem Lett. 2003. PMID: 12639550

6

Discovery of 1-amino-4-phenylcyclohexane-1-carboxylic acid and its influence on agonist selectivity between human melanocortin-4 and -1 receptors in linear pentapeptides.

Chu XJ, Bartkovitz D, Danho W, Swistok J, Cheung AW, Kurylko G, Rowan K, Yeon M, Franco L, Qi L, Chen L, Yagaloff K. Chu XJ, et al. Among authors: cheung aw. Bioorg Med Chem Lett. 2005 Nov 15;15(22):4910-4. doi: 10.1016/j.bmcl.2005.08.012. Bioorg Med Chem Lett. 2005. PMID: 16169218

7

Preparation of human Melanocortin-4 receptor agonist libraries: linear peptides X-Y-DPhe7-Arg8-Trp(or 2-Nal)9-Z-NH2.

Cheung AW, Qi L, Gore V, Chu XJ, Bartkovitz D, Kurylko G, Swistok J, Danho W, Chen L, Yagaloff K. Cheung AW, et al. Bioorg Med Chem Lett. 2005 Dec 15;15(24):5504-8. doi: 10.1016/j.bmcl.2005.08.083. Epub 2005 Oct 3. Bioorg Med Chem Lett. 2005. PMID: 16203134

8

Opportunities and challenges of developing peptide drugs in the pharmaceutical industry.

Danho W, Swistok J, Khan W, Chu XJ, Cheung A, Fry D, Sun H, Kurylko G, Rumennik L, Cefalu J, Cefalu G, Nunn P. Danho W, et al. Adv Exp Med Biol. 2009;611:467-9. doi: 10.1007/978-0-387-73657-0_201. Adv Exp Med Biol. 2009. PMID: 19400268 No abstract available.

9

4-Substituted-7-N-alkyl-N-acetyl 2-aminobenzothiazole amides: drug-like and non-xanthine based A2B adenosine receptor antagonists.

Cheung AW, Brinkman J, Firooznia F, Flohr A, Grimsby J, Gubler ML, Guertin K, Hamid R, Marcopulos N, Norcross RD, Qi L, Ramsey G, Tan J, Wen Y, Sarabu R. Cheung AW, et al. Bioorg Med Chem Lett. 2010 Jul 15;20(14):4140-6. doi: 10.1016/j.bmcl.2010.05.056. Epub 2010 May 20. Bioorg Med Chem Lett. 2010. PMID: 20541935

10

Discovery of benzothiazole-based adenosine A2B receptor antagonists with improved A2A selectivity.

Firooznia F, Cheung AW, Brinkman J, Grimsby J, Gubler ML, Hamid R, Marcopulos N, Ramsey G, Tan J, Wen Y, Sarabu R. Firooznia F, et al. Among authors: cheung aw. Bioorg Med Chem Lett. 2011 Apr 1;21(7):1933-6. doi: 10.1016/j.bmcl.2011.02.053. Epub 2011 Feb 17. Bioorg Med Chem Lett. 2011. PMID: 21388809

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

142 results

Search Page

Filters