Kohn H - Search Results

1

Quantitative structure-activity relationship analysis of functionalized amino acid anticonvulsant agents using k nearest neighbor and simulated annealing PLS methods.

Shen M, LeTiran A, Xiao Y, Golbraikh A, Kohn H, Tropsha A. Shen M, et al. Among authors: kohn h. J Med Chem. 2002 Jun 20;45(13):2811-23. doi: 10.1021/jm010488u. J Med Chem. 2002. PMID: 12061883

2

Design and evaluation of affinity labels of functionalized amino acid anticonvulsants.

LeTiran A, Stables JP, Kohn H. LeTiran A, et al. Among authors: kohn h. J Med Chem. 2002 Oct 10;45(21):4762-73. doi: 10.1021/jm020225f. J Med Chem. 2002. PMID: 12361404

3

Application of predictive QSAR models to database mining: identification and experimental validation of novel anticonvulsant compounds.

Shen M, Béguin C, Golbraikh A, Stables JP, Kohn H, Tropsha A. Shen M, et al. Among authors: kohn h. J Med Chem. 2004 Apr 22;47(9):2356-64. doi: 10.1021/jm030584q. J Med Chem. 2004. PMID: 15084134

4

N-Substituted amino acid N'-benzylamides: synthesis, anticonvulsant, and metabolic activities.

Béguin C, LeTiran A, Stables JP, Voyksner RD, Kohn H. Béguin C, et al. Among authors: kohn h. Bioorg Med Chem. 2004 Jun 1;12(11):3079-96. doi: 10.1016/j.bmc.2004.02.043. Bioorg Med Chem. 2004. PMID: 15142567

5

A novel automated lazy learning QSAR (ALL-QSAR) approach: method development, applications, and virtual screening of chemical databases using validated ALL-QSAR models.

Zhang S, Golbraikh A, Oloff S, Kohn H, Tropsha A. Zhang S, et al. Among authors: kohn h. J Chem Inf Model. 2006 Sep-Oct;46(5):1984-95. doi: 10.1021/ci060132x. J Chem Inf Model. 2006. PMID: 16995729 Free PMC article.

6

Functionalized amino acid anticonvulsants: synthesis and pharmacological evaluation of conformationally restricted analogues.

LeTiran A, Stables JP, Kohn H. LeTiran A, et al. Among authors: kohn h. Bioorg Med Chem. 2001 Oct;9(10):2693-708. doi: 10.1016/s0968-0896(01)00204-8. Bioorg Med Chem. 2001. PMID: 11557357

7

Primary amino acid derivatives: compounds with anticonvulsant and neuropathic pain protection activities.

King AM, Salomé C, Dinsmore J, Salomé-Grosjean E, De Ryck M, Kaminski R, Valade A, Kohn H. King AM, et al. Among authors: kohn h. J Med Chem. 2011 Jul 14;54(13):4815-30. doi: 10.1021/jm2004305. Epub 2011 Jun 15. J Med Chem. 2011. PMID: 21639114

8

Defining the structural parameters that confer anticonvulsant activity by the site-by-site modification of (R)-N'-benzyl 2-amino-3-methylbutanamide.

King AM, De Ryck M, Kaminski R, Valade A, Stables JP, Kohn H. King AM, et al. Among authors: kohn h. J Med Chem. 2011 Oct 13;54(19):6432-42. doi: 10.1021/jm200760a. Epub 2011 Sep 13. J Med Chem. 2011. PMID: 21861466 Free PMC article.

9

Merging the structural motifs of functionalized amino acids and alpha-aminoamides: compounds with significant anticonvulsant activities.

Salomé C, Salomé-Grosjean E, Stables JP, Kohn H. Salomé C, et al. Among authors: kohn h. J Med Chem. 2010 May 13;53(9):3756-71. doi: 10.1021/jm100185c. J Med Chem. 2010. PMID: 20394379 Free PMC article.

10

The structure-activity relationship of the 3-oxy site in the anticonvulsant (R)-N-benzyl 2-acetamido-3-methoxypropionamide.

Morieux P, Salomé C, Park KD, Stables JP, Kohn H. Morieux P, et al. Among authors: kohn h. J Med Chem. 2010 Aug 12;53(15):5716-26. doi: 10.1021/jm100508m. J Med Chem. 2010. PMID: 20614888 Free PMC article.

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