Kauss V - Search Results

1

Amino-alkyl-cyclohexanes as a novel class of uncompetitive NMDA receptor antagonists.

Danysz W, Parsons CG, Jirgensons A, Kauss V, Tillner J. Danysz W, et al. Among authors: kauss v. Curr Pharm Des. 2002;8(10):835-43. doi: 10.2174/1381612024607117. Curr Pharm Des. 2002. PMID: 11945134 Review.

2

A novel class of amino-alkylcyclohexanes as uncompetitive, fast, voltage-dependent, N-methyl-D-aspartate (NMDA) receptor antagonists--in vitro characterization.

Gilling K, Jatzke C, Wollenburg C, Vanejevs M, Kauss V, Jirgensons A, Parsons CG. Gilling K, et al. Among authors: kauss v. J Neural Transm (Vienna). 2007;114(12):1529-37. doi: 10.1007/s00702-007-0792-7. Epub 2007 Aug 31. J Neural Transm (Vienna). 2007. PMID: 17728997

3

Virtual screening for selective allosteric mGluR1 antagonists and structure-activity relationship investigations for coumarine derivatives.

Noeske T, Jirgensons A, Starchenkovs I, Renner S, Jaunzeme I, Trifanova D, Hechenberger M, Bauer T, Kauss V, Parsons CG, Schneider G, Weil T. Noeske T, et al. Among authors: kauss v. ChemMedChem. 2007 Dec;2(12):1763-73. doi: 10.1002/cmdc.200700151. ChemMedChem. 2007. PMID: 17868161

4

Synergism of virtual screening and medicinal chemistry: identification and optimization of allosteric antagonists of metabotropic glutamate receptor 1.

Noeske T, Trifanova D, Kauss V, Renner S, Parsons CG, Schneider G, Weil T. Noeske T, et al. Among authors: kauss v. Bioorg Med Chem. 2009 Aug 1;17(15):5708-15. doi: 10.1016/j.bmc.2009.05.072. Epub 2009 Jun 23. Bioorg Med Chem. 2009. PMID: 19574055

5

Synthesis and structure-affinity relationships of 1,3, 5-alkylsubstituted cyclohexylamines binding at NMDA receptor PCP site.

Jirgensons A, Kauss V, Kalvinsh I, Gold MR, Danysz W, Parsons CG, Quack G. Jirgensons A, et al. Among authors: kauss v. Eur J Med Chem. 2000 Jun;35(6):555-65. doi: 10.1016/s0223-5234(00)00153-7. Eur J Med Chem. 2000. PMID: 10906408

6

Positive and negative modulation of group I metabotropic glutamate receptors.

Vanejevs M, Jatzke C, Renner S, Müller S, Hechenberger M, Bauer T, Klochkova A, Pyatkin I, Kazyulkin D, Aksenova E, Shulepin S, Timonina O, Haasis A, Gutcaits A, Parsons CG, Kauss V, Weil T. Vanejevs M, et al. Among authors: kauss v. J Med Chem. 2008 Feb 14;51(3):634-47. doi: 10.1021/jm0611298. Epub 2008 Jan 4. J Med Chem. 2008. PMID: 18173231

7

Discovery, synthesis, and structure-activity relationships of 2-aminoquinazoline derivatives as a novel class of metabotropic glutamate receptor 5 negative allosteric modulators.

Kubas H, Meyer U, Krueger B, Hechenberger M, Vanejevs M, Zemribo R, Kauss V, Ambartsumova R, Pyatkin I, Polosukhin AI, Abel U. Kubas H, et al. Among authors: kauss v. Bioorg Med Chem Lett. 2013 Aug 15;23(16):4493-500. doi: 10.1016/j.bmcl.2013.06.049. Epub 2013 Jun 25. Bioorg Med Chem Lett. 2013. PMID: 23856046

8

Synthesis of 3,4-dihydro-2H-1,2-benzothiazine-3-carboxylic acid 1,1-dioxides and their evaluation as ligands for NMDA receptor glycine binding site.

Bluke Z, Paass E, Sladek M, Abel U, Kauss V. Bluke Z, et al. Among authors: kauss v. J Enzyme Inhib Med Chem. 2016 Aug;31(4):664-73. doi: 10.3109/14756366.2015.1057722. Epub 2015 Jun 26. J Enzyme Inhib Med Chem. 2016. PMID: 26114309 Free article.

9

A convenient synthesis of 5beta-cholestan-26-oic and 5beta-cholestan-26,27-dioic acids.

Starchenkov I, Trapencieris P, Kauss V, Jas G, Kalvinsh I. Starchenkov I, et al. Among authors: kauss v. Steroids. 2000 Mar;65(3):143-7. doi: 10.1016/s0039-128x(99)00099-9. Steroids. 2000. PMID: 10699593

10

Pharmacological approaches to tackle NCLs.

Kauss V, Dambrova M, Medina DL. Kauss V, et al. Biochim Biophys Acta Mol Basis Dis. 2020 Sep 1;1866(9):165553. doi: 10.1016/j.bbadis.2019.165553. Epub 2019 Sep 12. Biochim Biophys Acta Mol Basis Dis. 2020. PMID: 31521819 Free article. Review.

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