Gerrard JA - Search Results

1

Kinetic characterisation of ene-diol-based inhibitors of alpha-amylase.

Gerrard JA, Prince MJ, Abell AD. Gerrard JA, et al. Bioorg Med Chem Lett. 2000 Jul 17;10(14):1575-6. doi: 10.1016/s0960-894x(00)00288-2. Bioorg Med Chem Lett. 2000. PMID: 10915054

2

Ascorbic acid-based inhibitors of alpha-amylases.

Abell AD, Ratcliffe MJ, Gerrard J. Abell AD, et al. Bioorg Med Chem Lett. 1998 Jul 7;8(13):1703-6. doi: 10.1016/s0960-894x(98)00298-4. Bioorg Med Chem Lett. 1998. PMID: 9873419

3

The preparation of (S)-aspartate semi-aldehyde appropriate for use in biochemical studies.

Roberts SJ, Morris JC, Dobson RC, Gerrard JA. Roberts SJ, et al. Among authors: gerrard ja. Bioorg Med Chem Lett. 2003 Jan 20;13(2):265-7. doi: 10.1016/s0960-894x(02)00923-x. Bioorg Med Chem Lett. 2003. PMID: 12482436

4

New insights into protein crosslinking via the Maillard reaction: structural requirements, the effect on enzyme function, and predicted efficacy of crosslinking inhibitors as anti-ageing therapeutics.

Miller AG, Meade SJ, Gerrard JA. Miller AG, et al. Among authors: gerrard ja. Bioorg Med Chem. 2003 Mar 20;11(6):843-52. doi: 10.1016/s0968-0896(02)00565-5. Bioorg Med Chem. 2003. PMID: 12614869

5

The role of dicarbonyl compounds in non-enzymatic crosslinking: a structure-activity study.

Meade SJ, Miller AG, Gerrard JA. Meade SJ, et al. Among authors: gerrard ja. Bioorg Med Chem. 2003 Mar 20;11(6):853-62. doi: 10.1016/s0968-0896(02)00564-3. Bioorg Med Chem. 2003. PMID: 12614870

6

Heterocyclic inhibitors of dihydrodipicolinate synthase are not competitive.

Turner JJ, Gerrard JA, Hutton CA. Turner JJ, et al. Among authors: gerrard ja. Bioorg Med Chem. 2005 Mar 15;13(6):2133-40. doi: 10.1016/j.bmc.2005.01.001. Bioorg Med Chem. 2005. PMID: 15727866

7

Dihydrodipicolinate synthase is not inhibited by its substrate, (S)-aspartate beta-semialdehyde.

Dobson RC, Gerrard JA, Pearce FG. Dobson RC, et al. Among authors: gerrard ja. Biochem J. 2004 Feb 1;377(Pt 3):757-62. doi: 10.1042/BJ20031389. Biochem J. 2004. PMID: 14580236 Free PMC article.

8

Two new irreversible inhibitors of dihydrodipicolinate synthase: diethyl (E,E)-4-oxo-2,5-heptadienedioate and diethyl (E)-4-oxo-2-heptenedioate.

Turner JJ, Healy JP, Dobson RC, Gerrard JA, Hutton CA. Turner JJ, et al. Among authors: gerrard ja. Bioorg Med Chem Lett. 2005 Feb 15;15(4):995-8. doi: 10.1016/j.bmcl.2004.12.043. Bioorg Med Chem Lett. 2005. PMID: 15686899

9

Conformationally constrained diketopimelic acid analogues as inhibitors of dihydrodipicolinate synthase.

Boughton BA, Dobson RC, Gerrard JA, Hutton CA. Boughton BA, et al. Among authors: gerrard ja. Bioorg Med Chem Lett. 2008 Jan 15;18(2):460-3. doi: 10.1016/j.bmcl.2007.11.108. Epub 2007 Dec 3. Bioorg Med Chem Lett. 2008. PMID: 18077163

10

Irreversible inhibition of dihydrodipicolinate synthase by 4-oxo-heptenedioic acid analogues.

Boughton BA, Griffin MD, O'Donnell PA, Dobson RC, Perugini MA, Gerrard JA, Hutton CA. Boughton BA, et al. Among authors: gerrard ja. Bioorg Med Chem. 2008 Dec 1;16(23):9975-83. doi: 10.1016/j.bmc.2008.10.026. Epub 2008 Oct 17. Bioorg Med Chem. 2008. PMID: 18977662

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