Domínguez C - Search Results

1

4-Alkyl- and 4-cinnamylglutamic acid analogues are potent GluR5 kainate receptor agonists.

Pedregal C, Collado I, Escribano A, Ezquerra J, Domínguez C, Mateo AI, Rubio A, Baker SR, Goldsworthy J, Kamboj RK, Ballyk BA, Hoo K, Bleakman D. Pedregal C, et al. Among authors: dominguez c. J Med Chem. 2000 May 18;43(10):1958-68. doi: 10.1021/jm9911682. J Med Chem. 2000. PMID: 10821708

2

4-Alkylidenyl glutamic acids, potent and selective GluR5 agonists.

Baker SR, Bleakman D, Ezquerra J, Ballyk BA, Deverill M, Ho K, Kamboj RK, Collado I, Domínguez C, Escribano A, Mateo AI, Pedregal C, Rubio A. Baker SR, et al. Among authors: dominguez c. Bioorg Med Chem Lett. 2000 Aug 21;10(16):1807-10. doi: 10.1016/s0960-894x(00)00346-2. Bioorg Med Chem Lett. 2000. PMID: 10969973

3

Dipeptides as effective prodrugs of the unnatural amino acid (+)-2-aminobicyclo[3.1.0]hexane-2,6-dicarboxylic acid (LY354740), a selective group II metabotropic glutamate receptor agonist.

Bueno AB, Collado I, de Dios A, Domínguez C, Martín JA, Martín LM, Martínez-Grau MA, Montero C, Pedregal C, Catlow J, Coffey DS, Clay MP, Dantzig AH, Lindstrom T, Monn JA, Jiang H, Schoepp DD, Stratford RE, Tabas LB, Tizzano JP, Wright RA, Herin MF. Bueno AB, et al. Among authors: dominguez c. J Med Chem. 2005 Aug 11;48(16):5305-20. doi: 10.1021/jm050235r. J Med Chem. 2005. PMID: 16078848

4

Methyl substitution of 2-aminobicyclo[3.1.0]hexane 2,6-dicarboxylate (LY354740) determines functional activity at metabotropic glutamate receptors: identification of a subtype selective mGlu2 receptor agonist.

Dominguez C, Prieto L, Valli MJ, Massey SM, Bures M, Wright RA, Johnson BG, Andis SL, Kingston A, Schoepp DD, Monn JA. Dominguez C, et al. J Med Chem. 2005 May 19;48(10):3605-12. doi: 10.1021/jm040222y. J Med Chem. 2005. PMID: 15887967

5

Synthesis and evaluation of conformationally restricted N-[2-(3,4-dichlorophenyl)ethyl]-N-methyl-2-(1-pyrrolidinyl)ethylamines at sigma receptors. 2. Piperazines, bicyclic amines, bridged bicyclic amines, and miscellaneous compounds.

de Costa BR, He XS, Linders JT, Dominguez C, Gu ZQ, Williams W, Bowen WD. de Costa BR, et al. Among authors: dominguez c. J Med Chem. 1993 Aug 6;36(16):2311-20. doi: 10.1021/jm00068a007. J Med Chem. 1993. PMID: 8360875

6

A new approach to the design of sigma-2-selective ligands: synthesis and evaluation of N-[2-(3,4-dichlorophenyl)ethyl]-N-methyl-2-(1- pyrrolidinyl)ethylamine-related polyamines at sigma-1 and sigma-2 receptor subtypes.

de Costa BR, He XS, Dominguez C, Cutts J, Williams W, Bowen WD. de Costa BR, et al. Among authors: dominguez c. J Med Chem. 1994 Jan 21;37(2):314-21. doi: 10.1021/jm00028a016. J Med Chem. 1994. PMID: 8295220

7

Imidazolyl benzimidazoles and imidazo[4,5-b]pyridines as potent p38alpha MAP kinase inhibitors with excellent in vivo antiinflammatory properties.

Mader M, de Dios A, Shih C, Bonjouklian R, Li T, White W, López de Uralde B, Sánchez-Martinez C, del Prado M, Jaramillo C, de Diego E, Martín Cabrejas LM, Dominguez C, Montero C, Shepherd T, Dally R, Toth JE, Chatterjee A, Pleite S, Blanco-Urgoiti J, Perez L, Barberis M, Lorite MJ, Jambrina E, Nevill CR Jr, Lee PA, Schultz RC, Wolos JA, Li LC, Campbell RM, Anderson BD. Mader M, et al. Among authors: dominguez c. Bioorg Med Chem Lett. 2008 Jan 1;18(1):179-83. doi: 10.1016/j.bmcl.2007.10.106. Epub 2007 Nov 1. Bioorg Med Chem Lett. 2008. PMID: 18039577

8

Design, synthesis, and biological evaluation of potent and selective amidino bicyclic factor Xa inhibitors.

Han Q, Dominguez C, Stouten PF, Park JM, Duffy DE, Galemmo RA Jr, Rossi KA, Alexander RS, Smallwood AM, Wong PC, Wright MM, Luettgen JM, Knabb RM, Wexler RR. Han Q, et al. Among authors: dominguez c. J Med Chem. 2000 Nov 16;43(23):4398-415. doi: 10.1021/jm000113t. J Med Chem. 2000. PMID: 11087565

9

Synthesis and biological evaluation of conformationally restricted 2-(1-pyrrolidinyl)-N-[2-(3,4-dichlorophenyl)ethyl]-N-methylethylenediam ines as sigma receptor ligands. 1. Pyrrolidine, piperidine, homopiperidine, and tetrahydroisoquinoline classes.

de Costa BR, Dominguez C, He XS, Williams W, Radesca L, Bowen W. de Costa BR, et al. Among authors: dominguez c. J Med Chem. 1992 Nov 13;35(23):4334-43. doi: 10.1021/jm00101a011. J Med Chem. 1992. PMID: 1447735

10

Synthesis and evaluation of imidazo[1,5-a][1,4]benzodiazepine esters with high affinities and selectivities at "diazepam-insensitive" benzodiazepine receptors.

Gu ZQ, Wong G, Dominguez C, de Costa BR, Rice KC, Skolnick P. Gu ZQ, et al. Among authors: dominguez c. J Med Chem. 1993 Apr 16;36(8):1001-6. doi: 10.1021/jm00060a007. J Med Chem. 1993. PMID: 8386769

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

877 results

Search Page

Filters