Timmerman H - Search Results

1

Characterization of the binding site of the histamine H(3) receptor. 2. Synthesis, in vitro pharmacology, and QSAR of a series of monosubstituted benzyl analogues of thioperamide.

Windhorst AD, Timmerman H, Worthington EA, Bijloo GJ, Nederkoorn PH, Menge WM, Leurs R, Herscheid JD. Windhorst AD, et al. Among authors: timmerman h. J Med Chem. 2000 May 4;43(9):1754-61. doi: 10.1021/jm981106w. J Med Chem. 2000. PMID: 10794692

2

A new potent and selective histamine H3 receptor agonist, 4-(1H-imidazol-4-ylmethyl)piperidine.

Vollinga RC, de Koning JP, Jansen FP, Leurs R, Menge WM, Timmerman H. Vollinga RC, et al. Among authors: timmerman h. J Med Chem. 1994 Feb 4;37(3):332-3. doi: 10.1021/jm00029a002. J Med Chem. 1994. PMID: 8308858 No abstract available.

3

Evaluation of the receptor selectivity of the H3 receptor antagonists, iodophenpropit and thioperamide: an interaction with the 5-HT3 receptor revealed.

Leurs R, Tulp MT, Menge WM, Adolfs MJ, Zuiderveld OP, Timmerman H. Leurs R, et al. Among authors: timmerman h. Br J Pharmacol. 1995 Oct;116(4):2315-21. doi: 10.1111/j.1476-5381.1995.tb15071.x. Br J Pharmacol. 1995. PMID: 8564266 Free PMC article.

4

Characterization of the binding site of the histamine H3 receptor. 1. Various approaches to the synthesis of 2-(1H-imidazol-4-yl)cyclopropylamine and histaminergic activity of (1R,2R)- and (1S,2S)-2-(1H-imidazol-4-yl)-cyclopropylamine.

De Esch IJ, Vollinga RC, Goubitz K, Schenk H, Appelberg U, Hacksell U, Lemstra S, Zuiderveld OP, Hoffmann M, Leurs R, Menge WM, Timmerman H. De Esch IJ, et al. Among authors: timmerman h. J Med Chem. 1999 Apr 8;42(7):1115-22. doi: 10.1021/jm9810912. J Med Chem. 1999. PMID: 10197956 Free article.

5

Evaluation of [18F]VUF 5000 as a potential PET ligand for brain imaging of the histamine H3 receptor.

Windhorst AD, Timmerman H, Klok RP, Menge WM, Leurs R, Herscheid JD. Windhorst AD, et al. Among authors: timmerman h. Bioorg Med Chem. 1999 Sep;7(9):1761-7. doi: 10.1016/s0968-0896(99)00108-x. Bioorg Med Chem. 1999. PMID: 10530922

6

Synthesis and histamine H3 receptor activity of 4-(n-alkyl)-1H-imidazoles and 4-(omega-phenylalkyl)-1H-imidazoles.

De Esch IJ, Gaffar A, Menge WM, Timmerman H. De Esch IJ, et al. Among authors: timmerman h. Bioorg Med Chem. 1999 Dec;7(12):3003-9. doi: 10.1016/s0968-0896(99)00253-9. Bioorg Med Chem. 1999. PMID: 10658607

7

Isoquinoline and quinazoline urea analogues as antagonists for the human adenosine A(3) receptor.

van Muijlwijk-Koezen JE, Timmerman H, van der Goot H, Menge WM, Frijtag Von Drabbe Künzel J, de Groote M, IJzerman AP. van Muijlwijk-Koezen JE, et al. Among authors: timmerman h. J Med Chem. 2000 Jun 1;43(11):2227-38. doi: 10.1021/jm000002u. J Med Chem. 2000. PMID: 10841801 Free article.

8

Solid-phase synthesis of 4-substituted imidazoles using a scaffold approach.

Gelens E, Koot WJ, Menge WM, Ottenheijm HC, Timmerman H. Gelens E, et al. Among authors: timmerman h. Bioorg Med Chem Lett. 2000 Sep 4;10(17):1935-8. doi: 10.1016/s0960-894x(00)00363-2. Bioorg Med Chem Lett. 2000. PMID: 10987421

9

Development of a pharmacophore model for histamine H3 receptor antagonists, using the newly developed molecular modeling program SLATE.

De Esch IJ, Mills JE, Perkins TD, Romeo G, Hoffmann M, Wieland K, Leurs R, Menge WM, Nederkoorn PH, Dean PM, Timmerman H. De Esch IJ, et al. Among authors: timmerman h. J Med Chem. 2001 May 24;44(11):1666-74. doi: 10.1021/jm001109k. J Med Chem. 2001. PMID: 11356102

10

Pharmacological analysis of immepip and imetit homologues. Further evidence for histamine H(3) receptor heterogeneity?

Alves-Rodrigues A, Lemstra S, Vollinga RC, Menge WM, Timmerman H, Leurs R. Alves-Rodrigues A, et al. Among authors: timmerman h. Behav Brain Res. 2001 Oct 15;124(2):121-7. doi: 10.1016/s0166-4328(01)00224-8. Behav Brain Res. 2001. PMID: 11640964

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