Synthesis and biological evaluation of 1,2-disubstituted carbonucleosides of 2-amino-6-substituted purine and 8-azapurine

Bioorg Med Chem Lett. 1998 Jun 2;8(11):1349-52. doi: 10.1016/s0960-894x(98)00216-9.

Abstract

One, two-disubstituted carbocyclic nucleoside analogues bearing a 2-amino-6-substituted (chloro, hydroxy or amino) purine or 8-azapurine base were prepared by constructing the base about (+/-)-2-aminocyclopentane methanol, and their activities against a selection of viruses and tumor cells were determined in vitro.

MeSH terms

  • Animals
  • Antineoplastic Agents / chemical synthesis*
  • Antineoplastic Agents / pharmacology
  • Antiviral Agents / chemical synthesis*
  • Antiviral Agents / pharmacology
  • Drug Screening Assays, Antitumor
  • Humans
  • Inhibitory Concentration 50
  • Microbial Sensitivity Tests
  • Purine Nucleosides / chemical synthesis*
  • Purine Nucleosides / pharmacology
  • Tumor Cells, Cultured
  • Viruses / drug effects

Substances

  • Antineoplastic Agents
  • Antiviral Agents
  • Purine Nucleosides