Orbital fibroblast chemokine modulation: effects of dexamethasone and cyclosporin A

Br J Ophthalmol. 1998 Mar;82(3):318-22. doi: 10.1136/bjo.82.3.318.

Abstract

Aim: Orbital inflammation is common, but the mechanisms underlying leucocytic infiltration of orbital tissue are poorly understood. Human orbital fibroblasts (OF) express chemokines, interleukin 8 (IL-8) and monocyte chemotactic protein 1 (MCP-1), when exposed to proinflammatory cytokines. The effect of dexamethasone (DEX) and cyclosporin A (CSA) on OF IL-8 and MCP-1 were examined.

Methods: Cultured human OF were incubated with recombinant interleukin 1 beta (rIL-1 beta; 0.2, 2.0, 20 ng/ml) alone or incubated with rIL-1 beta and DEX (10(-8), 10(-7), 10(-6) M) or CSA (3, 30, 300 ng/ml) for 24 hours. ELISA and northern blot analyses were performed to determine OF IL-8 and MCP-1 protein secretion and mRNA expression, respectively.

Results: OF lacked constitutive IL-8 or MCP-1 expression, but secreted significant amounts of these chemokines and expressed substantial steady state mRNA for both chemokines upon rIL-1 beta stimulation. DEX caused dose dependent inhibition of IL-1 induced IL-8 (p < 0.001) and MCP-1 (p < 0.05) secretion and mRNA expression at all concentrations of rIL-1 beta. CSA enhanced IL-1 induced OF IL-8 (p < 0.001) and suppressed rIL-1 beta induced OF MCP-1 (p < 0.05) secretion when lower doses of rIL-1 beta were used. These effects on secreted chemokines at different concentrations of rIL-1 beta and immunomodulating agents were corroborated by steady state OF IL-8 and MCP-1 mRNA expression.

Conclusions: DEX is a potent inhibitor of OF IL-8 and MCP-1. In contrast, CSA enhances IL-1 induced OF IL-8 and suppresses OF MCP-1. These observations may explain the relative lack of CSA effectiveness in human orbital diseases that respond to corticosteroids.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Anti-Inflammatory Agents / pharmacology*
  • Blotting, Northern
  • Cells, Cultured
  • Chemokine CCL2 / analysis
  • Chemokine CCL2 / antagonists & inhibitors
  • Chemokines / metabolism*
  • Cyclosporine / pharmacology*
  • Dexamethasone / pharmacology*
  • Enzyme-Linked Immunosorbent Assay
  • Eye Diseases / genetics
  • Eye Diseases / metabolism*
  • Fibroblasts / drug effects
  • Fibroblasts / metabolism
  • Humans
  • Immunosuppressive Agents / pharmacology*
  • Interleukin-8 / analysis
  • Interleukin-8 / antagonists & inhibitors
  • RNA, Messenger / analysis

Substances

  • Anti-Inflammatory Agents
  • Chemokine CCL2
  • Chemokines
  • Immunosuppressive Agents
  • Interleukin-8
  • RNA, Messenger
  • Dexamethasone
  • Cyclosporine