Myc is essential for transformation by TEL/platelet-derived growth factor receptor beta (PDGFRbeta)

Blood. 1998 May 1;91(9):3333-9.

Abstract

The t(5;12) translocation identified in patients with chronic myelomonocytic leukemia (CMML) encodes a TEL/platelet-derived growth factor receptor beta (PDGFRbeta) fusion protein. A key hypothesis for how the TEL/PDGFRbeta fusion protein would function as an oncogene is that it represents a constitutively active version of the normal PDGFRbeta. A link between the function of the t(5;12)-encoded TEL/PDGFRbeta fusion protein and Myc expression is suggested by the fact that Myc is induced by PDGF and is essential for entry of cells into the S phase of the cell cycle. We here show that the kinase activity of TEL/PDGFRbeta is necessary for Ba/F3 cells to acquire interleukin-3 (IL-3) independence and that, in contrast to their untransfected counterpart, Ba/F3 cells stably transfected with TEL/PDGFRbeta maintain a high level of Myc expression after removal of IL-3. Using dominant negative mutants of Myc, we show that a threshold of active Myc is essential for TEL/PDGFRbeta to transform Ba/F3 and Rat-1 cells. The findings that the kinase activity of TEL/PDGFRbeta and a threshold of active Myc are involved in TEL/PDGFRbeta transformation may allow for the development of therapeutic strategies in patients with t(5;12)+ CMML using specific inhibitors of the PDGFRbeta kinase as well as compounds designed to interfere specifically with Myc.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Cell Division
  • Cell Transformation, Neoplastic*
  • Enzyme Inhibitors / pharmacology
  • Gene Expression Regulation, Neoplastic
  • Genes, Dominant
  • Genes, myc
  • Interleukin-3 / physiology
  • Proto-Oncogene Proteins c-myc / physiology*
  • Pyridines / pharmacology
  • Pyrimidines / pharmacology
  • Rats
  • Receptor Protein-Tyrosine Kinases / antagonists & inhibitors
  • Receptor Protein-Tyrosine Kinases / physiology
  • Receptors, Platelet-Derived Growth Factor / physiology*
  • Signal Transduction

Substances

  • CGP 53716
  • Enzyme Inhibitors
  • Interleukin-3
  • Proto-Oncogene Proteins c-myc
  • Pyridines
  • Pyrimidines
  • Receptor Protein-Tyrosine Kinases
  • Receptors, Platelet-Derived Growth Factor