Stimulation of membrane serine-threonine phosphatase in erythrocytes by hydrogen peroxide and staurosporine

Am J Physiol. 1998 Feb;274(2):C440-6. doi: 10.1152/ajpcell.1998.274.2.C440.

Abstract

Indirect evidence has suggested that K-Cl cotransport in human and sheep erythrocytes is activated physiologically by a serine-threonine phosphatase. It is activated experimentally by H2O2 and by staurosporine, a kinase inhibitor. Activation by H2O2 and staurosporine is inhibited by serine-threonine phosphatase inhibitors, suggesting that the activators stimulate the phosphatase. The present study shows that sheep and human erythrocytes contain membrane-associated as well as cytosolic serine-threonine phosphatases, assayed from the dephosphorylation of 32P-labeled glycogen phosphorylase. In cells from both species, the relatively low sensitivity of the membrane enzyme to okadaic acid suggests it is type 1 protein phosphatase. The cytosolic phosphatase was much more sensitive to okadaic acid. Membrane-associated phosphatase was stimulated by both H2O2 and staurosporine. The results support earlier conclusions that the membrane-associated type 1 phosphatase identified here is regulated by phosphorylation and oxidation. The results are consistent with the phosphatase, or a portion of it, being responsible for activating K-Cl cotransport.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Carrier Proteins / blood
  • Cytosol / drug effects
  • Cytosol / enzymology
  • Enzyme Activation
  • Enzyme Inhibitors / pharmacology
  • Erythrocyte Membrane / drug effects
  • Erythrocyte Membrane / enzymology
  • Erythrocytes / drug effects
  • Erythrocytes / enzymology*
  • Humans
  • Hydrogen Peroxide / pharmacology*
  • In Vitro Techniques
  • K Cl- Cotransporters
  • Okadaic Acid / pharmacology
  • Phosphoprotein Phosphatases / metabolism*
  • Sheep
  • Staurosporine / pharmacology*
  • Symporters*

Substances

  • Carrier Proteins
  • Enzyme Inhibitors
  • Symporters
  • Okadaic Acid
  • Hydrogen Peroxide
  • Phosphoprotein Phosphatases
  • Staurosporine