Pathological mutations of nicotinic receptors and nicotine-based therapies for brain disorders

Curr Opin Neurobiol. 1997 Oct;7(5):674-82. doi: 10.1016/s0959-4388(97)80088-8.

Abstract

Nicotinic acetylcholine receptors are allosteric ligand-gated ion channels present in muscle and brain. Recent studies suggest that mutations altering their functional properties may produce congenital myasthenia and familial frontal lobe epilepsy. Current research also indicates that although nicotinic ligands often possess addictive properties, they could serve as therapeutic agents for Alzheimer's disease and Tourette's syndrome, as well as for schizophrenia.

Publication types

  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Brain Diseases / drug therapy*
  • Brain Diseases / genetics
  • Cholinergic Agents / therapeutic use*
  • Humans
  • Molecular Sequence Data
  • Nicotine / therapeutic use*
  • Receptors, Nicotinic / drug effects
  • Receptors, Nicotinic / genetics*

Substances

  • Cholinergic Agents
  • Receptors, Nicotinic
  • Nicotine