Hormone-regulatable neoplastic transformation induced by a Jun-estrogen receptor chimera

Proc Natl Acad Sci U S A. 1997 Nov 11;94(23):12396-400. doi: 10.1073/pnas.94.23.12396.

Abstract

The v-jun oncogene encodes a nuclear DNA binding protein that functions as a transcription factor and is part of the activator protein 1 complex. Oncogenic transformation by v-jun is thought to be mediated by the aberrant expression of specific target genes. To identify such Jun-regulated genes and to explore the mechanisms by which Jun affects their expression, we have fused the full-length v-Jun and an amino-terminally truncated form of v-Jun to the hormone-binding domain of the human estrogen receptor. The two chimeric proteins function as ligand-inducible transactivators. Expression of the fusion proteins in chicken embryo fibroblasts causes estrogen-dependent transformation.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Cell Transformation, Neoplastic / genetics*
  • Cells, Cultured
  • Chick Embryo
  • Estrogens / pharmacology*
  • Fibroblasts / pathology
  • Gene Expression Regulation, Neoplastic / drug effects
  • Gene Targeting*
  • Genes, jun*
  • Humans
  • Receptors, Estrogen / genetics*
  • Receptors, Estrogen / metabolism
  • Recombinant Fusion Proteins / genetics*

Substances

  • Estrogens
  • Receptors, Estrogen
  • Recombinant Fusion Proteins